TargetGlutamate receptor 1(Mus musculus)
The Danish University Of Pharmaceutical Sciences
Curated by ChEMBL
The Danish University Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 4.70E+3nMAssay Description:Effective concentration of compound was determined for electrophysiological properties on Ionotropic glutamate receptor AMPA 1 (GluR1) using rat cort...More data for this Ligand-Target Pair
TargetGlutamate receptor 2(Rattus norvegicus)
The Danish University Of Pharmaceutical Sciences
Curated by ChEMBL
The Danish University Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 1.70E+3nMAssay Description:Effective concentration of compound was determined for electrophysiological properties on Ionotropic glutamate receptor AMPA 2 (GluR2) using rat cort...More data for this Ligand-Target Pair
TargetGlutamate receptor 4(Rattus norvegicus)
The Danish University Of Pharmaceutical Sciences
Curated by ChEMBL
The Danish University Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 1.30E+6nMAssay Description:Effective concentration of compound was determined for electrophysiological properties on Ionotropic glutamate receptor AMPA 4 (GluR4) using rat cort...More data for this Ligand-Target Pair
Affinity DataEC50: 2.70E+6nMAssay Description:Effective concentration of compound was determined for electrophysiological properties on Ionotropic glutamate receptor AMPA 3 (GluR3) using rat cort...More data for this Ligand-Target Pair
Affinity DataEC50: 4.70E+3nMAssay Description:Agonist activity at recombinant GluA1 receptor flip isoform expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataEC50: 1.70E+3nMAssay Description:Agonist activity at recombinant GluA2 receptor flop isoform expressed in Xenopus oocytesMore data for this Ligand-Target Pair
TargetGlutamate receptor 4(Rattus norvegicus)
The Danish University Of Pharmaceutical Sciences
Curated by ChEMBL
The Danish University Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 1.30E+6nMAssay Description:Agonist activity at rat recombinant GluA4i expressed in Xenopus laevis oocytes by two-electrode voltage clamp assayMore data for this Ligand-Target Pair
Affinity DataEC50: 4.10E+3nMAssay Description:Agonist activity at GluA1 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 1.70E+3nMAssay Description:Agonist activity at GluA2 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 2.70E+6nMAssay Description:Agonist activity at GluA3 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 4.70E+3nMAssay Description:Agonist activity at rat recombinant GluA1i expressed in Xenopus laevis oocytes by two-electrode voltage clamp assayMore data for this Ligand-Target Pair
TargetGlutamate receptor 2(Rattus norvegicus)
The Danish University Of Pharmaceutical Sciences
Curated by ChEMBL
The Danish University Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 1.70E+3nMAssay Description:Agonist activity at rat recombinant GluA2(Q)i expressed in Xenopus laevis oocytes by two-electrode voltage clamp assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.70E+6nMAssay Description:Agonist activity at rat recombinant GluA3i expressed in Xenopus laevis oocytes by two-electrode voltage clamp assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.70E+6nMAssay Description:Agonist activity at recombinant GluA3 receptor flip isoform expressed in Xenopus oocytesMore data for this Ligand-Target Pair