Compile Data Set for Download or QSAR
maximum 50k data
Found 15 of ic50 data for polymerid = 2436
TargetCalpain-1 catalytic subunit(Sus scrofa (pig))
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50114340((S)-2-(4-Fluoro-benzenesulfonylamino)-N-((S)-1-for...)
Affinity DataIC50:  35nMAssay Description:Tested for inhibitory activity against porcine erythrocyte Mu-calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Sus scrofa (pig))
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50114336((S)-2-(4-Fluoro-benzenesulfonylamino)-N-{(S)-1-[(2...)
Affinity DataIC50:  190nMAssay Description:Tested for inhibitory activity against porcine erythrocyte Mu-calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Sus scrofa (pig))
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50114342((E)-2-(dimethylamino)-N'-((S)-2-((S)-2-(4-fluoroph...)
Affinity DataIC50:  370nMAssay Description:Tested for inhibitory activity against porcine erythrocyte Mu-calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Sus scrofa (pig))
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50114341((2S)-N-((1S)-1-{(E)-[(aminocarbonyl)hydrazono]meth...)
Affinity DataIC50:  680nMAssay Description:Tested for inhibitory activity against porcine erythrocyte Mu-calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Sus scrofa (pig))
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50114337((S)-2-(4-Fluoro-benzenesulfonylamino)-3-methyl-N-{...)
Affinity DataIC50:  790nMAssay Description:Tested for inhibitory activity against porcine erythrocyte Mu-calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Sus scrofa (pig))
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50114339((S)-2-(4-Fluoro-benzenesulfonylamino)-3-methyl-N-{...)
Affinity DataIC50:  6.20E+3nMAssay Description:Tested for inhibitory activity against porcine erythrocyte Mu-calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Sus scrofa (pig))
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50363928(CHEMBL1951575)
Affinity DataIC50:  7.50E+3nMAssay Description:Inhibition of full length porcine Calpain-1 complex using (H2NeK(-FAM)-EVYGMMK(DABCYL)eOH) substrate by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Sus scrofa (pig))
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50114338((S)-N-{2-[(2-Dimethylamino-acetyl)-hydrazono]-ethy...)
Affinity DataIC50: >1.00E+4nMAssay Description:Tested for inhibitory activity against porcine erythrocyte Mu-calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Sus scrofa (pig))
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50466172(CHEMBL366254 | PD-150606)
Affinity DataIC50:  1.78E+4nMAssay Description:Inhibition of porcine Calpain-1 active site domain using (H2NeK(-FAM)-EVYGMMK(DABCYL)eOH) substrate by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Sus scrofa (pig))
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50466172(CHEMBL366254 | PD-150606)
Affinity DataIC50:  1.93E+4nMAssay Description:Inhibition of full length porcine Calpain-1 complex using (H2NeK(-FAM)-EVYGMMK(DABCYL)eOH) substrate by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Sus scrofa (pig))
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50466175(CHEMBL4289886)
Affinity DataIC50:  2.05E+4nMAssay Description:Inhibition of full length porcine Calpain-1 complex using (H2NeK(-FAM)-EVYGMMK(DABCYL)eOH) substrate by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Sus scrofa (pig))
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50466174(CHEMBL4293475)
Affinity DataIC50:  2.97E+4nMAssay Description:Inhibition of full length porcine Calpain-1 complex using (H2NeK(-FAM)-EVYGMMK(DABCYL)eOH) substrate by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Sus scrofa (pig))
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50466173(CHEMBL4288775)
Affinity DataIC50:  4.11E+4nMAssay Description:Inhibition of porcine Calpain-1 active site domain using (H2NeK(-FAM)-EVYGMMK(DABCYL)eOH) substrate by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Sus scrofa (pig))
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50466173(CHEMBL4288775)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of full length porcine Calpain-1 complex using (H2NeK(-FAM)-EVYGMMK(DABCYL)eOH) substrate by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Sus scrofa (pig))
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50363928(CHEMBL1951575)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of porcine Calpain-1 active site domain using (H2NeK(-FAM)-EVYGMMK(DABCYL)eOH) substrate by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed