TargetAcetylcholinesterase(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Affinity DataKd: 0nMAssay Description:Binding affinity to acetylcholine esterase (unknown origin)More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataKd: 0nMAssay Description:Binding affinity to Torpedo californica acetylcholinesterase by fluorescence methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Affinity DataKd: 0nMAssay Description:Binding affinity to acetylcholine esterase (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 0nMAssay Description:Inhibition of mouse AChE active site after 12 hrs by LC/MS-SIM analysisMore data for this Ligand-Target Pair
Affinity DataKd: 0nMAssay Description:Inhibition of mouse AChE active site after 12 hrs by LC/MS-SIM analysisMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Groningen
Curated by ChEMBL
University Of Groningen
Curated by ChEMBL
Affinity DataKd: 0nMAssay Description:Binding affinity to electric eel AChE after 24 hrs by LC/MS-SIM analysisMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Groningen
Curated by ChEMBL
University Of Groningen
Curated by ChEMBL
Affinity DataKd: 0nMAssay Description:Binding affinity to electric eel AChE after 24 hrs by LC/MS-SIM analysisMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Groningen
Curated by ChEMBL
University Of Groningen
Curated by ChEMBL
Affinity DataKd: 0nMAssay Description:Binding affinity to electric eel AChE after 24 hrs by LC/MS-SIM analysisMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Groningen
Curated by ChEMBL
University Of Groningen
Curated by ChEMBL
Affinity DataKd: 0nMAssay Description:Binding affinity to electric eel AChE after 24 hrs by LC/MS-SIM analysisMore data for this Ligand-Target Pair
Affinity DataKd: 0nMAssay Description:Inhibition of mouse AChE active site after 12 hrs by LC/MS-SIM analysisMore data for this Ligand-Target Pair
Affinity DataKd: 0nMAssay Description:Inhibition of mouse AChE active site after 12 hrs by LC/MS-SIM analysisMore data for this Ligand-Target Pair
Affinity DataKd: 0nMAssay Description:Inhibition of mouse AChE active site after 12 hrs by LC/MS-SIM analysisMore data for this Ligand-Target Pair
Affinity DataKd: 0nMAssay Description:Inhibition of mouse AChE active site after 12 hrs by LC/MS-SIM analysisMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Groningen
Curated by ChEMBL
University Of Groningen
Curated by ChEMBL
Affinity DataKd: 0nMAssay Description:Binding affinity to electric eel AChE after 24 hrs by LC/MS-SIM analysisMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Groningen
Curated by ChEMBL
University Of Groningen
Curated by ChEMBL
Affinity DataKd: 0nMAssay Description:Binding affinity to electric eel AChE after 24 hrs by LC/MS-SIM analysisMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Groningen
Curated by ChEMBL
University Of Groningen
Curated by ChEMBL
Affinity DataKd: 0nMAssay Description:Binding affinity to electric eel AChE after 24 hrs by LC/MS-SIM analysisMore data for this Ligand-Target Pair
Affinity DataKd: 0nMAssay Description:Inhibition of mouse AChE active site after 12 hrs by LC/MS-SIM analysisMore data for this Ligand-Target Pair
Affinity DataKd: 0nMAssay Description:Inhibition of mouse AChE active site after 12 hrs by LC/MS-SIM analysisMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Groningen
Curated by ChEMBL
University Of Groningen
Curated by ChEMBL
Affinity DataKd: 0nMAssay Description:Binding affinity to electric eel AChE after 24 hrs by LC/MS-SIM analysisMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Affinity DataKd: 0nMAssay Description:Binding affinity to acetylcholine esterase (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 0.000410nMAssay Description:Dissociation constant towards Acetylcholinesterase in mouseMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Affinity DataKd: 0.940nMAssay Description:Mixed-type inhibition of recombinant human AChE using varying concentration of acetylthiocholine iodide as substrate at 0.17 to 1.36 nM by Lineweaver...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Affinity DataKd: 2.80nMAssay Description:Binding affinity to CM5 sensor chip immobilized recombinant human AChE assessed as dissociation constant at 298.15 K by surface plasmon resonance ass...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Affinity DataKd: 3.5nMAssay Description:Binding affinity to CM5 sensor chip immobilized recombinant human AChE assessed as dissociation constant at 298.15 K by surface plasmon resonance ass...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Affinity DataKd: 3.5nMAssay Description:Binding affinity to CM5 sensor chip immobilized recombinant human AChE assessed as dissociation constant at 298.15 K by surface plasmon resonance ass...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Groningen
Curated by ChEMBL
University Of Groningen
Curated by ChEMBL
Affinity DataKd: 3.60nMAssay Description:Displacement of propidium iodide from PAS-region of electric eel AChE assessed as dissociation constant by spectrofluorimetric analysisMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Affinity DataKd: 4.60nMAssay Description:Binding affinity to CM5 sensor chip immobilized recombinant human AChE assessed as dissociation constant at 298.15 K by surface plasmon resonance ass...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Affinity DataKd: 5nMAssay Description:Binding affinity to CM5 sensor chip immobilized recombinant human AChE assessed as dissociation constant at 298.15 K by surface plasmon resonance ass...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Affinity DataKd: 5.20nMAssay Description:Binding affinity to CM5 sensor chip immobilized recombinant human AChE assessed as dissociation constant at 298.15 K by surface plasmon resonance ass...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Affinity DataKd: 8nMAssay Description:Binding affinity to CM5 sensor chip immobilized recombinant human AChE assessed as dissociation constant at 298.15 K by surface plasmon resonance ass...More data for this Ligand-Target Pair
Affinity DataKd: 10nMAssay Description:Binding affinity to mouse ACHE by fluorescence methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Groningen
Curated by ChEMBL
University Of Groningen
Curated by ChEMBL
Affinity DataKd: 16nMAssay Description:Binding affinity to electric eel AChE after 24 hrs by LC/MS-SIM analysisMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Affinity DataKd: 17nMAssay Description:Binding affinity to CM5 sensor chip immobilized recombinant human AChE assessed as dissociation constant at 298.15 K by surface plasmon resonance ass...More data for this Ligand-Target Pair
Affinity DataKd: 18nMAssay Description:Dissociation constant towards Acetylcholinesterase in mouseMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Groningen
Curated by ChEMBL
University Of Groningen
Curated by ChEMBL
Affinity DataKd: 400nMAssay Description:Binding affinity against adenosine A1 receptor from rat brain membranes using [3H]cyclohexyladenosine as radioligand.More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Groningen
Curated by ChEMBL
University Of Groningen
Curated by ChEMBL
Affinity DataKd: 610nMAssay Description:Binding affinity to electric eel AChEMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Affinity DataKd: 680nMAssay Description:Reactivation of paraoxon-inhibited human AChE assessed as dissociation constant incubated for 30 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Affinity DataKd: 750nMAssay Description:Reactivation of parathion-inhibited human AChE assessed as dissociation constant incubated for 30 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Affinity DataKd: 990nMAssay Description:Reactivation of dichlorvos-inhibited human AChE assessed as dissociation constant incubated for 30 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Groningen
Curated by ChEMBL
University Of Groningen
Curated by ChEMBL
Affinity DataKd: 1.10E+3nMAssay Description:Binding affinity to electric eel AChE after 24 hrs by LC/MS-SIM analysisMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Affinity DataKd: 1.10E+3nMAssay Description:Reactivation of paraoxon-inhibited recombinant human AChE measured up to 10 mins by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataKd: 1.10E+3nMAssay Description:Dissociation constant towards Acetylcholinesterase in mouseMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Affinity DataKd: 1.20E+3nMAssay Description:Reactivation of dichlorvos-inhibited human AChE assessed as dissociation constant incubated for 30 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Groningen
Curated by ChEMBL
University Of Groningen
Curated by ChEMBL
Affinity DataKd: 1.76E+3nMAssay Description:Displacement of propidium from electric eel AChE peripheral anionic site assessed as decrease in fluorescence intensity by spectrofluorometric analys...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Groningen
Curated by ChEMBL
University Of Groningen
Curated by ChEMBL
Affinity DataKd: 2.00E+3nMAssay Description:Binding affinity to Electric eel AChEMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Groningen
Curated by ChEMBL
University Of Groningen
Curated by ChEMBL
Affinity DataKd: 2.03E+3nMAssay Description:Displacement of propidium iodide from PAS region of electric eel AChE by fluorescence assayMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Affinity DataKd: 2.10E+3nMAssay Description:Reactivation of sarin-inhibited human AChE assessed as dissociation constant incubated for 30 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Groningen
Curated by ChEMBL
University Of Groningen
Curated by ChEMBL
Affinity DataKd: 2.18E+3nMAssay Description:Displacement of propidium from electric eel AChE peripheral anionic site assessed as decrease in fluorescence intensity by spectrofluorometric analys...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Groningen
Curated by ChEMBL
University Of Groningen
Curated by ChEMBL
Affinity DataKd: 2.20E+3nMAssay Description:Binding affinity to Electric eel AChEMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Affinity DataKd: 2.31E+3nMAssay Description:Binding affinity to sarin-inhibited hemoglobin free erythrocyte ghost human AChE using acetylcholine iodide as substrate measured for 1 hr by spectro...More data for this Ligand-Target Pair