TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
City Of Hope National Medical Center
Curated by ChEMBL
City Of Hope National Medical Center
Curated by ChEMBL
Affinity DataEC50: 3.00E+3nMAssay Description:Agonist activity at PXR (unknown origin) expressed in human HepG2 cells assessed as induction of CYP3A4 transactivation after 16 hrs by luciferase re...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
City Of Hope National Medical Center
Curated by ChEMBL
City Of Hope National Medical Center
Curated by ChEMBL
Affinity DataEC50: 1.00E+4nMAssay Description:Competitive binding affinity to human PXR LBD (111 to 434) by TR-FRET assayMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
City Of Hope National Medical Center
Curated by ChEMBL
City Of Hope National Medical Center
Curated by ChEMBL
Affinity DataEC50: 1.00E+4nMAssay Description:Activation of human PXR expressed in human HepG2 (DPX-2) cells after 24 hrs by luciferase reporter gene based luminescent analysisMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
City Of Hope National Medical Center
Curated by ChEMBL
City Of Hope National Medical Center
Curated by ChEMBL
Affinity DataEC50: 1.26E+4nMAssay Description:Activation of rat PXR expressed in human HepG2 cells after 24 hrs by luciferase reporter gene based luminescent analysisMore data for this Ligand-Target Pair