Compile Data Set for Download or QSAR
maximum 50k data
Found 80 of ki for monomerid = 26986
TargetCarbonic anhydrase 15 [19-324](Mus musculus (mouse))
Universita Degli Studi Di Firenze

LigandPNGBDBM26986(CHEMBL363707 | HCO3- | SODIUM BICARBONATE | bicarb...)
Affinity DataKi:  8.20E+3nMAssay Description:An Applied Photophysics stopped-flow instrument has been used for assaying the CA-catalyzed CO2 hydration activity. Phenol red has been used as indic...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM26986(CHEMBL363707 | HCO3- | SODIUM BICARBONATE | bicarb...)
Affinity DataKi:  8.60E+3nMAssay Description:Inhibitory activity against human Carbonic anhydrase IXMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 7(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM26986(CHEMBL363707 | HCO3- | SODIUM BICARBONATE | bicarb...)
Affinity DataKi:  2.70E+5nMAssay Description:Inhibition of human recombinant CA7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 7(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM26986(CHEMBL363707 | HCO3- | SODIUM BICARBONATE | bicarb...)
Affinity DataKi:  2.70E+5nMAssay Description:Inhibition of human recombinant CA7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase(Stylophora pistillata)
Centre Scientifique De Monaco

Curated by ChEMBL
LigandPNGBDBM26986(CHEMBL363707 | HCO3- | SODIUM BICARBONATE | bicarb...)
Affinity DataKi:  4.50E+5nMAssay Description:Inhibition of Stylophora pistillata carbonic anhydrase by stopped-flow CO2 hydration assayChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase(Helicobacter pylori)
Universit?? Degli Studi Di Firenze

LigandPNGBDBM26986(CHEMBL363707 | HCO3- | SODIUM BICARBONATE | bicarb...)
Affinity DataKi:  5.00E+5nM ΔG°:  -4.50kcal/molepH: 7.5 T: 2°CAssay Description:An Applied Photophysics stopped-flow instrument has been used for assaying the CA catalysed CO2 hydration activity Khalifah RG. The carbon dioxide hy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-carbonic anhydrase(Helicobacter pylori)
Universit?? Degli Studi Di Firenze

LigandPNGBDBM26986(CHEMBL363707 | HCO3- | SODIUM BICARBONATE | bicarb...)
Affinity DataKi:  7.50E+5nM ΔG°:  -4.26kcal/molepH: 7.5 T: 2°CAssay Description:An Applied Photophysics stopped-flow instrument has been used for assaying the CA catalysed CO2 hydration activity Khalifah RG. The carbon dioxide hy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-carbonic anhydrase(Helicobacter pylori (strain G27))
Universit£

LigandPNGBDBM26986(CHEMBL363707 | HCO3- | SODIUM BICARBONATE | bicarb...)
Affinity DataKi:  7.50E+5nM ΔG°:  -4.19kcal/molepH: 7.5 T: 2°CAssay Description:Inhibition of Vibrio cholerae alpha carbonic anhydrase preincubated for 15 mins by stopped-flow CO2 hydrase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 6(Homo sapiens (Human))
Centre Scientifique De Monaco

Curated by ChEMBL
LigandPNGBDBM26986(CHEMBL363707 | HCO3- | SODIUM BICARBONATE | bicarb...)
Affinity DataKi:  8.00E+5nMAssay Description:Inhibition of human recombinant CA6 by stopped-flow CO2 hydration assayChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma carbonic anhydrase family protein(Vibrio cholerae)
Universit£

LigandPNGBDBM26986(CHEMBL363707 | HCO3- | SODIUM BICARBONATE | bicarb...)
Affinity DataKi:  3.00E+6nM ΔG°:  -3.38kcal/molepH: 7.5 T: 2°CAssay Description:Inhibition of Vibrio cholerae recombinant carbonic anhydrase gamma expressed in Escherichia coli DE3 cells preincubated for 15 mins by stopped-flow C...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM26986(CHEMBL363707 | HCO3- | SODIUM BICARBONATE | bicarb...)
Affinity DataKi:  3.20E+6nMpH: 8.3Assay Description:Inhibition of Pseudomonas aeruginosa PAO1 type-2 beta-carbonic anhydrase psCA3 expressed in Escherichia coli Tuner BL21 (DE3) cells pre-incubated for...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase(Vibrio cholerae serotype O1 (strain ATCC 39315 / E...)
Universit£

LigandPNGBDBM26986(CHEMBL363707 | HCO3- | SODIUM BICARBONATE | bicarb...)
Affinity DataKi:  5.13E+6nM ΔG°:  -3.07kcal/molepH: 7.5 T: 2°CAssay Description:Inhibition of Flaveria bidentis carbonic anhydrase 1 preincubated for 15 mins by stopped-flow CO2 hydrase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 4(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM26986(CHEMBL363707 | HCO3- | SODIUM BICARBONATE | bicarb...)
Affinity DataKi:  5.70E+6nMAssay Description:Inhibitory activity against human Carbonic anhydrase IVMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase(Vibrio cholerae)
Universit£

LigandPNGBDBM26986(CHEMBL363707 | HCO3- | SODIUM BICARBONATE | bicarb...)
Affinity DataKi:  5.90E+6nM ΔG°:  -2.99kcal/molepH: 7.5 T: 2°CAssay Description:Inhibition of Vibrio cholerae carbonic anhydrase beta preincubated for 15 mins by stopped-flow CO2 hydrase assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 4(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM26986(CHEMBL363707 | HCO3- | SODIUM BICARBONATE | bicarb...)
Affinity DataKi:  6.60E+6nMAssay Description:Inhibition constant of anion against human carbonic anhydrase isozyme hCA IVMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 4(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM26986(CHEMBL363707 | HCO3- | SODIUM BICARBONATE | bicarb...)
Affinity DataKi:  6.60E+6nMAssay Description:Binding affinity against human cytosolic Carbonic anhydrase IVMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 4(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM26986(CHEMBL363707 | HCO3- | SODIUM BICARBONATE | bicarb...)
Affinity DataKi:  6.60E+6nMAssay Description:An Applied Photophysics stopped-flow instrument has been used for assaying the CA-catalyzed CO2 hydration activity. Phenol red has been used as indic...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 4(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM26986(CHEMBL363707 | HCO3- | SODIUM BICARBONATE | bicarb...)
Affinity DataKi:  6.60E+6nMAssay Description:Inhibition constant of anion against human carbonic anhydrase isozyme hCA IVMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 4(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM26986(CHEMBL363707 | HCO3- | SODIUM BICARBONATE | bicarb...)
Affinity DataKi:  6.60E+6nMAssay Description:Inhibition constant of anion against human carbonic anhydrase isozyme hCA IVMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase(Stylophora pistillata)
Centre Scientifique De Monaco

Curated by ChEMBL
LigandPNGBDBM26986(CHEMBL363707 | HCO3- | SODIUM BICARBONATE | bicarb...)
Affinity DataKi:  7.81E+6nMAssay Description:Inhibition of Stylophora pistillata carbonic anhydrase 2 by stopped-flow CO2 hydration assayChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Istituto Di Bioscienze E Biorisorse (Ibbr)-Cnr

Curated by ChEMBL
LigandPNGBDBM26986(CHEMBL363707 | HCO3- | SODIUM BICARBONATE | bicarb...)
Affinity DataKi:  1.20E+7nMAssay Description:Inhibition of human carbonic anhydrase 1 preincubated for 15 mins by stopped flow CO2 hydration methodMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Istituto Di Bioscienze E Biorisorse (Ibbr)-Cnr

Curated by ChEMBL
LigandPNGBDBM26986(CHEMBL363707 | HCO3- | SODIUM BICARBONATE | bicarb...)
Affinity DataKi:  1.20E+7nMAssay Description:Inhibition constant of anion against human carbonic anhydrase isozyme hCA IMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Istituto Di Bioscienze E Biorisorse (Ibbr)-Cnr

Curated by ChEMBL
LigandPNGBDBM26986(CHEMBL363707 | HCO3- | SODIUM BICARBONATE | bicarb...)
Affinity DataKi:  1.20E+7nMAssay Description:Binding affinity against human cytosolic Carbonic anhydrase IMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Istituto Di Bioscienze E Biorisorse (Ibbr)-Cnr

Curated by ChEMBL
LigandPNGBDBM26986(CHEMBL363707 | HCO3- | SODIUM BICARBONATE | bicarb...)
Affinity DataKi:  1.20E+7nMAssay Description:Inhibition of human recombinant CA1 by stopped-flow CO2 hydration assayChecked by AuthorMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Istituto Di Bioscienze E Biorisorse (Ibbr)-Cnr

Curated by ChEMBL
LigandPNGBDBM26986(CHEMBL363707 | HCO3- | SODIUM BICARBONATE | bicarb...)
Affinity DataKi:  1.20E+7nMAssay Description:Inhibition of human carbonic anhydrase 1 preincubated for 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Istituto Di Bioscienze E Biorisorse (Ibbr)-Cnr

Curated by ChEMBL
LigandPNGBDBM26986(CHEMBL363707 | HCO3- | SODIUM BICARBONATE | bicarb...)
Affinity DataKi:  1.20E+7nM ΔG°:  -2.57kcal/molepH: 7.5 T: 2°CAssay Description:An Applied Photophysics stopped-flow instrument has been used for assaying the CA-catalyzed CO2 hydration activity. Phenol red has been used as indic...More data for this Ligand-Target Pair
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Istituto Di Bioscienze E Biorisorse (Ibbr)-Cnr

Curated by ChEMBL
LigandPNGBDBM26986(CHEMBL363707 | HCO3- | SODIUM BICARBONATE | bicarb...)
Affinity DataKi:  1.20E+7nMpH: 7.5Assay Description:Inhibition of human carbonic anhydrase 1 after 15 mins by CO2 hydrase assay at pH 7.5More data for this Ligand-Target Pair
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Istituto Di Bioscienze E Biorisorse (Ibbr)-Cnr

Curated by ChEMBL
LigandPNGBDBM26986(CHEMBL363707 | HCO3- | SODIUM BICARBONATE | bicarb...)
Affinity DataKi:  1.20E+7nMpH: 8.3Assay Description:Inhibition of recombinant human carbonic anhydrase 1 after 15 mins by stopped flow CO2 hydration assay at pH 8.3More data for this Ligand-Target Pair
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Istituto Di Bioscienze E Biorisorse (Ibbr)-Cnr

Curated by ChEMBL
LigandPNGBDBM26986(CHEMBL363707 | HCO3- | SODIUM BICARBONATE | bicarb...)
Affinity DataKi:  1.20E+7nM ΔG°:  -2.57kcal/molepH: 7.5 T: 2°CAssay Description:Inhibition of human carbonic anhydrase 2 preincubated for 15 mins by stopped-flow CO2 hydrase assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Istituto Di Bioscienze E Biorisorse (Ibbr)-Cnr

Curated by ChEMBL
LigandPNGBDBM26986(CHEMBL363707 | HCO3- | SODIUM BICARBONATE | bicarb...)
Affinity DataKi:  1.20E+7nMAssay Description:Inhibitory constant against carbonic anhydrase IMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Istituto Di Bioscienze E Biorisorse (Ibbr)-Cnr

Curated by ChEMBL
LigandPNGBDBM26986(CHEMBL363707 | HCO3- | SODIUM BICARBONATE | bicarb...)
Affinity DataKi:  1.20E+7nMAssay Description:Inhibitory constant against carbonic anhydrase IMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Istituto Di Bioscienze E Biorisorse (Ibbr)-Cnr

Curated by ChEMBL
LigandPNGBDBM26986(CHEMBL363707 | HCO3- | SODIUM BICARBONATE | bicarb...)
Affinity DataKi:  1.20E+7nMAssay Description:Inhibitory activity against human carbonic anhydrase I expressed in Escherichia coliChecked by AuthorMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Istituto Di Bioscienze E Biorisorse (Ibbr)-Cnr

Curated by ChEMBL
LigandPNGBDBM26986(CHEMBL363707 | HCO3- | SODIUM BICARBONATE | bicarb...)
Affinity DataKi:  1.20E+7nMAssay Description:Inhibition of human recombinant wild type CA1 by stopped-flow CO2 hydration methodMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Istituto Di Bioscienze E Biorisorse (Ibbr)-Cnr

Curated by ChEMBL
LigandPNGBDBM26986(CHEMBL363707 | HCO3- | SODIUM BICARBONATE | bicarb...)
Affinity DataKi:  1.20E+7nMAssay Description:Inhibition constant of anion against human carbonic anhydrase isozyme hCA IMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Istituto Di Bioscienze E Biorisorse (Ibbr)-Cnr

Curated by ChEMBL
LigandPNGBDBM26986(CHEMBL363707 | HCO3- | SODIUM BICARBONATE | bicarb...)
Affinity DataKi:  1.20E+7nMAssay Description:Inhibition constant of anion against human carbonic anhydrase isozyme hCA IMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Istituto Di Bioscienze E Biorisorse (Ibbr)-Cnr

Curated by ChEMBL
LigandPNGBDBM26986(CHEMBL363707 | HCO3- | SODIUM BICARBONATE | bicarb...)
Affinity DataKi:  1.20E+7nMAssay Description:Inhibition of human cytosolic carbonic anhydrase 1 preincubated for 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Istituto Di Bioscienze E Biorisorse (Ibbr)-Cnr

Curated by ChEMBL
LigandPNGBDBM26986(CHEMBL363707 | HCO3- | SODIUM BICARBONATE | bicarb...)
Affinity DataKi:  1.20E+7nMAssay Description:Inhibition of human carbonic anhydrase-1 at 20 degC preincubated for 15 mins by stopped-flow CO2 hydrase assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM26986(CHEMBL363707 | HCO3- | SODIUM BICARBONATE | bicarb...)
Affinity DataKi:  1.30E+7nMAssay Description:Inhibition constant of anion against human carbonic anhydrase isozyme hCA IXMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM26986(CHEMBL363707 | HCO3- | SODIUM BICARBONATE | bicarb...)
Affinity DataKi:  1.30E+7nMAssay Description:Inhibition constant of anion against human carbonic anhydrase isozyme hCA IXMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM26986(CHEMBL363707 | HCO3- | SODIUM BICARBONATE | bicarb...)
Affinity DataKi:  1.30E+7nMAssay Description:Binding affinity against human cytosolic Carbonic anhydrase IXMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Istituto Di Bioscienze E Biorisorse (Ibbr)-Cnr

Curated by ChEMBL
LigandPNGBDBM26986(CHEMBL363707 | HCO3- | SODIUM BICARBONATE | bicarb...)
Affinity DataKi:  1.50E+7nMAssay Description:Inhibitory activity against human Carbonic anhydrase IMore data for this Ligand-Target Pair
TargetCarbonic anhydrase(Astrosclera willeyana)
Slovak Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM26986(CHEMBL363707 | HCO3- | SODIUM BICARBONATE | bicarb...)
Affinity DataKi:  2.28E+7nMAssay Description:Inhibition of Astrosclera willeyana recombinant GST-tagged astrosclerin 3 expressed in Escherichia coli BL21-DE3-RIPL cells preincubated for 15 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase(Methanosarcina thermophila)
Istituto Di Biochimica Delle Proteine-Cnr

Curated by ChEMBL
LigandPNGBDBM26986(CHEMBL363707 | HCO3- | SODIUM BICARBONATE | bicarb...)
Affinity DataKi:  4.20E+7nMAssay Description:Inhibition of Methanosarcina thermophila recombinant gamma-CA by CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase(Methanosarcina thermophila)
Istituto Di Biochimica Delle Proteine-Cnr

Curated by ChEMBL
LigandPNGBDBM26986(CHEMBL363707 | HCO3- | SODIUM BICARBONATE | bicarb...)
Affinity DataKi:  4.20E+7nMAssay Description:Inhibition of archaeon Methanosarcina thermophila gamma-CA after 15 mins by stopped-flow/Co2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase(Methanosarcina thermophila)
Istituto Di Biochimica Delle Proteine-Cnr

Curated by ChEMBL
LigandPNGBDBM26986(CHEMBL363707 | HCO3- | SODIUM BICARBONATE | bicarb...)
Affinity DataKi:  4.20E+7nMAssay Description:Inhibitory constant against Zn-Cam (Methanosarcina thermophila)More data for this Ligand-Target Pair
TargetCarbonic anhydrase(Methanosarcina thermophila)
Istituto Di Biochimica Delle Proteine-Cnr

Curated by ChEMBL
LigandPNGBDBM26986(CHEMBL363707 | HCO3- | SODIUM BICARBONATE | bicarb...)
Affinity DataKi:  4.20E+7nMAssay Description:Inhibitory constant against Zn-Cam (Methanosarcina thermophila)More data for this Ligand-Target Pair
TargetCarbonic anhydrase(Methanosarcina thermophila)
Istituto Di Biochimica Delle Proteine-Cnr

Curated by ChEMBL
LigandPNGBDBM26986(CHEMBL363707 | HCO3- | SODIUM BICARBONATE | bicarb...)
Affinity DataKi:  4.20E+7nMAssay Description:Inhibition of Methanosarcina thermophila recombinant carbonic anhydrase gamma assessed as inhibition of CO2 hydration preincubated for 15 mins by Lin...More data for this Ligand-Target Pair
TargetCarbonic anhydrase 4(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM26986(CHEMBL363707 | HCO3- | SODIUM BICARBONATE | bicarb...)
Affinity DataKi:  4.40E+7nMAssay Description:Inhibitory constant against carbonic anhydrase IVMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase(Methanobacterium thermoautotrophicum)
Universit£

Curated by ChEMBL
LigandPNGBDBM26986(CHEMBL363707 | HCO3- | SODIUM BICARBONATE | bicarb...)
Affinity DataKi:  4.49E+7nMAssay Description:Inhibitory constant against methanoarchaeon Methanobacterium thermoautotrophicum (Cab)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase(Methanobacterium thermoautotrophicum)
Universit£

Curated by ChEMBL
LigandPNGBDBM26986(CHEMBL363707 | HCO3- | SODIUM BICARBONATE | bicarb...)
Affinity DataKi:  4.49E+7nMAssay Description:Inhibitory constant against methanoarchaeon Methanobacterium thermoautotrophicum (Cab)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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