Affinity DataEC50: 1nMAssay Description:In vitro intrinsic activity against histamine H3 receptor from synaptosomes of rat cerebral cortexMore data for this Ligand-Target Pair
Affinity DataEC50: 2.80nMAssay Description:In vitro binding affinity against histamine H3 receptor from synaptosomes of rat cerebral cortexMore data for this Ligand-Target Pair
Affinity DataEC50: 2.40nMAssay Description:Agonist activity at human recombinant histamine H3 receptor expressed in CHO cells assessed as [35S]GTPgammaS binding after 1 hr by liquid scintillat...More data for this Ligand-Target Pair
Affinity DataEC50: 12.6nMAssay Description:Agonist activity at human histamine H4 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 51nMAssay Description:Inhibition of human Histamine H4 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 1nMAssay Description:The compound was evaluated for agonistic effect on release of [3H]-histamine from rat brain cortical slices with L-[3H]-histidine at 0.3 microMMore data for this Ligand-Target Pair
Affinity DataEC50: 1.90nMAssay Description:Inhibition of human Histamine H3 receptor using [3H]-N-alpha-methyl histamineMore data for this Ligand-Target Pair