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Found 6799 of ki for UniProtKB: P35462
TargetD(3) dopamine receptor(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM476758(US10870660, Compound III-024 | US11345716, Compoun...)
Affinity DataKi:  0.0120nMAssay Description:225 nL of the solutions of the non-specific ligand or the compounds of the present invention at each concentration (in case of vehicle, final concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
TargetD(3) dopamine receptor(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM476758(US10870660, Compound III-024 | US11345716, Compoun...)
Affinity DataKi:  0.0120nMAssay Description:225 nL of the solutions of the non-specific ligand or the compounds of the present invention at each concentration (in case of vehicle, final concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(3) dopamine receptor(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM556452(US11345716, Compound II-057)
Affinity DataKi:  0.0140nMAssay Description:225 nL of the solutions of the non-specific ligand or the compounds of the present invention at each concentration (in case of vehicle, final concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
TargetD(3) dopamine receptor(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM476918(US10870660, Compound II-057)
Affinity DataKi:  0.0140nMAssay Description:225 nL of the solutions of the non-specific ligand or the compounds of the present invention at each concentration (in case of vehicle, final concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(3) dopamine receptor(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM50290221(CHEMBL80919 | Thiophene-2-carboxylic acid (4-{2-[4...)
Affinity DataKi:  0.0200nMAssay Description:Ability to displace radioligand [3H]N-0437 from human dopamine D2 receptor transfected chinese hamster ovary cell membranes.More data for this Ligand-Target Pair
In DepthDetails Article
TargetD(3) dopamine receptor(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM50063292(CHEMBL349426 | {4-[2-(4-Phenyl-piperazin-1-yl)-eth...)
Affinity DataKi:  0.0200nMAssay Description:Binding affinity determined by measuring displacement of [3H]-spiperone from cloned Human Dopamine receptor D3 in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM476915(US10870660, Compound II-047)
Affinity DataKi:  0.0220nMAssay Description:225 nL of the solutions of the non-specific ligand or the compounds of the present invention at each concentration (in case of vehicle, final concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(3) dopamine receptor(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM476863(US10870660, Compound II-046 | US11345716, Compound...)
Affinity DataKi:  0.0220nMAssay Description:225 nL of the solutions of the non-specific ligand or the compounds of the present invention at each concentration (in case of vehicle, final concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
TargetD(3) dopamine receptor(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM476764(US10870660, Compound III-064 | US11345716, Compoun...)
Affinity DataKi:  0.0260nMAssay Description:225 nL of the solutions of the non-specific ligand or the compounds of the present invention at each concentration (in case of vehicle, final concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
TargetD(3) dopamine receptor(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM476764(US10870660, Compound III-064 | US11345716, Compoun...)
Affinity DataKi:  0.0260nMAssay Description:225 nL of the solutions of the non-specific ligand or the compounds of the present invention at each concentration (in case of vehicle, final concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(3) dopamine receptor(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM50341508((S)-N-(4-(4-Phenylbenzoylamino)butyl)-N-propyl-5-a...)
Affinity DataKi:  0.0270nMAssay Description:Displacement of [3H]7-OH-DPAT from human dopamine D3 receptor expressed in CHO cells after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM50207116(CHEMBL3905247 | US9550741, I-4)
Affinity DataKi:  0.0290nMAssay Description:Displacement of [3H]methyl-spiperone from recombinant human D3 receptor expressed in CHO cell membranes after 60 mins by scintillation counting metho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM476836(US10870660, Compound III-581 | US11345716, Compoun...)
Affinity DataKi:  0.0350nMAssay Description:225 nL of the solutions of the non-specific ligand or the compounds of the present invention at each concentration (in case of vehicle, final concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(3) dopamine receptor(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM476836(US10870660, Compound III-581 | US11345716, Compoun...)
Affinity DataKi:  0.0350nMAssay Description:225 nL of the solutions of the non-specific ligand or the compounds of the present invention at each concentration (in case of vehicle, final concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
TargetD(3) dopamine receptor(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM50008735((+)-3-(tert-butyl)-(3S,4aS,13bS)-2,3,4,4a,8,9,13b,...)
Affinity DataKi:  0.0400nMAssay Description:Displacement of [3H]methylspiperone from human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM50008735((+)-3-(tert-butyl)-(3S,4aS,13bS)-2,3,4,4a,8,9,13b,...)
Affinity DataKi:  0.0400nMAssay Description:Displacement of [3H]methylspiperone from human recombinant D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM50207162(CHEMBL3918755 | US9550741, IV-1)
Affinity DataKi:  0.0430nMAssay Description:Displacement of [3H]methyl-spiperone from recombinant human D3 receptor expressed in CHO cell membranes after 60 mins by scintillation counting metho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM50207143(CHEMBL3966842 | US9550741, II-1)
Affinity DataKi:  0.0430nMAssay Description:Displacement of [3H]methyl-spiperone from recombinant human D3 receptor expressed in CHO cell membranes after 60 mins by scintillation counting metho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM50207155(CHEMBL3895540)
Affinity DataKi:  0.0460nMAssay Description:Displacement of [3H]methyl-spiperone from recombinant human D3 receptor expressed in CHO cell membranes after 60 mins by scintillation counting metho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM50207141(CHEMBL3920252)
Affinity DataKi:  0.0470nMAssay Description:Displacement of [3H]methyl-spiperone from recombinant human D3 receptor expressed in CHO cell membranes after 60 mins by scintillation counting metho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM476923(US10870660, Compound II-081 | US11345716, Compound...)
Affinity DataKi:  0.0480nMAssay Description:225 nL of the solutions of the non-specific ligand or the compounds of the present invention at each concentration (in case of vehicle, final concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
TargetD(3) dopamine receptor(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM476923(US10870660, Compound II-081 | US11345716, Compound...)
Affinity DataKi:  0.0480nMAssay Description:225 nL of the solutions of the non-specific ligand or the compounds of the present invention at each concentration (in case of vehicle, final concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(3) dopamine receptor(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM476834(US10870660, Compound III-578 | US11345716, Compoun...)
Affinity DataKi:  0.0500nMAssay Description:225 nL of the solutions of the non-specific ligand or the compounds of the present invention at each concentration (in case of vehicle, final concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(3) dopamine receptor(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM476834(US10870660, Compound III-578 | US11345716, Compoun...)
Affinity DataKi:  0.0500nMAssay Description:225 nL of the solutions of the non-specific ligand or the compounds of the present invention at each concentration (in case of vehicle, final concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
TargetD(3) dopamine receptor(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM50207148(CHEMBL3932186)
Affinity DataKi:  0.0510nMAssay Description:Displacement of [3H]methyl-spiperone from recombinant human D3 receptor expressed in CHO cell membranes after 60 mins by scintillation counting metho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM476858(US10870660, Compound III-706 | US11345716, Compoun...)
Affinity DataKi:  0.0510nMAssay Description:225 nL of the solutions of the non-specific ligand or the compounds of the present invention at each concentration (in case of vehicle, final concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(3) dopamine receptor(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM476858(US10870660, Compound III-706 | US11345716, Compoun...)
Affinity DataKi:  0.0510nMAssay Description:225 nL of the solutions of the non-specific ligand or the compounds of the present invention at each concentration (in case of vehicle, final concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
TargetD(3) dopamine receptor(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM476924(US10870660, Compound II-084 | US11345716, Compound...)
Affinity DataKi:  0.0520nMAssay Description:225 nL of the solutions of the non-specific ligand or the compounds of the present invention at each concentration (in case of vehicle, final concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
TargetD(3) dopamine receptor(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM50207154(CHEMBL3902496)
Affinity DataKi:  0.0520nMAssay Description:Displacement of [3H]methyl-spiperone from recombinant human D3 receptor expressed in CHO cell membranes after 60 mins by scintillation counting metho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM476924(US10870660, Compound II-084 | US11345716, Compound...)
Affinity DataKi:  0.0520nMAssay Description:225 nL of the solutions of the non-specific ligand or the compounds of the present invention at each concentration (in case of vehicle, final concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(3) dopamine receptor(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM50207113(CHEMBL3896937 | US9550741, IV-3)
Affinity DataKi:  0.0550nMAssay Description:Displacement of [3H]methyl-spiperone from recombinant human D3 receptor expressed in CHO cell membranes after 60 mins by scintillation counting metho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM50207094(CHEMBL3976282 | US9550741, I-2)
Affinity DataKi:  0.0560nMAssay Description:Displacement of [3H]methyl-spiperone from recombinant human D3 receptor expressed in CHO cell membranes after 60 mins by scintillation counting metho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM476773(US10870660, Compound III-138 | US11345716, Compoun...)
Affinity DataKi:  0.0570nMAssay Description:225 nL of the solutions of the non-specific ligand or the compounds of the present invention at each concentration (in case of vehicle, final concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(3) dopamine receptor(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM476773(US10870660, Compound III-138 | US11345716, Compoun...)
Affinity DataKi:  0.0570nMAssay Description:225 nL of the solutions of the non-specific ligand or the compounds of the present invention at each concentration (in case of vehicle, final concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
TargetD(3) dopamine receptor(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM50207150(CHEMBL3933256)
Affinity DataKi:  0.0580nMAssay Description:Displacement of [3H]methyl-spiperone from recombinant human D3 receptor expressed in CHO cell membranes after 60 mins by scintillation counting metho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM476914(US10870660, Compound II-041)
Affinity DataKi:  0.0580nMAssay Description:225 nL of the solutions of the non-specific ligand or the compounds of the present invention at each concentration (in case of vehicle, final concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(3) dopamine receptor(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM50207158(CHEMBL3982486 | US9550741, III-2)
Affinity DataKi:  0.0580nMAssay Description:Displacement of [3H]methyl-spiperone from recombinant human D3 receptor expressed in CHO cell membranes after 60 mins by scintillation counting metho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM556448(US11345716, Compound II-041)
Affinity DataKi:  0.0580nMAssay Description:225 nL of the solutions of the non-specific ligand or the compounds of the present invention at each concentration (in case of vehicle, final concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
TargetD(3) dopamine receptor(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM476925(US10870660, Compound II-087)
Affinity DataKi:  0.0590nMAssay Description:225 nL of the solutions of the non-specific ligand or the compounds of the present invention at each concentration (in case of vehicle, final concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(3) dopamine receptor(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM476863(US10870660, Compound II-046 | US11345716, Compound...)
Affinity DataKi:  0.0590nMAssay Description:225 nL of the solutions of the non-specific ligand or the compounds of the present invention at each concentration (in case of vehicle, final concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
TargetD(3) dopamine receptor(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM50207115(CHEMBL3948056)
Affinity DataKi:  0.0620nMAssay Description:Displacement of [3H]methyl-spiperone from recombinant human D3 receptor expressed in CHO cell membranes after 60 mins by scintillation counting metho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM476759(US10870660, Compound III-027 | US11345716, Compoun...)
Affinity DataKi:  0.0640nMAssay Description:225 nL of the solutions of the non-specific ligand or the compounds of the present invention at each concentration (in case of vehicle, final concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
TargetD(3) dopamine receptor(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM476759(US10870660, Compound III-027 | US11345716, Compoun...)
Affinity DataKi:  0.0640nMAssay Description:225 nL of the solutions of the non-specific ligand or the compounds of the present invention at each concentration (in case of vehicle, final concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(3) dopamine receptor(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM476866(US10870660, Compound II-053 | US11345716, Compound...)
Affinity DataKi:  0.0670nMAssay Description:225 nL of the solutions of the non-specific ligand or the compounds of the present invention at each concentration (in case of vehicle, final concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
TargetD(3) dopamine receptor(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM476866(US10870660, Compound II-053 | US11345716, Compound...)
Affinity DataKi:  0.0670nMAssay Description:225 nL of the solutions of the non-specific ligand or the compounds of the present invention at each concentration (in case of vehicle, final concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(3) dopamine receptor(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM50192240(CHEMBL3941818 | US10239870, Example 278)
Affinity DataKi:  0.0676nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO-K1 cell membranes after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM50192240(CHEMBL3941818 | US10239870, Example 278)
Affinity DataKi:  0.0700nMAssay Description:Antagonist activity at human dopamine D3 receptor expressed in CHO cell membranes after 90 mins in presence of quinelorane by [35S]-GTPgammaS binding...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM50192240(CHEMBL3941818 | US10239870, Example 278)
Affinity DataKi:  0.0700nMAssay Description:Antagonist activity at human dopamine D3 receptor expressed in CHO cell membranes after 90 mins in presence of quinelorane by [35S]-GTPgammaS binding...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM476922(US10870660, Compound II-078 | US11345716, Compound...)
Affinity DataKi:  0.0750nMAssay Description:225 nL of the solutions of the non-specific ligand or the compounds of the present invention at each concentration (in case of vehicle, final concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
TargetD(3) dopamine receptor(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM476922(US10870660, Compound II-078 | US11345716, Compound...)
Affinity DataKi:  0.0750nMAssay Description:225 nL of the solutions of the non-specific ligand or the compounds of the present invention at each concentration (in case of vehicle, final concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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