Compile Data Set for Download or QSAR
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Found 190 of ki for UniProtKB: P28565
Target5-hydroxytryptamine receptor 1D(RAT)
University Of Alberta

Curated by PDSP Ki Database
LigandPNGBDBM50280055(50285557 | 7-Methyl-4,6,6a,7,8,9,10,10a-octahydro-...)
Affinity DataKi:  0.0600nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1D(RAT)
University Of Alberta

Curated by PDSP Ki Database
LigandPNGBDBM50027065((5'alpha)-12'-hydroxy-2'-methyl-5'-(phenylmethyl)e...)
Affinity DataKi:  0.0700nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1D(RAT)
University Of Alberta

Curated by PDSP Ki Database
LigandPNGBDBM21392(3-(2-aminoethyl)-1H-indole-5-carboxamide | 5-CT | ...)
Affinity DataKi:  0.370nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1D(RAT)
University Of Alberta

Curated by PDSP Ki Database
LigandPNGBDBM78940(METHIOTHEPIN | MLS000859918 | Methiothepin mesylat...)
Affinity DataKi:  0.580nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1D(RAT)
University Of Alberta

Curated by PDSP Ki Database
LigandPNGBDBM30704((phenylmethyl) N-[[(6aR,9S,10aR)-4,7-dimethyl-6,6a...)
Affinity DataKi:  0.770nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1D(RAT)
University Of Alberta

Curated by PDSP Ki Database
LigandPNGBDBM30712(6-tert-butyl-3-(2-imidazolin-2-ylmethyl)-2,4-dimet...)
Affinity DataKi:  1.28nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM10755(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Affinity DataKi:  2nMAssay Description:Evaluated for binding affinity towards rat cortical membranes at 5-hydroxytryptamine 1 receptor binding site by using [3H]-5-HT as a radioligand.More data for this Ligand-Target Pair
LigandPNGBDBM82087(2-(5-methoxy-1H-indol-3-yl)ethanamine | 5-MT | 5-M...)
Affinity DataKi:  2nMAssay Description:Evaluated for binding affinity towards rat cortical membranes at 5-hydroxytryptamine 1 receptor binding site by using [3H]-5-HT as a radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM81498(5-Methoxy-3-(1,2,3,6-tetrahydro-pyridin-4-yl)-1H-i...)
Affinity DataKi:  2nMAssay Description:Evaluated for binding affinity towards rat cortical membranes at 5-hydroxytryptamine 1 receptor binding site by using [3H]-5-HT as a radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1D(RAT)
University Of Alberta

Curated by PDSP Ki Database
LigandPNGBDBM82087(2-(5-methoxy-1H-indol-3-yl)ethanamine | 5-MT | 5-M...)
Affinity DataKi:  2.39nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1D(RAT)
University Of Alberta

Curated by PDSP Ki Database
LigandPNGBDBM10755(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Affinity DataKi:  2.51nMMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1D(RAT)
University Of Alberta

Curated by PDSP Ki Database
LigandPNGBDBM81497(4-(4-Methyl-piperazin-1-yl)-7-trifluoromethyl-pyrr...)
Affinity DataKi:  4.89nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50007407(1-NP | 1-Naphthalen-1-yl-piperazine | 4-Naphthalen...)
Affinity DataKi:  5nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1 receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50026968(9-Chloro-11-(1-methyl-piperidin-4-ylidene)-11H-ben...)
Affinity DataKi:  7.60nMAssay Description:Displacement of [3H]LSD radioligand binding at the serotonin-1 binding site of rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50026974(9-Bromo-11-(1-methyl-piperidin-4-ylidene)-6,11-dih...)
Affinity DataKi:  7.80nMAssay Description:Displacement of [3H]LSD radioligand binding at the serotonin-1 binding site of rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50026970(9-Chloro-11-(1-methyl-piperidin-4-ylidene)-6,11-di...)
Affinity DataKi:  8.20nMAssay Description:Displacement of [3H]LSD radioligand binding at the serotonin-1 binding site of rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50026964(9-Bromo-11-(1-methyl-piperidin-4-ylidene)-11H-benz...)
Affinity DataKi:  8.70nMAssay Description:Displacement of [3H]LSD radioligand binding at the serotonin-1 binding site of rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1D(RAT)
University Of Alberta

Curated by PDSP Ki Database
LigandPNGBDBM50005835((3-[2-(dimethylamino)ethyl]-1H-indol-5-yl)-N-methy...)
Affinity DataKi:  9.54nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1D(RAT)
University Of Alberta

Curated by PDSP Ki Database
LigandPNGBDBM50217230(CHEMBL95387)
Affinity DataKi:  10nMAssay Description:Binding affinity to 5-hydroxytryptamine 1D receptor in the rat forebrain by [3H]- SB-204269 displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1D(RAT)
University Of Alberta

Curated by PDSP Ki Database
LigandPNGBDBM50217225(CHEMBL98434)
Affinity DataKi:  10nMAssay Description:Binding affinity to 5-hydroxytryptamine 1D receptor in the rat forebrain by [3H]- SB-204269 displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50026971(11-(1-Methyl-piperidin-4-ylidene)-11H-benzo[d]pyrr...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]LSD radioligand binding at the serotonin-1 binding site of rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1D(RAT)
University Of Alberta

Curated by PDSP Ki Database
LigandPNGBDBM50217226(CHEMBL318906)
Affinity DataKi:  13nMAssay Description:Binding affinity to 5-hydroxytryptamine 1D receptor in the rat forebrain by [3H]- SB-204269 displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1D(RAT)
University Of Alberta

Curated by PDSP Ki Database
LigandPNGBDBM50217210(CHEMBL38918)
Affinity DataKi:  13nMAssay Description:Binding affinity to 5-hydroxytryptamine 1D receptor in the rat forebrain by [3H]- SB-204269 displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50026972(11-(1-Methyl-piperidin-4-ylidene)-11H-benzo[d]pyrr...)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]LSD radioligand binding at the serotonin-1 binding site of rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50026963(11-(1-Methyl-piperidin-4-ylidene)-6,11-dihydro-5H-...)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]LSD radioligand binding at the serotonin-1 binding site of rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1D(RAT)
University Of Alberta

Curated by PDSP Ki Database
LigandPNGBDBM50217211(CHEMBL318022)
Affinity DataKi:  16nMAssay Description:Binding affinity to 5-hydroxytryptamine 1D receptor in the rat forebrain by [3H]- SB-204269 displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1D(RAT)
University Of Alberta

Curated by PDSP Ki Database
LigandPNGBDBM50217182(CHEMBL318882)
Affinity DataKi:  16nMAssay Description:Binding affinity to 5-hydroxytryptamine 1D receptor in the rat forebrain by [3H]- SB-204269 displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50017453(1-(2-Ethyl-phenyl)-piperazine | CHEMBL9467)
Affinity DataKi:  17nMAssay Description:Binding affinity determined in radioreceptor binding assay by using [3H]5-HT radioligand against 5-hydroxytryptamine 1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50001855(1-{5-[4-(2-Isopropoxy-phenyl)-piperazin-1-ylmethyl...)
Affinity DataKi:  18nMAssay Description:The compound was tested for its binding affinity towards 5-hydroxytryptamine 1 receptor by displacing [3H]5-HT radioligand in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50026973(11-(1-Methyl-piperidin-4-ylidene)-9-trifluoromethy...)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]LSD radioligand binding at the serotonin-1 binding site of rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1D(RAT)
University Of Alberta

Curated by PDSP Ki Database
LigandPNGBDBM10755(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Affinity DataKi:  18nMMore data for this Ligand-Target Pair
LigandPNGBDBM50017460(1-(2-Butoxy-phenyl)-piperazine | CHEMBL9452)
Affinity DataKi:  19nMAssay Description:Inhibition of [3H]5-HT radioligand binding against 5-hydroxytryptamine 1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50017448(1-(2-Isopropoxy-phenyl)-piperazine | CHEMBL9669)
Affinity DataKi:  19nMAssay Description:Inhibition of [3H]5-HT radioligand binding against 5-hydroxytryptamine 1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1D(RAT)
University Of Alberta

Curated by PDSP Ki Database
LigandPNGBDBM50217231(CHEMBL98433)
Affinity DataKi:  20nMAssay Description:Binding affinity to 5-hydroxytryptamine 1D receptor in the rat forebrain by [3H]- SB-204269 displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM30704((phenylmethyl) N-[[(6aR,9S,10aR)-4,7-dimethyl-6,6a...)
Affinity DataKi:  20nMAssay Description:Evaluated for binding affinity towards rat cortical membranes at 5-hydroxytryptamine 1 receptor binding site by using [3H]-5-HT as a radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50007406(1-(3-(trifluoromethyl)phenyl)piperazine | 1-(3-Tri...)
Affinity DataKi:  20nMAssay Description:Evaluated for binding affinity towards rat cortical membranes at 5-hydroxytryptamine 1 receptor binding site by using [3H]-5-HT as a radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50007406(1-(3-(trifluoromethyl)phenyl)piperazine | 1-(3-Tri...)
Affinity DataKi:  20nMAssay Description:Binding affinity in radioreceptor binding assay by using [3H]5-HT radioligand against 5-hydroxytryptamine 1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50017450(1-(2-Isopropyl-phenyl)-piperazine | CHEMBL276156)
Affinity DataKi:  23nMAssay Description:Binding affinity determined in radioreceptor binding assay by using [3H]5-HT radioligand against 5-hydroxytryptamine 1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50026967(11-(1-Methyl-piperidin-4-ylidene)-9-trifluoromethy...)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]LSD radioligand binding at the serotonin-1 binding site of rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50001901(1-(2-Chloro-phenyl)-piperazine | CHEMBL9841)
Affinity DataKi:  24nMAssay Description:Binding affinity in radioreceptor binding assay by using [3H]5-HT radioligand against 5-hydroxytryptamine 1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50001915(1-(3-chlorophenyl)piperazine | CHEMBL478 | m-Chlor...)
Affinity DataKi:  25nMAssay Description:Inhibition of [3H]5-HT radioligand binding against 5-hydroxytryptamine 1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50026969(11-(1-Methyl-piperidin-4-ylidene)-6,11-dihydro-5H-...)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]LSD radioligand binding at the serotonin-1 binding site of rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50017458(2-Piperazin-1-yl-benzonitrile | CHEMBL275943)
Affinity DataKi:  26nMAssay Description:Inhibition of [3H]5-HT radioligand binding against 5-hydroxytryptamine 1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50001874(1-{5-[4-(2-Ethyl-phenyl)-piperazin-1-ylmethyl]-1-m...)
Affinity DataKi:  27nMAssay Description:The compound was tested for its binding affinity towards 5-hydroxytryptamine 1 receptor by displacing [3H]5-HT radioligand in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50001862((N-(o-methoxyphenyl)piperazine)1-(2-Methoxy-phenyl...)
Affinity DataKi:  28nMAssay Description:The compound was tested for its binding affinity towards 5-hydroxytryptamine 1 receptor by displacing [3H]5-HT radioligand in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50001862((N-(o-methoxyphenyl)piperazine)1-(2-Methoxy-phenyl...)
Affinity DataKi:  29nMAssay Description:Inhibition of [3H]5-HT radioligand binding against 5-hydroxytryptamine 1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50001889(1-{5-[4-(2-sec-Butoxy-phenyl)-piperazin-1-ylmethyl...)
Affinity DataKi:  29nMAssay Description:The compound was tested for its binding affinity towards 5-hydroxytryptamine 1 receptor by displacing [3H]5-HT radioligand in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1D(RAT)
University Of Alberta

Curated by PDSP Ki Database
LigandPNGBDBM35256((S)-mianserin | Lerivon | MIANSERIN | MIANSERIN (+...)
Affinity DataKi:  30.2nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1D(RAT)
University Of Alberta

Curated by PDSP Ki Database
LigandPNGBDBM50013515((+)-yohimbine | (16alpha,17alpha)-17-hydroxyyohimb...)
Affinity DataKi:  30.9nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1D(RAT)
University Of Alberta

Curated by PDSP Ki Database
LigandPNGBDBM50217229(CHEMBL317732)
Affinity DataKi:  32nMAssay Description:Binding affinity to 5-hydroxytryptamine 1D receptor in the rat forebrain by [3H]- SB-204269 displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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