Compile Data Set for Download or QSAR
maximum 50k data
Found 27 of ic50 for monomerid = 50263132
TargetProtein kinase C theta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263132(4-(4-methyl-1H-indol-5-ylamino)-2-(3-oxo-3-(pyrrol...)
Affinity DataIC50:  3.80nMAssay Description:Inhibition of PKCthetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Fyn(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263132(4-(4-methyl-1H-indol-5-ylamino)-2-(3-oxo-3-(pyrrol...)
Affinity DataIC50:  25nMAssay Description:Inhibition of FYNMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase HCK(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263132(4-(4-methyl-1H-indol-5-ylamino)-2-(3-oxo-3-(pyrrol...)
Affinity DataIC50:  26nMAssay Description:Inhibition of HCKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263132(4-(4-methyl-1H-indol-5-ylamino)-2-(3-oxo-3-(pyrrol...)
Affinity DataIC50:  28nMAssay Description:Inhibition of LYNMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263132(4-(4-methyl-1H-indol-5-ylamino)-2-(3-oxo-3-(pyrrol...)
Affinity DataIC50:  46nMAssay Description:Inhibition of LCKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263132(4-(4-methyl-1H-indol-5-ylamino)-2-(3-oxo-3-(pyrrol...)
Affinity DataIC50:  330nMAssay Description:Inhibition of SRCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263132(4-(4-methyl-1H-indol-5-ylamino)-2-(3-oxo-3-(pyrrol...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of PKCdeltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263132(4-(4-methyl-1H-indol-5-ylamino)-2-(3-oxo-3-(pyrrol...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of PKCepsilonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263132(4-(4-methyl-1H-indol-5-ylamino)-2-(3-oxo-3-(pyrrol...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of ITKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263132(4-(4-methyl-1H-indol-5-ylamino)-2-(3-oxo-3-(pyrrol...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of METMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263132(4-(4-methyl-1H-indol-5-ylamino)-2-(3-oxo-3-(pyrrol...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of PDGFRalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263132(4-(4-methyl-1H-indol-5-ylamino)-2-(3-oxo-3-(pyrrol...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Aurora BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263132(4-(4-methyl-1H-indol-5-ylamino)-2-(3-oxo-3-(pyrrol...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CHK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263132(4-(4-methyl-1H-indol-5-ylamino)-2-(3-oxo-3-(pyrrol...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of PKCalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit alpha(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263132(4-(4-methyl-1H-indol-5-ylamino)-2-(3-oxo-3-(pyrrol...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of IKKalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263132(4-(4-methyl-1H-indol-5-ylamino)-2-(3-oxo-3-(pyrrol...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of IKK-betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRho-associated protein kinase 1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263132(4-(4-methyl-1H-indol-5-ylamino)-2-(3-oxo-3-(pyrrol...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of ROCK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform gamma-1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263132(4-(4-methyl-1H-indol-5-ylamino)-2-(3-oxo-3-(pyrrol...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CK1gamma1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263132(4-(4-methyl-1H-indol-5-ylamino)-2-(3-oxo-3-(pyrrol...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of ERK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263132(4-(4-methyl-1H-indol-5-ylamino)-2-(3-oxo-3-(pyrrol...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of VEGFR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosomal protein S6 kinase alpha-1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263132(4-(4-methyl-1H-indol-5-ylamino)-2-(3-oxo-3-(pyrrol...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of RSK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263132(4-(4-methyl-1H-indol-5-ylamino)-2-(3-oxo-3-(pyrrol...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of P38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMAP kinase-activated protein kinase 2(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263132(4-(4-methyl-1H-indol-5-ylamino)-2-(3-oxo-3-(pyrrol...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of MK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263132(4-(4-methyl-1H-indol-5-ylamino)-2-(3-oxo-3-(pyrrol...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CDK1/cyclinBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C eta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263132(4-(4-methyl-1H-indol-5-ylamino)-2-(3-oxo-3-(pyrrol...)
Affinity DataIC50:  5.10E+4nMAssay Description:Inhibition of PKCetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C beta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263132(4-(4-methyl-1H-indol-5-ylamino)-2-(3-oxo-3-(pyrrol...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of PKCbetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263132(4-(4-methyl-1H-indol-5-ylamino)-2-(3-oxo-3-(pyrrol...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of PKCzetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed