Compile Data Set for Download or QSAR
maximum 50k data
Found 27 of kd for UniProtKB: A0A024R126
TargetNuclear receptor subfamily 4 group A member 1(Homo sapiens (Human))
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50570058(CHEMBL4867199)
Affinity DataKd:  33nMAssay Description:Binding affinity to recombinant human N-terminal His-tagged Nur77-LBD (367 to 598 residues) expressed in Escherichia coli BL21 DE3 by surface plasmon...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 4 group A member 1(Homo sapiens (Human))
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50570057(CHEMBL4857769)
Affinity DataKd:  36nMAssay Description:Binding affinity to recombinant human N-terminal His-tagged Nur77-LBD (367 to 598 residues) expressed in Escherichia coli BL21 DE3 by surface plasmon...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 4 group A member 1(Homo sapiens (Human))
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50570058(CHEMBL4867199)
Affinity DataKd:  66nMAssay Description:Binding affinity to recombinant human N-terminal His-tagged Nur77-LBD (367 to 598 residues) expressed in Escherichia coli BL21 DE3 by flourescence qu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 4 group A member 1(Homo sapiens (Human))
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50570057(CHEMBL4857769)
Affinity DataKd:  66nMAssay Description:Binding affinity to recombinant human N-terminal His-tagged Nur77-LBD (367 to 598 residues) expressed in Escherichia coli BL21 DE3 by flourescence qu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 4 group A member 1(Homo sapiens (Human))
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50570056(CHEMBL4877512)
Affinity DataKd:  110nMAssay Description:Binding affinity to recombinant human N-terminal His-tagged Nur77-LBD (367 to 598 residues) expressed in Escherichia coli BL21 DE3 by surface plasmon...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 4 group A member 1(Homo sapiens (Human))
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50570056(CHEMBL4877512)
Affinity DataKd:  217nMAssay Description:Binding affinity to recombinant human N-terminal His-tagged Nur77-LBD (367 to 598 residues) expressed in Escherichia coli BL21 DE3 by flourescence qu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 4 group A member 1(Homo sapiens (Human))
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50079524(CHEMBL3417313)
Affinity DataKd:  220nMAssay Description:Binding affinity to recombinant human N-terminal His-tagged Nur77 LBD (367 to 598 residues) expressed in Escherichia coli BL21(DE3) incubated for 30 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 4 group A member 1(Homo sapiens (Human))
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50524688(CHEMBL3980631)
Affinity DataKd:  270nMAssay Description:Binding affinity to recombinant human N-terminal His-tagged Nur77 LBD (367 to 598 residues) expressed in Escherichia coli BL21(DE3) incubated for 30 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 4 group A member 1(Homo sapiens (Human))
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50071058((2R,4aS,6aS,12bR,14aS,14bR)-10-Hydroxy-2,4a,6a,9,1...)
Affinity DataKd:  290nMAssay Description:Binding affinity to Nur77 LBD (unknown origin) expressed in Escherichia coli incubated for 3 hrs by circular dichroism analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 4 group A member 1(Homo sapiens (Human))
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50071058((2R,4aS,6aS,12bR,14aS,14bR)-10-Hydroxy-2,4a,6a,9,1...)
Affinity DataKd:  290nMAssay Description:Binding affinity to purified Nur77 LBD (unknown origin) by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 4 group A member 1(Homo sapiens (Human))
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50071058((2R,4aS,6aS,12bR,14aS,14bR)-10-Hydroxy-2,4a,6a,9,1...)
Affinity DataKd:  320nMAssay Description:Binding affinity to recombinant human N-terminal His-tagged Nur77 LBD (367 to 598 residues) expressed in Escherichia coli BL21(DE3) incubated for 30 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 4 group A member 1(Homo sapiens (Human))
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50524694(CHEMBL3892041)
Affinity DataKd:  520nMAssay Description:Binding affinity to recombinant human N-terminal His-tagged Nur77 LBD (367 to 598 residues) expressed in Escherichia coli BL21(DE3) incubated for 30 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 4 group A member 1(Homo sapiens (Human))
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50524693(CHEMBL4459092)
Affinity DataKd:  720nMAssay Description:Binding affinity to recombinant human N-terminal His-tagged Nur77 LBD (367 to 598 residues) expressed in Escherichia coli BL21(DE3) incubated for 30 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 4 group A member 1(Homo sapiens (Human))
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50378798(CYTOSPORONE B)
Affinity DataKd:  740nMAssay Description:Binding affinity to Nur77 receptor expressed in human BGC823 cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 4 group A member 1(Homo sapiens (Human))
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50079525(CHEMBL3417314)
Affinity DataKd:  800nMAssay Description:Binding affinity to recombinant human N-terminal His-tagged Nur77 LBD (367 to 598 residues) expressed in Escherichia coli BL21(DE3) incubated for 30 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 4 group A member 1(Homo sapiens (Human))
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50524687(CHEMBL3928971)
Affinity DataKd:  830nMAssay Description:Binding affinity to recombinant human N-terminal His-tagged Nur77 LBD (367 to 598 residues) expressed in Escherichia coli BL21(DE3) incubated for 30 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 4 group A member 1(Homo sapiens (Human))
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50481949(Dihydrocelastrol | acs.jmedchem.1c00409_ST.616)
Affinity DataKd:  870nMAssay Description:Binding affinity to recombinant human N-terminal His-tagged Nur77 LBD (367 to 598 residues) expressed in Escherichia coli BL21(DE3) incubated for 30 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 4 group A member 1(Homo sapiens (Human))
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50481947(CHEBI:8416 | GNF-Pf-476 | PRISTIMERIN | Pristimeri...)
Affinity DataKd:  960nMAssay Description:Binding affinity to recombinant human N-terminal His-tagged Nur77 LBD (367 to 598 residues) expressed in Escherichia coli BL21(DE3) incubated for 30 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 4 group A member 1(Homo sapiens (Human))
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50565399(CHEMBL4795792)
Affinity DataKd:  1.34E+3nMAssay Description:Binding affinity to Nur77 ligand binding domain (unknown origin) assessed as dissociation constant by fluorescence titration based analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 4 group A member 1(Homo sapiens (Human))
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50378798(CYTOSPORONE B)
Affinity DataKd:  1.51E+3nMAssay Description:Binding affinity to NuR77-LBD receptor expressed in human BGC823 cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 4 group A member 1(Homo sapiens (Human))
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50524691(CHEMBL4207143)
Affinity DataKd:  2.69E+3nMAssay Description:Binding affinity to recombinant human N-terminal His-tagged Nur77 LBD (367 to 598 residues) expressed in Escherichia coli BL21(DE3) incubated for 30 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 4 group A member 1(Homo sapiens (Human))
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50524686(CHEMBL4470378)
Affinity DataKd:  2.94E+3nMAssay Description:Binding affinity to recombinant human N-terminal His-tagged Nur77 LBD (367 to 598 residues) expressed in Escherichia coli BL21(DE3) incubated for 30 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 4 group A member 1(Homo sapiens (Human))
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50524695(CHEMBL4446742)
Affinity DataKd:  3.30E+3nMAssay Description:Binding affinity to recombinant human N-terminal His-tagged Nur77 LBD (367 to 598 residues) expressed in Escherichia coli BL21(DE3) incubated for 30 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 4 group A member 1(Homo sapiens (Human))
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50565399(CHEMBL4795792)
Affinity DataKd:  3.58E+3nMAssay Description:Binding affinity to Nur77 ligand binding domain (unknown origin) assessed as dissociation constant by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 4 group A member 1(Homo sapiens (Human))
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50524692(CHEMBL4470497)
Affinity DataKd:  3.80E+3nMAssay Description:Binding affinity to recombinant human N-terminal His-tagged Nur77 LBD (367 to 598 residues) expressed in Escherichia coli BL21(DE3) incubated for 30 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 4 group A member 1(Homo sapiens (Human))
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50524689(CHEMBL4451088)
Affinity DataKd:  4.13E+3nMAssay Description:Binding affinity to recombinant human N-terminal His-tagged Nur77 LBD (367 to 598 residues) expressed in Escherichia coli BL21(DE3) incubated for 30 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 4 group A member 1(Homo sapiens (Human))
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50524690(CHEMBL4463133)
Affinity DataKd:  5.56E+3nMAssay Description:Binding affinity to recombinant human N-terminal His-tagged Nur77 LBD (367 to 598 residues) expressed in Escherichia coli BL21(DE3) incubated for 30 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed