Affinity DataKd: <3.02E+4nMAssay Description:Binding affinity to human partial length DNA-tagged SMARCA4 expressed in bacteria by BROMOscan methodMore data for this Ligand-Target Pair
Affinity DataKd: 63nMAssay Description:Inhibition of BRD4-BD2 (unknown origin) (K333 to E460 residues) expressed in bacterial system assessed as dissociation constant by BROMOscan methodMore data for this Ligand-Target Pair
TargetHistone acetyltransferase KAT2B(Homo sapiens (Human))
University Of Strathclyde
Curated by ChEMBL
University Of Strathclyde
Curated by ChEMBL
Affinity DataKd: <3.02E+4nMAssay Description:Binding affinity to human partial length DNA-tagged PCAF expressed in mammalian expression system by BROMOscan methodMore data for this Ligand-Target Pair
TargetBromodomain and PHD finger-containing protein 3(Homo sapiens (Human))
University Of Strathclyde
Curated by ChEMBL
University Of Strathclyde
Curated by ChEMBL
Affinity DataKd: <3.02E+4nMAssay Description:Binding affinity to human partial length DNA-tagged BRPF3 expressed in bacteria by BROMOscan methodMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 3(Homo sapiens (Human))
University Of Strathclyde
Curated by ChEMBL
University Of Strathclyde
Curated by ChEMBL
Affinity DataKd: 912nMAssay Description:Binding affinity to human partial length DNA-tagged BRD3 BD1 expressed in bacterial by BROMOscan methodMore data for this Ligand-Target Pair
TargetTranscription initiation factor TFIID subunit 1(Homo sapiens (Human))
University Of Strathclyde
Curated by ChEMBL
University Of Strathclyde
Curated by ChEMBL
Affinity DataKd: 1.45E+4nMAssay Description:Binding affinity to human partial length DNA-tagged TAF1 BD2 expressed in bacterial by BROMOscan methodMore data for this Ligand-Target Pair
TargetATPase family AAA domain-containing protein 2(Homo sapiens (Human))
University Of Strathclyde
Curated by ChEMBL
University Of Strathclyde
Curated by ChEMBL
Affinity DataKd: <3.02E+4nMAssay Description:Binding affinity to human partial length DNA-tagged ATAD2B expressed in bacterial by BROMOscan methodMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 8(Homo sapiens (Human))
University Of Strathclyde
Curated by ChEMBL
University Of Strathclyde
Curated by ChEMBL
Affinity DataKd: <3.02E+4nMAssay Description:Binding affinity to DNA-tagged BRD8 (unknown origin) by BROMOscan methodMore data for this Ligand-Target Pair
Affinity DataKd: <3.02E+4nMAssay Description:Binding affinity to human partial length DNA-tagged CREBBP expressed in bacteria by BROMOscan methodMore data for this Ligand-Target Pair
Affinity DataKd: <3.02E+4nMAssay Description:Binding affinity to human partial length DNA-tagged PBRM1 BD1 expressed in bacteria by BROMOscan methodMore data for this Ligand-Target Pair
TargetBromodomain testis-specific protein(Homo sapiens (Human))
University Of Strathclyde
Curated by ChEMBL
University Of Strathclyde
Curated by ChEMBL
Affinity DataKd: 21nMAssay Description:Binding affinity to human partial length DNA-tagged BRDT isoform b BD2 expressed in bacterial by BROMOscan methodMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 7(Homo sapiens (Human))
University Of Strathclyde
Curated by ChEMBL
University Of Strathclyde
Curated by ChEMBL
Affinity DataKd: <3.02E+4nMAssay Description:Binding affinity to human partial length DNA-tagged BRD7 expressed in mammalian expression system by BROMOscan methodMore data for this Ligand-Target Pair
Affinity DataKd: 6.60nMAssay Description:Binding affinity to human partial length DNA-tagged BRD4 isoform long BD2 expressed in bacterial by BROMOscan methodMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 2(Homo sapiens (Human))
University Of Strathclyde
Curated by ChEMBL
University Of Strathclyde
Curated by ChEMBL
Affinity DataKd: 32nMAssay Description:Binding affinity to human partial length DNA-tagged BRD2 isoform 1 BD2 expressed in bacterial by BROMOscan methodMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 3(Homo sapiens (Human))
University Of Strathclyde
Curated by ChEMBL
University Of Strathclyde
Curated by ChEMBL
Affinity DataKd: 19nMAssay Description:Binding affinity to human partial length DNA-tagged BRD3 BD2 expressed in bacterial by BROMOscan methodMore data for this Ligand-Target Pair
TargetBromodomain and WD repeat-containing protein 1(Homo sapiens (Human))
University Of Strathclyde
Curated by ChEMBL
University Of Strathclyde
Curated by ChEMBL
Affinity DataKd: 1.51E+4nMAssay Description:Binding affinity to human partial length DNA-tagged WRD9 BD2 expressed in bacterial by BROMOscan methodMore data for this Ligand-Target Pair
TargetATPase family AAA domain-containing protein 2(Homo sapiens (Human))
University Of Strathclyde
Curated by ChEMBL
University Of Strathclyde
Curated by ChEMBL
Affinity DataKd: <3.02E+4nMAssay Description:Binding affinity to human partial length DNA-tagged ATAD2A expressed in bacterial by BROMOscan methodMore data for this Ligand-Target Pair
TargetBromodomain adjacent to zinc finger domain protein 2A(Homo sapiens (Human))
University Of Strathclyde
Curated by ChEMBL
University Of Strathclyde
Curated by ChEMBL
Affinity DataKd: <3.02E+4nMAssay Description:Binding affinity to human partial length DNA-tagged BAZ2A expressed in bacterial by BROMOscan methodMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 1(Homo sapiens (Human))
University Of Strathclyde
Curated by ChEMBL
University Of Strathclyde
Curated by ChEMBL
Affinity DataKd: <3.02E+4nMAssay Description:Binding affinity to human partial length DNA-tagged BRD1 expressed in bacterial by BROMOscan methodMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 9(Homo sapiens (Human))
University Of Strathclyde
Curated by ChEMBL
University Of Strathclyde
Curated by ChEMBL
Affinity DataKd: <3.02E+4nMAssay Description:Binding affinity to human partial length DNA-tagged BRD9 isoform 1 expressed in bacteria by BROMOscan methodMore data for this Ligand-Target Pair
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
University Of Strathclyde
Curated by ChEMBL
University Of Strathclyde
Curated by ChEMBL
Affinity DataKd: <3.02E+4nMAssay Description:Binding affinity to human partial length DNA-tagged CECR2 expressed in bacteria by BROMOscan methodMore data for this Ligand-Target Pair
TargetHistone acetyltransferase p300(Homo sapiens (Human))
University Of Strathclyde
Curated by ChEMBL
University Of Strathclyde
Curated by ChEMBL
Affinity DataKd: <3.02E+4nMAssay Description:Binding affinity to human partial length DNA-tagged EP300 expressed in bacteria by BROMOscan methodMore data for this Ligand-Target Pair
TargetHistone acetyltransferase KAT2A(Homo sapiens (Human))
University Of Strathclyde
Curated by ChEMBL
University Of Strathclyde
Curated by ChEMBL
Affinity DataKd: <3.02E+4nMAssay Description:Binding affinity to human partial length DNA-tagged GCN5L2 expressed in bacteria by BROMOscan methodMore data for this Ligand-Target Pair
TargetProbable global transcription activator SNF2L2(Homo sapiens (Human))
University Of Strathclyde
Curated by ChEMBL
University Of Strathclyde
Curated by ChEMBL
Affinity DataKd: <3.02E+4nMAssay Description:Binding affinity to human partial length DNA-tagged SMARCA2 expressed in bacteria by BROMOscan methodMore data for this Ligand-Target Pair
TargetTranscription initiation factor TFIID subunit 1-like(Homo sapiens (Human))
University Of Strathclyde
Curated by ChEMBL
University Of Strathclyde
Curated by ChEMBL
Affinity DataKd: <3.02E+4nMAssay Description:Binding affinity to human partial length DNA-tagged TAF1L BD2 expressed in bacteria by BROMOscan methodMore data for this Ligand-Target Pair
TargetNucleosome-remodeling factor subunit BPTF(Homo sapiens (Human))
University Of Strathclyde
Curated by ChEMBL
University Of Strathclyde
Curated by ChEMBL
Affinity DataKd: <3.02E+4nMAssay Description:Binding affinity to human partial length DNA-tagged FALZ isoform1 expressed in bacteria by BROMOscan methodMore data for this Ligand-Target Pair
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
University Of Strathclyde
Curated by ChEMBL
University Of Strathclyde
Curated by ChEMBL
Affinity DataKd: <3.02E+4nMAssay Description:Binding affinity to human partial length DNA-tagged TRIM24(PHD,Bromo.) expressed in bacteria by BROMOscan methodMore data for this Ligand-Target Pair
Affinity DataKd: 1.55E+3nMAssay Description:Binding affinity to human partial length DNA-tagged BRD4 isoform long BD1 expressed in bacterial by BROMOscan methodMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase TRIM33(Homo sapiens (Human))
University Of Strathclyde
Curated by ChEMBL
University Of Strathclyde
Curated by ChEMBL
Affinity DataKd: <3.02E+4nMAssay Description:Binding affinity to human partial length DNA-tagged TRIM33(PHD,Bromo.) expressed in bacteria by BROMOscan methodMore data for this Ligand-Target Pair
TargetBromodomain testis-specific protein(Homo sapiens (Human))
University Of Strathclyde
Curated by ChEMBL
University Of Strathclyde
Curated by ChEMBL
Affinity DataKd: 1.86E+3nMAssay Description:Binding affinity to human partial length DNA-tagged BRDT isoform b BD1 expressed in bacterial by BROMOscan methodMore data for this Ligand-Target Pair
TargetBromodomain adjacent to zinc finger domain protein 2B(Homo sapiens (Human))
University Of Strathclyde
Curated by ChEMBL
University Of Strathclyde
Curated by ChEMBL
Affinity DataKd: <3.02E+4nMAssay Description:Binding affinity to human partial length DNA-tagged BAZ2B expressed in bacterial by BROMOscan methodMore data for this Ligand-Target Pair
Affinity DataKd: <3.02E+4nMAssay Description:Binding affinity to human partial length DNA-tagged PBRM1 BD5 expressed in bacteria by BROMOscan methodMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 2(Homo sapiens (Human))
University Of Strathclyde
Curated by ChEMBL
University Of Strathclyde
Curated by ChEMBL
Affinity DataKd: 1.32E+3nMAssay Description:Binding affinity to human partial length DNA-tagged BRD2 isoform 1 BD1 expressed in bacterial by BROMOscan methodMore data for this Ligand-Target Pair
Affinity DataKd: 3.00E+3nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) (N44 to E168 residues) expressed in bacterial expression system assessed as dissociation constant by BROMOsca...More data for this Ligand-Target Pair
Affinity DataKd: 2.46E+3nMAssay Description:Binding affinity to human partial length DNA-tagged BRPF1 expressed in bacterial by BROMOscan methodMore data for this Ligand-Target Pair