TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)
Curated by ChEMBL
Institute Genomics Functional (Igf)
Curated by ChEMBL
Affinity DataKi: 0.0320nMAssay Description:Inhibition of human vasopressin V1a receptor expressed in CHO cells by polarisation binding assay using 384-well plate membranesMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)
Curated by ChEMBL
Institute Genomics Functional (Igf)
Curated by ChEMBL
Affinity DataKi: 0.0360nMAssay Description:Inhibition of human vasopressin V1a receptor expressed in CHO cells by polarisation binding assay using 96-well plate membranesMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)
Curated by ChEMBL
Institute Genomics Functional (Igf)
Curated by ChEMBL
Affinity DataKi: 0.0372nMAssay Description:Displacement of [3H]AVP from human V1A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)
Curated by ChEMBL
Institute Genomics Functional (Igf)
Curated by ChEMBL
Affinity DataKi: 0.0398nMAssay Description:Displacement of [3H]AVP from human V1A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)
Curated by ChEMBL
Institute Genomics Functional (Igf)
Curated by ChEMBL
Affinity DataKi: 0.0500nMAssay Description:Displacement [3H]Arg human recombinant Vasopressin V1a receptorMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)
Curated by ChEMBL
Institute Genomics Functional (Igf)
Curated by ChEMBL
Affinity DataKi: 0.0600nMAssay Description:Displacement [3H]Arg human recombinant Vasopressin V1a receptorMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)
Curated by ChEMBL
Institute Genomics Functional (Igf)
Curated by ChEMBL
Affinity DataKi: 0.0630nMAssay Description:The human V1a receptor was cloned by RT-PCR from total human liver RNA. The coding sequence was subcloned in an expression vector after sequencing to...More data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)
Curated by ChEMBL
Institute Genomics Functional (Igf)
Curated by ChEMBL
Affinity DataKi: 0.0700nMAssay Description:Displacement of [125I]- HO-LVA from human Vasopressin V1a receptor in membranes of CHO cellsMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)
Curated by ChEMBL
Institute Genomics Functional (Igf)
Curated by ChEMBL
Affinity DataKi: 0.0800nMAssay Description:Displacement of [125I]- HO-LVA from human Vasopressin V1a receptor in membranes of CHO cellsMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)
Curated by ChEMBL
Institute Genomics Functional (Igf)
Curated by ChEMBL
Affinity DataKi: 0.0900nMAssay Description:Displacement of [3H]AVP from human vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)
Curated by ChEMBL
Institute Genomics Functional (Igf)
Curated by ChEMBL
Affinity DataKi: 0.0955nMAssay Description:Displacement of [3H]AVP from human V1A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)
Curated by ChEMBL
Institute Genomics Functional (Igf)
Curated by ChEMBL
Affinity DataKi: 0.100nMAssay Description:Displacement [3H]Arg human recombinant Vasopressin V1a receptorMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)
Curated by ChEMBL
Institute Genomics Functional (Igf)
Curated by ChEMBL
Affinity DataKi: 0.170nMAssay Description:Displacement of [125I]- HO-LVA from human Vasopressin V1a receptor in membranes of CHO cellsMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)
Curated by ChEMBL
Institute Genomics Functional (Igf)
Curated by ChEMBL
Affinity DataKi: 0.170nMAssay Description:Displacement of [125I]- HO-LVA from human Vasopressin V1a receptor in membranes of CHO cellsMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)
Curated by ChEMBL
Institute Genomics Functional (Igf)
Curated by ChEMBL
Affinity DataKi: 0.182nMAssay Description:Displacement of [3H]AVP from human V1A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)
Curated by ChEMBL
Institute Genomics Functional (Igf)
Curated by ChEMBL
Affinity DataKi: 0.190nMAssay Description:Inhibition of human vasopressin V1a receptor expressed in COS7 cells by HTRF-FRET assay using 96-well plate membranesMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)
Curated by ChEMBL
Institute Genomics Functional (Igf)
Curated by ChEMBL
Affinity DataKi: 0.200nMAssay Description:Binding affinity for human cloned vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)
Curated by ChEMBL
Institute Genomics Functional (Igf)
Curated by ChEMBL
Affinity DataKi: 0.200nMAssay Description:The human V1a receptor was cloned by RT-PCR from total human liver RNA. The coding sequence was subcloned in an expression vector after sequencing to...More data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)
Curated by ChEMBL
Institute Genomics Functional (Igf)
Curated by ChEMBL
Affinity DataKi: 0.200nMAssay Description:Displacement of [Se-Se]-AVP from human V1A receptor expressed in CHO cells after 4 hrs by RP-LC-ICPMS analysisMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)
Curated by ChEMBL
Institute Genomics Functional (Igf)
Curated by ChEMBL
Affinity DataKi: 0.209nMAssay Description:Displacement of [3H]AVP from human V1A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)
Curated by ChEMBL
Institute Genomics Functional (Igf)
Curated by ChEMBL
Affinity DataKi: 0.209nMAssay Description:Displacement of [3H]AVP from human V1A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)
Curated by ChEMBL
Institute Genomics Functional (Igf)
Curated by ChEMBL
Affinity DataKi: 0.210nMAssay Description:Inhibition of human vasopressin V1a receptor expressed in COS7 cells by HTRF-FRET assay using 384-well plate membranesMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)
Curated by ChEMBL
Institute Genomics Functional (Igf)
Curated by ChEMBL
Affinity DataKi: 0.210nMAssay Description:Inhibition of human vasopressin V1a receptor expressed in COS7 cells by HTRF-FRET assay using 96-well plate membranesMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)
Curated by ChEMBL
Institute Genomics Functional (Igf)
Curated by ChEMBL
Affinity DataKi: 0.230nMAssay Description:Displacement of [125I]- HO-LVA from human Vasopressin V1a receptor in membranes of CHO cellsMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)
Curated by ChEMBL
Institute Genomics Functional (Igf)
Curated by ChEMBL
Affinity DataKi: 0.234nMAssay Description:Displacement of [3H]AVP from human V1A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)
Curated by ChEMBL
Institute Genomics Functional (Igf)
Curated by ChEMBL
Affinity DataKi: 0.234nMAssay Description:Displacement of [3H]AVP from human V1A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)
Curated by ChEMBL
Institute Genomics Functional (Igf)
Curated by ChEMBL
Affinity DataKi: 0.240nMAssay Description:Displacement of [3H]AVP from human V1A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)
Curated by ChEMBL
Institute Genomics Functional (Igf)
Curated by ChEMBL
Affinity DataKi: 0.251nMAssay Description:Displacement of [3H]AVP from human V1A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)
Curated by ChEMBL
Institute Genomics Functional (Igf)
Curated by ChEMBL
Affinity DataKi: 0.270nMAssay Description:Binding affinity for human cloned vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)
Curated by ChEMBL
Institute Genomics Functional (Igf)
Curated by ChEMBL
Affinity DataKi: 0.280nMAssay Description:Inhibition of human vasopressin V1a receptor expressed in COS7 cells by HTRF-FRET assay using 96-well plate cellsMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)
Curated by ChEMBL
Institute Genomics Functional (Igf)
Curated by ChEMBL
Affinity DataKi: 0.300nMAssay Description:Displacement of [3H]-arginine-vasopressin from human V1A receptor expressed in human 1321N1 cell membranes incubated for 60 mins by radioligand bindi...More data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)
Curated by ChEMBL
Institute Genomics Functional (Igf)
Curated by ChEMBL
Affinity DataKi: 0.300nMAssay Description:Displacement of [3H]-arginine-vasopressin from human V1A receptor expressed in human 1321N1 cell membranes incubated for 60 mins by radioligand bindi...More data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)
Curated by ChEMBL
Institute Genomics Functional (Igf)
Curated by ChEMBL
Affinity DataKi: 0.300nMAssay Description:Binding affinity for human cloned vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)
Curated by ChEMBL
Institute Genomics Functional (Igf)
Curated by ChEMBL
Affinity DataKi: 0.300nMAssay Description:Displacement of [3H]-arginine-vasopressin from human V1A receptor expressed in human 1321N1 cell membranes incubated for 60 mins by radioligand bindi...More data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)
Curated by ChEMBL
Institute Genomics Functional (Igf)
Curated by ChEMBL
Affinity DataKi: 0.300nMAssay Description:Displacement of [3H]-AVP from human V1A receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)
Curated by ChEMBL
Institute Genomics Functional (Igf)
Curated by ChEMBL
Affinity DataKi: 0.310nMAssay Description:Displacement [3H]Arg human recombinant Vasopressin V1a receptorMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)
Curated by ChEMBL
Institute Genomics Functional (Igf)
Curated by ChEMBL
Affinity DataKi: 0.316nMAssay Description:The human V1a receptor was cloned by RT-PCR from total human liver RNA. The coding sequence was subcloned in an expression vector after sequencing to...More data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)
Curated by ChEMBL
Institute Genomics Functional (Igf)
Curated by ChEMBL
Affinity DataKi: 0.370nMAssay Description:Displacement [3H]Arg human recombinant Vasopressin V1a receptorMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)
Curated by ChEMBL
Institute Genomics Functional (Igf)
Curated by ChEMBL
Affinity DataKi: 0.372nMAssay Description:Displacement of [3H]AVP from human V1A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)
Curated by ChEMBL
Institute Genomics Functional (Igf)
Curated by ChEMBL
Affinity DataKi: 0.372nMAssay Description:Displacement of [3H]AVP from human V1A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)
Curated by ChEMBL
Institute Genomics Functional (Igf)
Curated by ChEMBL
Affinity DataKi: 0.380nMAssay Description:Binding affinity for human cloned vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)
Curated by ChEMBL
Institute Genomics Functional (Igf)
Curated by ChEMBL
Affinity DataKi: 0.398nM ΔG°: -12.8kcal/moleT: 2°CAssay Description:The human V1a receptor was cloned by RT-PCR from total human liver RNA. The coding sequence was subcloned in an expression vector after sequencing to...More data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)
Curated by ChEMBL
Institute Genomics Functional (Igf)
Curated by ChEMBL
Affinity DataKi: 0.398nM ΔG°: -12.8kcal/moleT: 2°CAssay Description:The human V1a receptor was cloned by RT-PCR from total human liver RNA. The coding sequence was subcloned in an expression vector after sequencing to...More data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)
Curated by ChEMBL
Institute Genomics Functional (Igf)
Curated by ChEMBL
Affinity DataKi: 0.398nMAssay Description:The human V1a receptor was cloned by RT-PCR from total human liver RNA. The coding sequence was subcloned in an expression vector after sequencing to...More data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)
Curated by ChEMBL
Institute Genomics Functional (Igf)
Curated by ChEMBL
Affinity DataKi: 0.400nMAssay Description:Displacement of [3H]-arginine-vasopressin from human V1A receptor expressed in human 1321N1 cell membranes incubated for 60 mins by radioligand bindi...More data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)
Curated by ChEMBL
Institute Genomics Functional (Igf)
Curated by ChEMBL
Affinity DataKi: 0.400nMAssay Description:Displacement of [Se-Se]-AVP from human V1A receptor expressed in CHO cells after 4 hrs by RP-LC-ICPMS analysisMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)
Curated by ChEMBL
Institute Genomics Functional (Igf)
Curated by ChEMBL
Affinity DataKi: 0.410nMAssay Description:Binding affinity for human cloned vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)
Curated by ChEMBL
Institute Genomics Functional (Igf)
Curated by ChEMBL
Affinity DataKi: 0.430nMAssay Description:Displacement [3H]Arg human recombinant Vasopressin V1a receptorMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)
Curated by ChEMBL
Institute Genomics Functional (Igf)
Curated by ChEMBL
Affinity DataKi: 0.450nMAssay Description:Displacement of [3H]AVP from human V1a receptor expressed in 1132N1 cells assessed as dissociation constant by radioligand binding assayMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)
Curated by ChEMBL
Institute Genomics Functional (Igf)
Curated by ChEMBL
Affinity DataKi: 0.460nMAssay Description:Binding affinity for human cloned vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair