TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
BMSSI UMR 5086 CNRS/Universit£ Lyon 1
Curated by ChEMBL
BMSSI UMR 5086 CNRS/Universit£ Lyon 1
Curated by ChEMBL
Affinity DataEC50: 29nMAssay Description:Inhibition of ABCG2 (unknown origin) transfected in HEK293 cells assessed as inhibition of mitoxantrone efflux after 30 mins by flow cytometry relati...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
BMSSI UMR 5086 CNRS/Universit£ Lyon 1
Curated by ChEMBL
BMSSI UMR 5086 CNRS/Universit£ Lyon 1
Curated by ChEMBL
Affinity DataEC50: 90nMAssay Description:Inhibition of ABCG2 (unknown origin) in HEK293 cells assessed as maximal inhibition of mitoxantrone efflux by fluorescence based flow cytometryMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
BMSSI UMR 5086 CNRS/Universit£ Lyon 1
Curated by ChEMBL
BMSSI UMR 5086 CNRS/Universit£ Lyon 1
Curated by ChEMBL
Affinity DataEC50: 74nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in HEK293 cells assessed as reduction in mitoxantrone efflux after 30 mins by flow cytometric analysisMore data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Hong Kong Polytechnic University
Curated by ChEMBL
Hong Kong Polytechnic University
Curated by ChEMBL
Affinity DataEC50: 1.95E+3nMAssay Description:Inhibition of MRP1 (unknown origin) expressed in human 2008/MRP1 assessed as reversal of doxorubicin resistance after 5 days by MTS/PMS assayMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Hong Kong Polytechnic University
Curated by ChEMBL
Hong Kong Polytechnic University
Curated by ChEMBL
Affinity DataEC50: 943nMAssay Description:Inhibition of P-gp (unknown origin) expressed in human LCC6MDR cells assessed as potentiation of mitoxantrone-induced cytotoxicity after 5 days by MT...More data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Hong Kong Polytechnic University
Curated by ChEMBL
Hong Kong Polytechnic University
Curated by ChEMBL
Affinity DataEC50: 1.80E+3nMAssay Description:Inhibition of MRP1 (unknown origin) expressed in human 2008/MRP1 cells assessed as potentiation of mitoxantrone-induced cytotoxicity after 5 days by ...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
BMSSI UMR 5086 CNRS/Universit£ Lyon 1
Curated by ChEMBL
BMSSI UMR 5086 CNRS/Universit£ Lyon 1
Curated by ChEMBL
Affinity DataEC50: 10nMAssay Description:Inhibition of BCRP (unknown origin)More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
BMSSI UMR 5086 CNRS/Universit£ Lyon 1
Curated by ChEMBL
BMSSI UMR 5086 CNRS/Universit£ Lyon 1
Curated by ChEMBL
Affinity DataEC50: 8.70nMAssay Description:Inhibition of BCRP (unknown origin) transfected in HEK293/R2 cells assessed as reversal of topotecan resistance after 5 days by MTS/PMS assayMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
BMSSI UMR 5086 CNRS/Universit£ Lyon 1
Curated by ChEMBL
BMSSI UMR 5086 CNRS/Universit£ Lyon 1
Curated by ChEMBL
Affinity DataEC50: 9nMAssay Description:Inhibition of BCRP in human MCF7/MX100 cells assessed as reversal of topotecan resistance after 5 days by MTS/PMS assayMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Hong Kong Polytechnic University
Curated by ChEMBL
Hong Kong Polytechnic University
Curated by ChEMBL
Affinity DataEC50: 1.06E+3nMAssay Description:Inhibition of P-gp (unknown origin) expressed in human LCC6MDR cells assessed as reversal of paclitaxel resistance after 5 days by MTS/PMS assayMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
BMSSI UMR 5086 CNRS/Universit£ Lyon 1
Curated by ChEMBL
BMSSI UMR 5086 CNRS/Universit£ Lyon 1
Curated by ChEMBL
Affinity DataEC50: 5.40nMAssay Description:Inhibition of BCRP (unknown origin) expressed in human HEK293/R2 cells assessed as potentiation of mitoxantrone-induced cytotoxicity after 5 days by ...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
BMSSI UMR 5086 CNRS/Universit£ Lyon 1
Curated by ChEMBL
BMSSI UMR 5086 CNRS/Universit£ Lyon 1
Curated by ChEMBL
Affinity DataEC50: 70nMAssay Description:Inhibition of ABCG2-mediated mitoxantrone efflux in mitoxantrone-selected human H460 cells after 30 mins by flow cytometric analysisMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
BMSSI UMR 5086 CNRS/Universit£ Lyon 1
Curated by ChEMBL
BMSSI UMR 5086 CNRS/Universit£ Lyon 1
Curated by ChEMBL
Affinity DataEC50: 90nMAssay Description:Inhibition of ABCG2 (unknown origin)-mediated mitoxantrone efflux expressed in HEK293 cells after 30 mins by flow cytometric analysisMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Hong Kong Polytechnic University
Curated by ChEMBL
Hong Kong Polytechnic University
Curated by ChEMBL
Affinity DataEC50: 70nMAssay Description:Activation of ABCB1 ATPase activity (unknown origin) expressed in baculovirus infected Sf9 insect cells using ATP as substrate measured after 1 hr by...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
BMSSI UMR 5086 CNRS/Universit£ Lyon 1
Curated by ChEMBL
BMSSI UMR 5086 CNRS/Universit£ Lyon 1
Curated by ChEMBL
Affinity DataEC50: 12nMAssay Description:Inhibition of ABCG2 (unknown origin) transfected in HEK293 cells assessed as inhibition of mitoxantrone efflux at 5 uM after 30 mins in presence of 0...More data for this Ligand-Target Pair