Compile Data Set for Download or QSAR
maximum 50k data
Found 38 of ic50 for monomerid = 50335374
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335374((3S,9S)-9,16-dihydroxy-14-methoxy-3-methyl-3,4,9,1...)
Affinity DataIC50:  5.80nMAssay Description:Inhibition of VEGFR2 by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335374((3S,9S)-9,16-dihydroxy-14-methoxy-3-methyl-3,4,9,1...)
Affinity DataIC50:  150nMAssay Description:Inhibition of MNK2 by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335374((3S,9S)-9,16-dihydroxy-14-methoxy-3-methyl-3,4,9,1...)
Affinity DataIC50:  190nMAssay Description:Inhibition of VEGFR2 by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335374((3S,9S)-9,16-dihydroxy-14-methoxy-3-methyl-3,4,9,1...)
Affinity DataIC50:  673nMAssay Description:Inhibition of cKIT by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335374((3S,9S)-9,16-dihydroxy-14-methoxy-3-methyl-3,4,9,1...)
Affinity DataIC50:  763nMAssay Description:Inhibition of ALK by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335374((3S,9S)-9,16-dihydroxy-14-methoxy-3-methyl-3,4,9,1...)
Affinity DataIC50:  4.40E+3nMAssay Description:Inhibition of TYK2 by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335374((3S,9S)-9,16-dihydroxy-14-methoxy-3-methyl-3,4,9,1...)
Affinity DataIC50:  4.70E+3nMAssay Description:Inhibition of LCK by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335374((3S,9S)-9,16-dihydroxy-14-methoxy-3-methyl-3,4,9,1...)
Affinity DataIC50:  6.40E+3nMAssay Description:Inhibition of ERK2 by Caliper mobility shift assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335374((3S,9S)-9,16-dihydroxy-14-methoxy-3-methyl-3,4,9,1...)
Affinity DataIC50:  7.20E+3nMAssay Description:Inhibition of RET by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335374((3S,9S)-9,16-dihydroxy-14-methoxy-3-methyl-3,4,9,1...)
Affinity DataIC50:  7.40E+3nMAssay Description:Inhibition of EPHB4 by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335374((3S,9S)-9,16-dihydroxy-14-methoxy-3-methyl-3,4,9,1...)
Affinity DataIC50:  7.60E+3nMAssay Description:Inhibition of cKIT by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335374((3S,9S)-9,16-dihydroxy-14-methoxy-3-methyl-3,4,9,1...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CDK2A by Caliper mobility shift assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ZAP-70(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335374((3S,9S)-9,16-dihydroxy-14-methoxy-3-methyl-3,4,9,1...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of ZAP70 by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-A receptor 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335374((3S,9S)-9,16-dihydroxy-14-methoxy-3-methyl-3,4,9,1...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of EPHA4 by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335374((3S,9S)-9,16-dihydroxy-14-methoxy-3-methyl-3,4,9,1...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of FGFR3 by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335374((3S,9S)-9,16-dihydroxy-14-methoxy-3-methyl-3,4,9,1...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GSK3-beta by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335374((3S,9S)-9,16-dihydroxy-14-methoxy-3-methyl-3,4,9,1...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of HER2 by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335374((3S,9S)-9,16-dihydroxy-14-methoxy-3-methyl-3,4,9,1...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of HGFR by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335374((3S,9S)-9,16-dihydroxy-14-methoxy-3-methyl-3,4,9,1...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of IGF1R by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335374((3S,9S)-9,16-dihydroxy-14-methoxy-3-methyl-3,4,9,1...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of JAK1 by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335374((3S,9S)-9,16-dihydroxy-14-methoxy-3-methyl-3,4,9,1...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of JAK2 by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335374((3S,9S)-9,16-dihydroxy-14-methoxy-3-methyl-3,4,9,1...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of JAK3 by Caliper mobility shift assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50335374((3S,9S)-9,16-dihydroxy-14-methoxy-3-methyl-3,4,9,1...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of PDK1 by Caliper mobility shift assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase catalytic subunit alpha(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335374((3S,9S)-9,16-dihydroxy-14-methoxy-3-methyl-3,4,9,1...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of PKAalpha by Caliper mobility shift assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335374((3S,9S)-9,16-dihydroxy-14-methoxy-3-methyl-3,4,9,1...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of PKN1 by Caliper mobility shift assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335374((3S,9S)-9,16-dihydroxy-14-methoxy-3-methyl-3,4,9,1...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of PKN2 by Caliper mobility shift assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335374((3S,9S)-9,16-dihydroxy-14-methoxy-3-methyl-3,4,9,1...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of BTK by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335374((3S,9S)-9,16-dihydroxy-14-methoxy-3-methyl-3,4,9,1...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Axl by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335374((3S,9S)-9,16-dihydroxy-14-methoxy-3-methyl-3,4,9,1...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Aurora A kinase by Caliper mobility shift assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335374((3S,9S)-9,16-dihydroxy-14-methoxy-3-methyl-3,4,9,1...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of RET by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335374((3S,9S)-9,16-dihydroxy-14-methoxy-3-methyl-3,4,9,1...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of EPHB4 by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335374((3S,9S)-9,16-dihydroxy-14-methoxy-3-methyl-3,4,9,1...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of ERK2 by Caliper mobility shift assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335374((3S,9S)-9,16-dihydroxy-14-methoxy-3-methyl-3,4,9,1...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of ALK by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRho-associated protein kinase 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335374((3S,9S)-9,16-dihydroxy-14-methoxy-3-methyl-3,4,9,1...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of ROCK2 by Caliper mobility shift assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335374((3S,9S)-9,16-dihydroxy-14-methoxy-3-methyl-3,4,9,1...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of INSR by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335374((3S,9S)-9,16-dihydroxy-14-methoxy-3-methyl-3,4,9,1...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of TYK2 by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335374((3S,9S)-9,16-dihydroxy-14-methoxy-3-methyl-3,4,9,1...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of p38alpha by Caliper mobility shift assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335374((3S,9S)-9,16-dihydroxy-14-methoxy-3-methyl-3,4,9,1...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of LCK by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed