Compile Data Set for Download or QSAR
maximum 50k data
Found 21 of ic50 for monomerid = 50033376
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50033376(CHEMBL3357634)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of wild type EGFR (unknown origin) incubated for 5 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50033376(CHEMBL3357634)
Affinity DataIC50:  6.70nMAssay Description:Inhibition of wild type EGFR T790M mutant (unknown origin) incubated for 5 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-4(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50033376(CHEMBL3357634)
Affinity DataIC50:  23nMAssay Description:Inhibition of wild type HER4 (unknown origin) incubated for 5 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50033376(CHEMBL3357634)
Affinity DataIC50:  75nMAssay Description:Inhibition of wild type HER2 (unknown origin) incubated for 5 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50033376(CHEMBL3357634)
Affinity DataIC50:  1.73E+3nMAssay Description:Inhibition of wild type SRC (unknown origin) incubated for 5 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor beta(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50033376(CHEMBL3357634)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of wild type PDGFRbeta (unknown origin) incubated for 5 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50033376(CHEMBL3357634)
Affinity DataIC50:  2.26E+3nMAssay Description:Inhibition of wild type ABL (unknown origin) incubated for 5 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50033376(CHEMBL3357634)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibition of wild type PDGFRalpha (unknown origin) incubated for 5 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50033376(CHEMBL3357634)
Affinity DataIC50:  6.81E+3nMAssay Description:Inhibition of wild type FLT3 (unknown origin) incubated for 5 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50033376(CHEMBL3357634)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of wild type SYK (unknown origin) incubated for 5 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50033376(CHEMBL3357634)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of wild type JAK2 (unknown origin) incubated for 5 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50033376(CHEMBL3357634)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of wild type ALK (unknown origin) incubated for 5 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50033376(CHEMBL3357634)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of wild type AKT1 (unknown origin) incubated for 5 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50033376(CHEMBL3357634)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of wild type AKT2 (unknown origin) incubated for 5 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50033376(CHEMBL3357634)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of wild type c-Met (unknown origin) incubated for 5 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFibroblast growth factor receptor 2(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50033376(CHEMBL3357634)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of wild type FGFR2 (unknown origin) incubated for 5 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50033376(CHEMBL3357634)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP3A4 in human hepatic microsomes after 20 mins by LC/MS/MS methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50033376(CHEMBL3357634)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP2D6 in human hepatic microsomes after 20 mins by LC/MS/MS methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50033376(CHEMBL3357634)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP2C9 in human hepatic microsomes after 20 mins by LC/MS/MS methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C19(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50033376(CHEMBL3357634)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP2C19 in human hepatic microsomes after 20 mins by LC/MS/MS methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50033376(CHEMBL3357634)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP1A2 in human hepatic microsomes after 20 mins by LC/MS/MS methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed