Compile Data Set for Download or QSAR
maximum 50k data
Found 468 of ec50 data for polymerid = 2129
TargetAdenosine receptor A1(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM191826(US9187428, 54)
Affinity DataEC50:  0.0400nMpH: 7.4 T: 2°CAssay Description:The following test protocol is used for pharmacologically characterizing cells and for the robot-assisted substance screening:The stock cultures ar...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM191818(US9187428, 46)
Affinity DataEC50:  0.0400nMpH: 7.4 T: 2°CAssay Description:The following test protocol is used for pharmacologically characterizing cells and for the robot-assisted substance screening:The stock cultures ar...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM191778(US9187428, 6)
Affinity DataEC50:  0.0600nMpH: 7.4 T: 2°CAssay Description:The following test protocol is used for pharmacologically characterizing cells and for the robot-assisted substance screening:The stock cultures ar...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM191785(US9187428, 13)
Affinity DataEC50:  0.0800nMpH: 7.4 T: 2°CAssay Description:The following test protocol is used for pharmacologically characterizing cells and for the robot-assisted substance screening:The stock cultures ar...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM191850(US9187428, 78)
Affinity DataEC50:  0.100nMpH: 7.4 T: 2°CAssay Description:The following test protocol is used for pharmacologically characterizing cells and for the robot-assisted substance screening:The stock cultures ar...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM50003646(CHEMBL3235279)
Affinity DataEC50:  0.100nMAssay Description:Agonist activity at adenosine A1 receptor (unknown origin) expressed in CHO cells assessed as increase in intracellular cAMP level by RIAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM50588454(CHEMBL5174052)
Affinity DataEC50:  0.100nMAssay Description:Agonist activity at human adenosine A1 receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM191779(US9187428, 7)
Affinity DataEC50:  0.100nMpH: 7.4 T: 2°CAssay Description:The following test protocol is used for pharmacologically characterizing cells and for the robot-assisted substance screening:The stock cultures ar...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM21220((2S,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-N-ethyl-3,...)
Affinity DataEC50:  0.120nMAssay Description:Agonist activity at human A1A adenosine receptor expressed in HEK cell membranes incubated for 60 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM50588462(CHEMBL5195714)
Affinity DataEC50:  0.123nMAssay Description:Agonist activity at human adenosine A1 receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM50588460(CHEMBL5187330)
Affinity DataEC50:  0.132nMAssay Description:Agonist activity at human adenosine A1 receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM50588447(CHEMBL5172389)
Affinity DataEC50:  0.141nMAssay Description:Agonist activity at human adenosine A1 receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
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US Patent
LigandPNGBDBM25400((2R,3R,4S,5R)-2-[6-(cyclopentylamino)-9H-purin-9-y...)
Affinity DataEC50:  0.190nMAssay Description:Compound was evaluated for the Adenosine A1 receptor agonist potency.More data for this Ligand-Target Pair
In DepthDetails Article
TargetAdenosine receptor A1(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM191842(US9187428, 70)
Affinity DataEC50:  0.200nMpH: 7.4 T: 2°CAssay Description:The following test protocol is used for pharmacologically characterizing cells and for the robot-assisted substance screening:The stock cultures ar...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM191775(US9187428, 3)
Affinity DataEC50:  0.200nMpH: 7.4 T: 2°CAssay Description:The following test protocol is used for pharmacologically characterizing cells and for the robot-assisted substance screening:The stock cultures ar...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM191873(US9187428, 101)
Affinity DataEC50:  0.200nMpH: 7.4 T: 2°CAssay Description:The following test protocol is used for pharmacologically characterizing cells and for the robot-assisted substance screening:The stock cultures ar...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM191866(US9187428, 94)
Affinity DataEC50:  0.200nMpH: 7.4 T: 2°CAssay Description:The following test protocol is used for pharmacologically characterizing cells and for the robot-assisted substance screening:The stock cultures ar...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM191855(US9187428, 83)
Affinity DataEC50:  0.200nMpH: 7.4 T: 2°CAssay Description:The following test protocol is used for pharmacologically characterizing cells and for the robot-assisted substance screening:The stock cultures ar...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Homo sapiens (Human))
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US Patent
LigandPNGBDBM191854(US9187428, 82)
Affinity DataEC50:  0.200nMpH: 7.4 T: 2°CAssay Description:The following test protocol is used for pharmacologically characterizing cells and for the robot-assisted substance screening:The stock cultures ar...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM191847(US9187428, 75)
Affinity DataEC50:  0.200nMpH: 7.4 T: 2°CAssay Description:The following test protocol is used for pharmacologically characterizing cells and for the robot-assisted substance screening:The stock cultures ar...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM191823(US9187428, 51)
Affinity DataEC50:  0.200nMpH: 7.4 T: 2°CAssay Description:The following test protocol is used for pharmacologically characterizing cells and for the robot-assisted substance screening:The stock cultures ar...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM191798(US9187428, 26)
Affinity DataEC50:  0.200nMpH: 7.4 T: 2°CAssay Description:The following test protocol is used for pharmacologically characterizing cells and for the robot-assisted substance screening:The stock cultures ar...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM50588461(CHEMBL5203632)
Affinity DataEC50:  0.240nMAssay Description:Agonist activity at human adenosine A1 receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM50588458(CHEMBL5171042)
Affinity DataEC50:  0.295nMAssay Description:Agonist activity at human adenosine A1 receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM191776(US9187428, 4 | US9187428, 53)
Affinity DataEC50:  0.300nMpH: 7.4 T: 2°CAssay Description:The following test protocol is used for pharmacologically characterizing cells and for the robot-assisted substance screening:The stock cultures ar...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM191805(US9187428, 33)
Affinity DataEC50:  0.300nMpH: 7.4 T: 2°CAssay Description:The following test protocol is used for pharmacologically characterizing cells and for the robot-assisted substance screening:The stock cultures ar...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM191799(US9187428, 27)
Affinity DataEC50:  0.300nMpH: 7.4 T: 2°CAssay Description:The following test protocol is used for pharmacologically characterizing cells and for the robot-assisted substance screening:The stock cultures ar...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM191821(US9187428, 49)
Affinity DataEC50:  0.300nMpH: 7.4 T: 2°CAssay Description:The following test protocol is used for pharmacologically characterizing cells and for the robot-assisted substance screening:The stock cultures ar...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM191774(US9187428, 2)
Affinity DataEC50:  0.300nMpH: 7.4 T: 2°CAssay Description:The following test protocol is used for pharmacologically characterizing cells and for the robot-assisted substance screening:The stock cultures ar...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM191776(US9187428, 4 | US9187428, 53)
Affinity DataEC50:  0.300nMpH: 7.4 T: 2°CAssay Description:The following test protocol is used for pharmacologically characterizing cells and for the robot-assisted substance screening:The stock cultures ar...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM191870(US9187428, 98)
Affinity DataEC50:  0.300nMpH: 7.4 T: 2°CAssay Description:The following test protocol is used for pharmacologically characterizing cells and for the robot-assisted substance screening:The stock cultures ar...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM191834(US9187428, 62)
Affinity DataEC50:  0.300nMpH: 7.4 T: 2°CAssay Description:The following test protocol is used for pharmacologically characterizing cells and for the robot-assisted substance screening:The stock cultures ar...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM191816(US9187428, 44)
Affinity DataEC50:  0.400nMpH: 7.4 T: 2°CAssay Description:The following test protocol is used for pharmacologically characterizing cells and for the robot-assisted substance screening:The stock cultures ar...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM191804(US9187428, 32)
Affinity DataEC50:  0.400nMpH: 7.4 T: 2°CAssay Description:The following test protocol is used for pharmacologically characterizing cells and for the robot-assisted substance screening:The stock cultures ar...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM191840(US9187428, 68)
Affinity DataEC50:  0.400nMpH: 7.4 T: 2°CAssay Description:The following test protocol is used for pharmacologically characterizing cells and for the robot-assisted substance screening:The stock cultures ar...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM191800(US9187428, 28)
Affinity DataEC50:  0.400nMpH: 7.4 T: 2°CAssay Description:The following test protocol is used for pharmacologically characterizing cells and for the robot-assisted substance screening:The stock cultures ar...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM191802(US9187428, 30)
Affinity DataEC50:  0.400nMpH: 7.4 T: 2°CAssay Description:The following test protocol is used for pharmacologically characterizing cells and for the robot-assisted substance screening:The stock cultures ar...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM191868(US9187428, 96)
Affinity DataEC50:  0.400nMpH: 7.4 T: 2°CAssay Description:The following test protocol is used for pharmacologically characterizing cells and for the robot-assisted substance screening:The stock cultures ar...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM191827(US9187428, 55)
Affinity DataEC50:  0.400nMpH: 7.4 T: 2°CAssay Description:The following test protocol is used for pharmacologically characterizing cells and for the robot-assisted substance screening:The stock cultures ar...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM191832(US9187428, 60)
Affinity DataEC50:  0.400nMpH: 7.4 T: 2°CAssay Description:The following test protocol is used for pharmacologically characterizing cells and for the robot-assisted substance screening:The stock cultures ar...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM191856(US9187428, 84)
Affinity DataEC50:  0.400nMpH: 7.4 T: 2°CAssay Description:The following test protocol is used for pharmacologically characterizing cells and for the robot-assisted substance screening:The stock cultures ar...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM21220((2S,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-N-ethyl-3,...)
Affinity DataEC50:  0.437nMAssay Description:Agonist activity at human A1AR expressed in FlpIn-CHO cells assessed as intracellular calcium mobilization by Fluo-4 dye-based fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM191801(US9187428, 29)
Affinity DataEC50:  0.5nMpH: 7.4 T: 2°CAssay Description:The following test protocol is used for pharmacologically characterizing cells and for the robot-assisted substance screening:The stock cultures ar...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM191810(US9187428, 38)
Affinity DataEC50:  0.5nMpH: 7.4 T: 2°CAssay Description:The following test protocol is used for pharmacologically characterizing cells and for the robot-assisted substance screening:The stock cultures ar...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM191844(US9187428, 72)
Affinity DataEC50:  0.5nMpH: 7.4 T: 2°CAssay Description:The following test protocol is used for pharmacologically characterizing cells and for the robot-assisted substance screening:The stock cultures ar...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM191857(US9187428, 85)
Affinity DataEC50:  0.5nMpH: 7.4 T: 2°CAssay Description:The following test protocol is used for pharmacologically characterizing cells and for the robot-assisted substance screening:The stock cultures ar...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM191822(US9187428, 50)
Affinity DataEC50:  0.5nMpH: 7.4 T: 2°CAssay Description:The following test protocol is used for pharmacologically characterizing cells and for the robot-assisted substance screening:The stock cultures ar...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM21220((2S,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-N-ethyl-3,...)
Affinity DataEC50:  0.501nMAssay Description:Irreversible agonist activity at human adenosine A1 receptor expressed in Flp-In-CHO cells assessed as stimulation of ERK1/2 phosphorylation incubate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM50588463(CHEMBL5174429)
Affinity DataEC50:  0.525nMAssay Description:Agonist activity at human adenosine A1 receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM50588453(CHEMBL5201013)
Affinity DataEC50:  0.525nMAssay Description:Agonist activity at human adenosine A1 receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
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