TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Medical University Of South Carolina
Curated by ChEMBL
Medical University Of South Carolina
Curated by ChEMBL
Affinity DataKd: 501nMAssay Description:Binding affinity to beta-2 adrenergic receptor (unknown origin) at 1 to 10000 nMMore data for this Ligand-Target Pair
Affinity DataKd: 4.27E+3nMAssay Description:Affinity for cow beta-2 adrenergic receptor by measuring displacement (-)-[3H]dihydroalprenolol (DHA)More data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Medical University Of South Carolina
Curated by ChEMBL
Medical University Of South Carolina
Curated by ChEMBL
Affinity DataKd: 4.81E+3nMAssay Description:Binding affinity to human adrenergic beta2 receptorMore data for this Ligand-Target Pair
Affinity DataKd: 9.12E+3nMAssay Description:Affinity for cow beta-2 adrenergic receptor by measuring displacement (-)-[3H]dihydroalprenolol (DHA)More data for this Ligand-Target Pair
TargetBeta-adrenergic receptor kinase 1(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories
Merck Sharp And Dohme Research Laboratories
Affinity DataKd: 1.30E+4nMAssay Description:The binding of ligands to wild-type beta-AR was measured by competition with 35 pM 125I-CYP.More data for this Ligand-Target Pair