Affinity DataKd: 2.67E+5nMAssay Description:In vitro affinity at mutant D2 receptor (S194A) in C6 (glioma) cell membranes.More data for this Ligand-Target Pair
Affinity DataKd: 4.90E+4nMAssay Description:In vitro affinity at mutant D2 receptor (S197A) in C6 (glioma) cell membranes.More data for this Ligand-Target Pair
Affinity DataKd: 6.20E+3nMAssay Description:In vitro affinity at wild type Dopamine receptor D2 on C6 (glioma) cell membranes.More data for this Ligand-Target Pair
Affinity DataKd: 3.70E+4nMAssay Description:In vitro affinity at mutant D2 receptor (S194A) in C6 (glioma) cell membranes.More data for this Ligand-Target Pair
Affinity DataKd: 1.70E+4nMAssay Description:Equilibrium dissociation constant against recombinant Dopamine receptor D2A expressed in COS7 cellsMore data for this Ligand-Target Pair
Affinity DataKd: 2.50E+3nMAssay Description:Equilibrium dissociation constant against recombinant Dopamine receptor D1A expressed in COS7 cellsMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Instituto Polit£Cnico Nacional (Ipn)
Curated by ChEMBL
Instituto Polit£Cnico Nacional (Ipn)
Curated by ChEMBL
Affinity DataKd: 6.46E+4nMAssay Description:Binding affinity to human adrenergic beta2 receptorMore data for this Ligand-Target Pair