BindingDB PrimarySearch

Found 179 of kd for monomerid = 50505542

Fibroblast growth factor receptor 4(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL

Kd: 1.50E+3nMAssay Description:Binding affinity to recombinant N-terminal His-FLAG-GST-tagged FGFR4 (unknown origin) (460 to 802 residues) expressed in baculovirus infected Sf9 ins...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

PC cid PC sid

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Mitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL

BDBM50505542(CHEMBL4576489)

Kd: 248nMAssay Description:Binding affinity to recombinant full-length N-terminal His-FLAG-GST-tagged MAP3K5 (unknown origin) (654 to 971 residues) expressed in baculovirus inf...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Serine/threonine-protein kinase Sgk1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL

BDBM50505542(CHEMBL4576489)

Kd: 566nMAssay Description:Binding affinity to recombinant full-length N-terminal His-FLAG-GST-tagged SGK1 (unknown origin) (60 to 431 residues) expressed in baculovirus infect...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Interleukin-1 receptor-associated kinase 4(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL

BDBM50505542(CHEMBL4576489)

Kd: 75nMAssay Description:Binding affinity to recombinant full-length human N-terminal his-tagged IRAK4 expressed in baculovirus expression system using IRAK1 peptide as subst...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Calcium/calmodulin-dependent protein kinase type II subunit gamma(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL

BDBM50505542(CHEMBL4576489)

Kd: 9nMAssay Description:Binding affinity to recombinant full-length N-terminal His-FLAG-GST-tagged CAMK2G (unknown origin) expressed in baculovirus infected Sf9 insect cells...More data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Serine/threonine-protein kinase Sgk3(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL

BDBM50505542(CHEMBL4576489)

Kd: 338nMAssay Description:Binding affinity to recombinant full-length N-terminal His-FLAG-GST-tagged SGK3 (unknown origin) (119 to 496 residues) expressed in baculovirus infec...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Dual specificity protein kinase CLK2(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL

BDBM50505542(CHEMBL4576489)

Kd: 396nMAssay Description:Binding affinity to recombinant full-length N-terminal His-FLAG-GST-tagged CLK2 (unknown origin) expressed in baculovirus infected Sf9 insect cells i...More data for this Ligand-Target Pair

PDB
UniProtKB/SwissProt
B.MOAD GoogleScholar

PC cid PC sid

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Macrophage colony-stimulating factor 1 receptor(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL

BDBM50505542(CHEMBL4576489)

Kd: 324nMAssay Description:Binding affinity to recombinant N-terminal His-FLAG-GST-tagged CSF1R (unknown origin) (538 to 972 residues) expressed in baculovirus infected Sf9 ins...More data for this Ligand-Target Pair

PDB
UniProtKB/SwissProt
antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL

BDBM50505542(CHEMBL4576489)

Kd: 8nMAssay Description:Binding affinity to recombinant full-length N-terminal His-FLAG-GST-tagged PDPK1 (unknown origin) expressed in baculovirus infected Sf9 insect cells ...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

PC cid PC sid

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Dual specificity protein kinase CLK4(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL

BDBM50505542(CHEMBL4576489)

Kd: 81nMAssay Description:Binding affinity to recombinant human full length N-terminal GST-tagged CLK4 expressed in baculovirus expression system incubated for 1 hr by TR-FRET...More data for this Ligand-Target Pair

PDB MMDB KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Death-associated protein kinase 1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL

BDBM50505542(CHEMBL4576489)

Kd: 59nMAssay Description:Binding affinity to recombinant full-length N-terminal His-FLAG-GST-tagged DAPK1 (unknown origin) (1 to 289 residues) expressed in baculovirus infect...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

PC cid PC sid

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Serine/threonine-protein kinase 17A(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL

BDBM50505542(CHEMBL4576489)

Kd: 367nMAssay Description:Binding affinity to recombinant full length N-terminal His-FLAG-GST-tagged STK17A (unknown origin) expressed in baculovirus infected Sf9 insect cells...More data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar

PC cid PC sid

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Serine/threonine-protein kinase N2(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL

BDBM50505542(CHEMBL4576489)

Kd: 4nMAssay Description:Binding affinity to recombinant full-length N-terminal His-FLAG-GST-tagged PKN2 (unknown origin) expressed in baculovirus infected Sf9 insect cells i...More data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Serine/threonine-protein kinase 3(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL

BDBM50505542(CHEMBL4576489)

Kd: 3nMAssay Description:Binding affinity to recombinant full-length N-terminal His-FLAG-GST-tagged STK3 (unknown origin) expressed in baculovirus infected Sf9 insect cells i...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Ribosomal protein S6 kinase alpha-5(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL

BDBM50505542(CHEMBL4576489)

Kd: 249nMAssay Description:Binding affinity to recombinant full-length N-terminal His-FLAG-GST-tagged RPS6KA5 (unknown origin) expressed in baculovirus infected Sf9 insect cell...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank GoogleScholar

PC cid PC sid

Details Article PubMed

Protein kinase C theta type(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL

BDBM50505542(CHEMBL4576489)

Kd: 19nMAssay Description:Binding affinity to recombinant full-length N-terminal His-GST-tagged PRKCQ (unknown origin) expressed in baculovirus infected Sf9 insect cells incub...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Ribosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL

BDBM50505542(CHEMBL4576489)

Kd: 2nMAssay Description:Binding affinity to recombinant human full length N-terminal GST-tagged RPS6KA3 expressed in baculovirus expression system using S6K peptide as subst...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

PC cid PC sid

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Protein kinase C beta type(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL

BDBM50505542(CHEMBL4576489)

Kd: 17nMAssay Description:Binding affinity to recombinant full-length N-terminal His-FLAG-tagged PRKCB (unknown origin) expressed in baculovirus infected Sf9 insect cells incu...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Maternal embryonic leucine zipper kinase(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL

BDBM50505542(CHEMBL4576489)

Kd: 41nMAssay Description:Binding affinity to recombinant full-length N-terminal His-FLAG-GST-tagged MELK (unknown origin) (1 to 493 residues) expressed in baculovirus infecte...More data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Myosin light chain kinase, smooth muscle(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL

BDBM50505542(CHEMBL4576489)

Kd: 298nMAssay Description:Binding affinity to recombinant full-length N-terminal His-FLAG-GST-tagged MYLK (unknown origin) (1428 to 1771 residues) expressed in baculovirus inf...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

NT-3 growth factor receptor(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL

BDBM50505542(CHEMBL4576489)

Kd: 19nMAssay Description:Binding affinity to recombinant full-length N-terminal His-FLAG-GST-tagged NTRK3 (unknown origin) expressed in baculovirus infected Sf9 insect cells ...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

TRAF2 and NCK-interacting protein kinase(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL

BDBM50505542(CHEMBL4576489)

Kd: 97nMAssay Description:Binding affinity to recombinant full-length N-terminal His-FLAG-GST-tagged TNIK (unknown origin) (1 to 314 residues) expressed in baculovirus infecte...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
B.MOAD GoogleScholar

PC cid PC sid

Details Article PubMed

Serine/threonine-protein kinase 38-like(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL

BDBM50505542(CHEMBL4576489)

Kd: >2.00E+3nMAssay Description:Binding affinity to recombinant full-length N-terminal His-FLAG-GST-tagged STK38L (unknown origin) expressed in baculovirus infected Sf9 insect cells...More data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

TGF-beta receptor type-2(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL

BDBM50505542(CHEMBL4576489)

Kd: >2.00E+3nMAssay Description:Binding affinity to recombinant N-terminal His-FLAG-GST-tagged TGFBR2 (unknown origin) (194 to 567 residues) expressed in baculovirus infected Sf9 in...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt UniProtKB/TrEMBL
B.MOAD DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Non-receptor tyrosine-protein kinase TYK2(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL

BDBM50505542(CHEMBL4576489)

Kd: 49nMAssay Description:Binding affinity to recombinant N-terminal His-FLAG-GST-tagged TYK2 (unknown origin) (871 to 1187 residues) expressed in baculovirus infected Sf9 ins...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt UniProtKB/TrEMBL
B.MOAD DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

LIM domain kinase 1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL

BDBM50505542(CHEMBL4576489)

Kd: 32nMAssay Description:Binding affinity to truncated human N-terminal GST-tagged LIMK1 (285 to 638 residues) expressed in baculovirus expression system using cofilin2 as su...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Non-receptor tyrosine-protein kinase TNK1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL

BDBM50505542(CHEMBL4576489)

Kd: 13nMAssay Description:Binding affinity to recombinant human N-terminal GST-tagged TNK1 (106 to 390 residues) expressed in baculovirus expression system using CSKtide as su...More data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Calcium/calmodulin-dependent protein kinase kinase 2(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL

BDBM50505542(CHEMBL4576489)

Kd: 6nMAssay Description:Binding affinity to recombinant full-length N-terminal His-FLAG-GST-tagged CAMKK2 (unknown origin) expressed in baculovirus infected Sf9 insect cells...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Fibroblast growth factor receptor 1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL

BDBM50505542(CHEMBL4576489)

Kd: 643nMAssay Description:Binding affinity to recombinant N-terminal His-FLAG-GST-tagged FGFR1 (unknown origin) (396 to 820 residues) expressed in baculovirus infected Sf9 ins...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL

BDBM50505542(CHEMBL4576489)

Kd: 3nMAssay Description:Binding affinity to recombinant full-length N-terminal His-FLAG-GST-tagged PHKG1 (unknown origin) expressed in baculovirus infected Sf9 insect cells ...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Serine/threonine-protein kinase ULK1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL

BDBM50505542(CHEMBL4576489)

Kd: 311nMAssay Description:Binding affinity to recombinant N-terminal His-FLAG-GST-tagged ULK1 (unknown origin) (1 to 649 residues) expressed in baculovirus infected Sf9 insect...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Serine/threonine-protein kinase 32B(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL

BDBM50505542(CHEMBL4576489)

Kd: 984nMAssay Description:Binding affinity to recombinant full-length N-terminal His-FLAG-GST-tagged STK32B (unknown origin) expressed in baculovirus infected Sf9 insect cells...More data for this Ligand-Target Pair

KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Fibroblast growth factor receptor 3(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL

BDBM50505542(CHEMBL4576489)

Kd: 848nMAssay Description:Binding affinity to recombinant N-terminal His-FLAG-GST-tagged FGFR3 (unknown origin) (436 to 806 residues) expressed in baculovirus infected Sf9 ins...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Interleukin-1 receptor-associated kinase 1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL

BDBM50505542(CHEMBL4576489)

Kd: 609nMAssay Description:Binding affinity to recombinant N-terminal His-FLAG-GST-tagged IRAK1 (unknown origin) (194 to 712 residues) expressed in baculovirus infected Sf9 ins...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Tyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL

BDBM50505542(CHEMBL4576489)

Kd: 765nMAssay Description:Binding affinity to recombinant human full-length N-terminal GST-tagged ITK expressed in baculovirus expression system using srctide as substrate inc...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Tyrosine-protein kinase receptor TYRO3(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL

BDBM50505542(CHEMBL4576489)

Kd: 1.05E+3nMAssay Description:Binding affinity to recombinant full-length N-terminal His-FLAG-GST-tagged TYRO3 (unknown origin) expressed in baculovirus infected Sf9 insect cells ...More data for this Ligand-Target Pair

PDB MMDB KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Tyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL

BDBM50505542(CHEMBL4576489)

Kd: 559nMAssay Description:Binding affinity to recombinant full-length N-terminal His-FLAG-GST-tagged AXL (unknown origin) expressed in baculovirus infected Sf9 insect cells in...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Tyrosine-protein kinase ABL2(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL

BDBM50505542(CHEMBL4576489)

Kd: 947nMAssay Description:Binding affinity to recombinant full-length N-terminal His-FLAG-GST-tagged ABL2 (unknown origin) (2 to 52 and 74 to 1182 residues) expressed in bacul...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Serine/threonine-protein kinase BRSK1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL

BDBM50505542(CHEMBL4576489)

Kd: 194nMAssay Description:Binding affinity to recombinant full-length N-terminal His-FLAG-GST-tagged BRSK1 (unknown origin) expressed in baculovirus infected Sf9 insect cells ...More data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Serine/threonine-protein kinase D2(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL

BDBM50505542(CHEMBL4576489)

Kd: 140nMAssay Description:Binding affinity to recombinant full-length N-terminal His-FLAG-tagged PRKD2 (unknown origin) expressed in baculovirus infected Sf9 insect cells incu...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Serine/threonine-protein kinase 24(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL

BDBM50505542(CHEMBL4576489)

Kd: 767nMAssay Description:Binding affinity to recombinant full-length N-terminal His-FLAG-tagged STK24 (unknown origin) expressed in baculovirus infected Sf9 insect cells incu...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Receptor tyrosine-protein kinase erbB-4(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL

BDBM50505542(CHEMBL4576489)

Kd: 798nMAssay Description:Binding affinity to recombinant human full-length N-terminal GST-tagged ERBB4 expressed in baculovirus expression system using srctide as substrate i...More data for this Ligand-Target Pair

PDB MMDB
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Platelet-derived growth factor receptor beta(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL

BDBM50505542(CHEMBL4576489)

Kd: 257nMAssay Description:Binding affinity to recombinant human N-terminal his-tagged PDGFRB (558 to 1106 residues) expressed in baculovirus expression system incubated for 1 ...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Fibroblast growth factor receptor 2(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL

BDBM50505542(CHEMBL4576489)

Kd: 361nMAssay Description:Binding affinity to recombinant N-terminal His-FLAG-GST-tagged FGFR2 (unknown origin) (399 to 821 residues) expressed in baculovirus infected Sf9 ins...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Serine/threonine-protein kinase Sgk2(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL

BDBM50505542(CHEMBL4576489)

Kd: 1.77E+3nMAssay Description:Binding affinity to recombinant full-length N-terminal His-FLAG-tagged SGK2 (unknown origin) expressed in baculovirus infected Sf9 insect cells incub...More data for this Ligand-Target Pair

Reactome pathway KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Mitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL

BDBM50505542(CHEMBL4576489)

Kd: 24nMAssay Description:Binding affinity to recombinant N-terminal His-FLAG-GST-tagged MAP4K1 (unknown origin) (1 to 346 residues) expressed in baculovirus infected Sf9 inse...More data for this Ligand-Target Pair

PDB NCI pathway KEGG
UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

Details Article PubMed

Mitogen-activated protein kinase kinase kinase 2(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL

BDBM50505542(CHEMBL4576489)

Kd: 53nMAssay Description:Binding affinity to recombinant full-length N-terminal His-FLAG-GST-tagged MAP3K2 (unknown origin) (337 to 620 residues) expressed in baculovirus inf...More data for this Ligand-Target Pair

PDB MMDB KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Serine/threonine-protein kinase pim-1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL

BDBM50505542(CHEMBL4576489)

Kd: 285nMAssay Description:Binding affinity to recombinant human full-length N-terminal his-tagged PIM1 expressed in baculovirus expression system using S6K2 peptide as substra...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Mitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL

BDBM50505542(CHEMBL4576489)

Kd: 60nMAssay Description:Binding affinity to recombinant full-length N-terminal His-FLAG-tagged MAP3K7 (unknown origin) expressed in baculovirus infected Sf9 insect cells inc...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Dual specificity protein kinase CLK1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL

BDBM50505542(CHEMBL4576489)

Kd: 125nMAssay Description:Binding affinity to recombinant N-terminal His-FLAG-GST-tagged CLK1 (unknown origin) (129 to 484 residues) expressed in baculovirus infected Sf9 inse...More data for this Ligand-Target Pair

PDB MMDB KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Displayed 1 to 50 (of 179 total ) | Next | Last >>

Filter my 179 hits

Targets 179▿
- Tyrosine-protein kinase Tec 1
- Peripheral plasma membrane protein CASK 1
- 5'-AMP-activated protein kinase catalytic subunit alpha-1/subunit beta-1/subunit gamma-1 1
- Receptor tyrosine-protein kinase erbB-4 1
- BMP-2-inducible protein kinase 1
- Rhodopsin kinase GRK1 1
- Tyrosine-protein kinase FRK 1
- LIM domain kinase 1 1
- Hepatocyte growth factor receptor 1
- ALK tyrosine kinase receptor 1
- NUAK family SNF1-like kinase 2 1
- Non-receptor tyrosine-protein kinase TYK2 1
- Glycogen synthase kinase-3 alpha 1
- Glycogen synthase kinase-3 beta 1
- Protein kinase C iota type 1
- NUAK family SNF1-like kinase 1 1
- AP2-associated protein kinase 1 1
- Calcium/calmodulin-dependent protein kinase type II subunit beta 1
- Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform 1
- MAP/microtubule affinity-regulating kinase 3 1
- Homeodomain-interacting protein kinase 4 1
- Protein kinase C theta type 1
- Homeodomain-interacting protein kinase 3 1
- MAP kinase-interacting serine/threonine-protein kinase 2 1
- Serine/threonine-protein kinase PAK 4 1
- Serine/threonine-protein kinase PAK 5 1
- Serine/threonine-protein kinase PAK 6 1
- Tyrosine-protein kinase JAK3 1
- Dual specificity mitogen-activated protein kinase kinase 1 1
- Proto-oncogene tyrosine-protein kinase receptor Ret 1
- Dual specificity mitogen-activated protein kinase kinase 6 1
- Serine/threonine-protein kinase Sgk2 1
- Serine/threonine-protein kinase Sgk1 1
- Serine/threonine-protein kinase Sgk3 1
- Ephrin type-A receptor 1 1
- Serine/threonine-protein kinase 38-like 1
- Myosin-IIIb 1
- Tyrosine-protein kinase BTK 1
- Ephrin type-A receptor 7 1
- Myotonin-protein kinase 1
- Tyrosine-protein kinase ITK/TSK 1
- Tyrosine-protein kinase receptor UFO 1
- Cyclin-C 1
- Protein kinase C eta type 1
- Tyrosine-protein kinase Blk 1
- Serine/threonine-protein kinase 16 1
- Non-receptor tyrosine-protein kinase TNK1 1
- Inhibitor of nuclear factor kappa-B kinase subunit epsilon 1
- Homeodomain-interacting protein kinase 2 1
- Ribosomal protein S6 kinase beta-1 1
- Protein kinase C beta type 1
- Tyrosine-protein kinase Lyn 1
- Serine/threonine-protein kinase 26 1
- Focal adhesion kinase 1 1
- Serine/threonine-protein kinase 24 1
- Serine/threonine-protein kinase 25 1
- Serine/threonine-protein kinase 33 1
- cAMP-dependent protein kinase catalytic subunit gamma 1
- Activated CDC42 kinase 1 1
- Platelet-derived growth factor receptor beta 1
- Epithelial discoidin domain-containing receptor 1 1
- [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial 1
- Death-associated protein kinase 2 1
- Death-associated protein kinase 1 1
- Tyrosine-protein kinase Fer 1
- Serine/threonine-protein kinase D2 1
- TGF-beta receptor type-2 1
- 5'-AMP-activated protein kinase catalytic subunit alpha-2 1
- Calcium/calmodulin-dependent protein kinase type II subunit delta 1
- Dual specificity tyrosine-phosphorylation-regulated kinase 1B 1
- Death-associated protein kinase 3 1
- Dual specificity tyrosine-phosphorylation-regulated kinase 1A 1
- Serine/threonine-protein kinase pim-1 1
- Serine/threonine-protein kinase TAO1 1
- Calcium/calmodulin-dependent protein kinase kinase 1 1
- Serine/threonine-protein kinase TAO3 1
- Calcium/calmodulin-dependent protein kinase kinase 2 1
- Serine/threonine-protein kinase DCLK3 1
- Testis-specific serine/threonine-protein kinase 1 1
- Serine/threonine-protein kinase TNNI3K 1
- Angiopoietin-1 receptor 1
- Mitogen-activated protein kinase kinase kinase kinase 2 1
- Protein kinase C epsilon type 1
- Mitogen-activated protein kinase kinase kinase kinase 1 1
- Serine/threonine-protein kinase MRCK alpha 1
- Mitogen-activated protein kinase kinase kinase kinase 5 1
- Mitogen-activated protein kinase 15 1
- Testis-specific serine/threonine-protein kinase 3 1
- Leukocyte tyrosine kinase receptor 1
- Interleukin-1 receptor-associated kinase 4 1
- Cytoplasmic tyrosine-protein kinase BMX 1
- Mitogen-activated protein kinase kinase kinase 9 1
- RAC-gamma serine/threonine-protein kinase 1
- Mitogen-activated protein kinase kinase kinase 5 1
- Interleukin-1 receptor-associated kinase 1 1
- Tyrosine-protein kinase ABL2 1
- Mitogen-activated protein kinase kinase kinase 7 1
- Mitogen-activated protein kinase kinase kinase 2 1
- Cyclin-C/Cyclin-dependent kinase 19 1
- Calcium/calmodulin-dependent protein kinase type II subunit alpha 1
- cGMP-dependent protein kinase 2 1
- Rho-associated protein kinase 2 1
- cGMP-dependent protein kinase 1 1
- Rho-associated protein kinase 1 1
- Serine/threonine-protein kinase ULK1 1
- Proto-oncogene tyrosine-protein kinase Src 1
- Tyrosine-protein kinase Fes/Fps 1
- Serine/threonine-protein kinase SIK2 1
- Myosin light chain kinase, smooth muscle 1
- Serine/threonine-protein kinase SIK1 1
- Serine/threonine-protein kinase ULK2 1
- Serine/threonine-protein kinase ULK3 1
- Serine/threonine-protein kinase 3 1
- 3-phosphoinositide-dependent protein kinase 1 1
- Serine/threonine-protein kinase 17A 1
- Tyrosine-protein kinase Lck 1
- Serine/threonine-protein kinase 4 1
- Dual specificity protein kinase CLK1 1
- CDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7 1
- Mitogen-activated protein kinase kinase kinase 14 1
- Protein kinase C delta type 1
- NT-3 growth factor receptor 1
- Mitogen-activated protein kinase 9 1
- Dual specificity protein kinase CLK4 1
- Dual specificity protein kinase CLK2 1
- Protein-tyrosine kinase 2-beta 1
- Tyrosine-protein kinase Mer 1
- High affinity nerve growth factor receptor 1
- Serine/threonine-protein kinase N2 1
- cAMP-dependent protein kinase catalytic subunit beta 1
- Calcium/calmodulin-dependent protein kinase type II subunit gamma 1
- Mitogen-activated protein kinase 8 1
- Serine/threonine-protein kinase N1 1
- Ribosomal protein S6 kinase alpha-2 1
- Tyrosine-protein kinase SYK 1
- Ribosomal protein S6 kinase alpha-3 1
- Ribosomal protein S6 kinase alpha-1 1
- Serine/threonine-protein kinase TBK1 1
- Cyclin-T1/Cyclin-dependent kinase 9 1
- Phosphorylase b kinase gamma catalytic chain, liver/testis isoform 1
- STE20-like serine/threonine-protein kinase 1
- Calcium/calmodulin-dependent protein kinase type 1G 1
- Fibroblast growth factor receptor 4 1
- Serine/threonine-protein kinase 32B 1
- Serine/threonine-protein kinase 32A 1
- Serine/threonine-protein kinase 32C 1
- Vascular endothelial growth factor receptor 2 1
- Tyrosine-protein kinase Fgr 1
- Insulin receptor 1
- Vascular endothelial growth factor receptor 3 1
- Tyrosine-protein kinase HCK 1
- Aurora kinase A 1
- Fibroblast growth factor receptor 1 1
- Fibroblast growth factor receptor 2 1
- Fibroblast growth factor receptor 3 1
- Serine/threonine-protein kinase PLK4 1
- Mitogen-activated protein kinase 12 1
- Tyrosine-protein kinase receptor TYRO3 1
- RAC-beta serine/threonine-protein kinase 1
- Mitogen-activated protein kinase 10 1
- Serine/threonine-protein kinase BRSK1 1
- Protein kinase C gamma type 1
- Serine/threonine-protein kinase LATS2 1
- Misshapen-like kinase 1 1
- Tyrosine-protein kinase Fyn 1
- Tyrosine-protein kinase CSK 1
- Macrophage colony-stimulating factor 1 receptor 1
- cAMP-dependent protein kinase catalytic subunit alpha 1
- Citron Rho-interacting kinase 1
- Ribosomal protein S6 kinase alpha-6 1
- Protein kinase C alpha type 1
- Ribosomal protein S6 kinase alpha-5 1
- Maternal embryonic leucine zipper kinase 1
- Protein kinase C zeta type 1
- Serine/threonine-protein kinase MARK1 1
- Serine/threonine-protein kinase MARK2 1
- TRAF2 and NCK-interacting protein kinase 1
- Tyrosine-protein kinase Yes 1
- Mitogen-activated protein kinase kinase kinase 11 1
Publications 1▿
- Bioorg Med Chem Lett 29: (2019) 179
Institutions 1▿
- Takeda Pharmaceutical 179
Affinity: 2 to 2.0E+3 nM▿
- Kd 179
- Affinity ≤ nM
Xtal structures: 0
Docked structures: 0
Catalog Cmpds: 0