TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Affinity DataKi: 0.0150nMAssay Description:Competitive binding assay against Dopamine receptor D2 in rat striatal membranes and [125I]-IBF radioligandMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Affinity DataKi: 0.0170nMAssay Description:Inhibition of [125I]- NCQ 298 binding to D2 receptor of rat striatal tissueMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Affinity DataKi: 0.0180nMAssay Description:Inhibition of [3H]raclopride binding to rat striatal dopamine receptor D2More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Affinity DataKi: 0.0190nMAssay Description:Inhibition constant against dopamine receptor D2 in ratMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Affinity DataKi: 0.0200nMAssay Description:Inhibition of [125I]- NCQ 298 binding to D2 receptor of rat striatal tissueMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Affinity DataKi: 0.0200nMAssay Description:Inhibition constant against dopamine receptor D2 in ratMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Affinity DataKi: 0.0230nMAssay Description:Displacement of [3H]-spiperone from dopamine receptor D2More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Affinity DataKi: 0.0230nMAssay Description:Inhibition of [3H]spiperone binding to rat striatal membrane Dopamine receptor D2More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Affinity DataKi: 0.0230nMAssay Description:Displacement of [3H]-spiperone from dopamine receptor D2More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Affinity DataKi: 0.0240nMAssay Description:Inhibition of [3H]raclopride binding to rat striatal dopamine receptor D2More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Affinity DataKi: 0.0250nMAssay Description:Inhibition constant against dopamine receptor D2 in ratMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Affinity DataKi: 0.0280nMAssay Description:Inhibition of [125I]- NCQ 298 binding to D2 receptor of rat striatal tissueMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Affinity DataKi: 0.0290nMAssay Description:Displacement of [3H]-spiperone from dopamine receptor D2More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Affinity DataKi: 0.0330nMAssay Description:Inhibition of [3H]spiperone binding to rat striatal membrane Dopamine receptor D2More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Affinity DataKi: 0.0330nMAssay Description:Inhibition of [125I]- NCQ 298 binding to D2 receptor of rat striatal tissueMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Affinity DataKi: 0.0330nMAssay Description:Displacement of [3H]-spiperone from dopamine receptor D2More data for this Ligand-Target Pair
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Rattus norvegicus (rat))
Northeastern University
Curated by ChEMBL
Northeastern University
Curated by ChEMBL
Affinity DataKi: 0.0340nMAssay Description:Compound was evaluated for its ability to inhibit Striatal Dopamine Receptor in rat brain through radioreceptor assay carried out with agonist ligand...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Affinity DataKi: 0.0350nMAssay Description:Displacement of [3H]-spiperone from dopamine receptor D2More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Affinity DataKi: 0.0360nMAssay Description:Inhibition of [125I]- NCQ 298 binding to D2 receptor of rat striatal tissueMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Affinity DataKi: 0.0360nMAssay Description:Displacement of [3H]-spiperone from dopamine receptor D2More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Affinity DataKi: 0.0380nMAssay Description:Inhibition of [125I]- NCQ 298 binding to D2 receptor of rat striatal tissueMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Affinity DataKi: 0.0390nMAssay Description:Displacement of [3H]-spiperone from dopamine receptor D2More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Affinity DataKi: 0.0430nMAssay Description:Displacement of [3H]-spiperone from dopamine receptor D2More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Affinity DataKi: 0.0450nMAssay Description:Binding affinity of compound against Dopamine receptor D2 binding site using radioligand [3H]spiperoneMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Affinity DataKi: 0.0470nMAssay Description:Binding affinity towards Dopamine receptor D2 by displacing [3H]-spiperoneMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Affinity DataKi: 0.0500nMAssay Description:Binding affinity for dopamine receptor D2 long expressed in Sf9 cells using [125I]-IABN radioligand.More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Affinity DataKi: 0.0530nMAssay Description:Displacement of [3H]raclopride from rat dopamine D2 receptorMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Affinity DataKi: 0.0530nMAssay Description:Binding affinity at rat striatal Dopamine receptor D2 using [3H]- piperone radioligandMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Affinity DataKi: 0.0570nMAssay Description:Binding affinity towards Dopamine receptor D2 by displacing [3H]-spiperoneMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Affinity DataKi: 0.0580nMAssay Description:Displacement of [3H]-spiperone from dopamine receptor D2More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Affinity DataKi: 0.0600nMAssay Description:Binding affinity against D2 receptor in rat striatum using [3H]-RacloprideMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Affinity DataKi: 0.0620nMAssay Description:Displacement of [3H]-spiperone from dopamine receptor D2More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Affinity DataKi: 0.0630nMAssay Description:Binding affinity towards Dopamine receptor D2 by displacing [3H]-spiperoneMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Affinity DataKi: 0.0630nMAssay Description:Displacement of [3H]-spiperone from dopamine receptor D2More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Affinity DataKi: 0.0640nMAssay Description:Inhibition of [3H]raclopride binding to rat striatal dopamine receptor D2More data for this Ligand-Target Pair