Found 28 of ec50 for monomerid = 50119368 
Affinity DataEC50: 1.40E+3nMAssay Description:In vitro cAMP accumulation in HEK cells transfected with human Melanocortin 3 receptor (hMC3R)More data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Nanyang Technological University
Curated by ChEMBL
Nanyang Technological University
Curated by ChEMBL
Affinity DataEC50: 5nMAssay Description:Displacement of europium labeled NDP-alpha-MSH from human MC1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 1.33E+3nMAssay Description:Functional activity as concentration of the compound at 50% maximum cAMP accumulation in rat Melanocortin-3 receptor (rMC3R)More data for this Ligand-Target Pair
Affinity DataEC50: 2.10nMAssay Description:Functional activity as concentration of the compound at 50% maximum cAMP accumulation in human Melanocortin-4 receptorMore data for this Ligand-Target Pair
3D Structure (crystal)Affinity DataEC50: 2.10nMAssay Description:Evaluated for Functional Activity at Melanocortin-4 receptor as effective concentration at 50% maximum CMP accumulationMore data for this Ligand-Target Pair
Affinity DataEC50: 2.49E+3nMAssay Description:Evaluated for Functional Activity at MC3R as effective concentration at 50% maximum CMP accumulationMore data for this Ligand-Target Pair
Affinity DataEC50: 2.49E+3nMAssay Description:Functional activity as concentration of the compound at 50% maximum cAMP accumulation in human melanocortin 1 (MC3R) receptorMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Nanyang Technological University
Curated by ChEMBL
Nanyang Technological University
Curated by ChEMBL
Affinity DataEC50: 2.85E+3nMAssay Description:Functional activity as concentration at 50% maximum cAMP accumulation in human melanocortin 1 (MC1R) receptorMore data for this Ligand-Target Pair
Affinity DataEC50: >3.00E+3nMAssay Description:Functional activity as concentration of the compound at 50% maximum cAMP accumulation in rat Melanocortin-5 receptor (rMC5R)More data for this Ligand-Target Pair
Affinity DataEC50: 736nMAssay Description:Evaluated for Functional Activity at MC5R as effective concentration at 50% maximum CMP accumulationMore data for this Ligand-Target Pair
Affinity DataEC50: 737nMAssay Description:Functional activity as concentration at 50% maximum cAMP accumulation in human melanocortin 1 (MC5R) receptorMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Nanyang Technological University
Curated by ChEMBL
Nanyang Technological University
Curated by ChEMBL
Affinity DataEC50: 2.85E+3nMAssay Description:Activity against human MC1BR by cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataEC50: 2.49E+3nMAssay Description:Activity against human MC3R by cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataEC50: 2.10nMAssay Description:Activity against human MC4R by cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataEC50: 2.10nMAssay Description:Agonist activity at human MC4 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 1nMAssay Description:Agonist activity at human MC4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 160nMAssay Description:Agonist activity at human MC3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 2.90nMAssay Description:Functional activity as concentration of the compound at 50% maximum cAMP accumulation in rat Melanocortin-4 receptor (rMC4R)More data for this Ligand-Target Pair
Affinity DataEC50: 3.60nMAssay Description:Stimulation of adenylate cyclase in HEK293 cells expressing the human MC4R receptor was determined by measuring cAMP accumulation using the RPA559 SP...More data for this Ligand-Target Pair
Affinity DataEC50: 5.70nMAssay Description:Effective concentration against cAMP release in CHO cells expressing human melanocortin-4 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 49nMAssay Description:Agonist activity at human MC4 D122A mutant expressed in HEK293 cells assessed as stimulation of cAMP productionMore data for this Ligand-Target Pair
Affinity DataEC50: 737nMAssay Description:Activity against human MC5R by cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:In vitro cAMP accumulation in Y1 cells transfected with mouse Melanocortin 2 receptor (mMC2R)More data for this Ligand-Target Pair
Affinity DataEC50: 2.70E+3nMAssay Description:In vitro cAMP accumulation in HEK cells transfected with human Melanocortin 5 receptor (hMC5R)More data for this Ligand-Target Pair
Affinity DataEC50: 4nMAssay Description:Agonistic activity measured as inhibition of cAMP accumulation in HEK cells expressing human Melanocortin 4 receptor (hMC4R)More data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Nanyang Technological University
Curated by ChEMBL
Nanyang Technological University
Curated by ChEMBL
Affinity DataEC50: 1.40E+3nMAssay Description:In vitro cAMP accumulation in HEK cells transfected with human Melanocortin 1 receptor (hMC1R)More data for this Ligand-Target Pair
Affinity DataEC50: 7.60nMAssay Description:In vitro cAMP accumulation in Y1 cells transfected with mouse Melanocortin 4 receptor (mMC4R)More data for this Ligand-Target Pair
Affinity DataEC50: 1.5nMAssay Description:Agonist activity at human MC4 receptor expressed in HEK293 cells assessed as stimulation of cAMP productionMore data for this Ligand-Target Pair
