Compile Data Set for Download or QSAR
maximum 50k data
Found 56 of ki data for polymerid = 49000244,49000246
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM25761(Anapriline | Avlocardyl | CHEMBL27 | PROPANOLOL(-)...)
Affinity DataKi:  5.24nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM50019443(1-(1H-Indol-4-yloxy)-3-isopropylamino-propan-2-ol ...)
Affinity DataKi:  7.24nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM82484(TMQ, 3'-Iodo)
Affinity DataKi:  10nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM82487(TMQ, 3',5'-Diiodo)
Affinity DataKi:  10.5nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM82481(CAS_128657 | NSC_128657 | TMQ, 5-Fluoro)
Affinity DataKi:  24.5nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM82491(TMQ, 3'-Nitro)
Affinity DataKi:  31.6nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM82488(TMQ, 5-Iodo)
Affinity DataKi:  33.9nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM82498(TMQ, 5,8-Difluoro)
Affinity DataKi:  34.7nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM82482(TMQ, S-(+)-8-Fluoro)
Affinity DataKi:  75.8nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM82482(TMQ, S-(+)-8-Fluoro)
Affinity DataKi:  76nMAssay Description:Binding affinity against Beta-1 adrenergic receptor in guinea pig left ventricleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM50019355(1-(3,4,5-Trimethoxy-benzyl)-1,2,3,4-tetrahydro-iso...)
Affinity DataKi:  87nMAssay Description:Binding affinity against Beta-1 adrenergic receptor in guinea pig left ventricleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM50019355(1-(3,4,5-Trimethoxy-benzyl)-1,2,3,4-tetrahydro-iso...)
Affinity DataKi:  87.1nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM82493(CAS_128658 | NSC_128658 | TMQ, (+/-)-8-Fluoro)
Affinity DataKi:  97.7nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM82493(CAS_128658 | NSC_128658 | TMQ, (+/-)-8-Fluoro)
Affinity DataKi:  98nMAssay Description:Binding affinity against beta-1 adrenergic receptor in guinea pig left ventricleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM82503(CAS_65772 | NSC_65772 | TMQ, S-(-))
Affinity DataKi:  110nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM50002146(3,6-Dimethyl-8-piperazin-1-yl-imidazo[1,2-a]pyrazi...)
Affinity DataKi:  150nMAssay Description:Binding affinity at Beta-1 adrenergic receptor in guinea pigs by [125I]CYP displacementMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM50002150(5-Bromo-8-piperazin-1-yl-imidazo[1,2-a]pyrazine | ...)
Affinity DataKi:  170nMAssay Description:Binding affinity at Beta-1 adrenergic receptor in guinea pigs by [125I]CYP displacementMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM50002152(6-Methyl-8-piperazin-1-yl-imidazo[1,2-a]pyrazine; ...)
Affinity DataKi:  220nMAssay Description:Binding affinity at Beta-1 adrenergic receptor in guinea pigs by [125I]CYP displacementMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM50002156(2-Methyl-8-piperazin-1-yl-imidazo[1,2-a]pyrazine; ...)
Affinity DataKi:  310nMAssay Description:Binding affinity at Beta-1 adrenergic receptor in guinea pigs by [125I]CYP displacementMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM82486(TMQ, N-methoxybenzyl | TMQ, N-methyl)
Affinity DataKi:  324nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM50019060((+/-)4-(2-Amino-1-hydroxy-ethyl)-3-fluoro-benzene-...)
Affinity DataKi:  350nMAssay Description:Binding affinity against beta-1 adrenergic receptor in guinea pig cerebral cortical membranes by displacement of Dihydro-[3H]-alprenololMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM50002142(5-Methyl-8-piperazin-1-yl-imidazo[1,2-a]pyrazine; ...)
Affinity DataKi:  360nMAssay Description:Binding affinity at Beta-1 adrenergic receptor in guinea pigs by [125I]CYP displacementMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM50002151(8-Piperazin-1-yl-imidazo[1,2-a]pyrazine | CHEMBL33...)
Affinity DataKi:  400nMAssay Description:Binding affinity at Beta-1 adrenergic receptor in guinea pigs by [125I]CYP displacementMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM50002138(3,5-Dimethyl-8-piperazin-1-yl-imidazo[1,2-a]pyrazi...)
Affinity DataKi:  400nMAssay Description:Binding affinity at Beta-1 adrenergic receptor in guinea pigs by [125I]CYP displacementMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM50029051((-)-arterenol | (-)-noradrenaline | (-)-norepineph...)
Affinity DataKi:  400nMAssay Description:Binding affinity against beta-1 adrenergic receptor in guinea pig cerebral cortical membranes by displacement of Dihydro-[3H]-alprenololMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM82500(TMQ, 3'-Amino)
Affinity DataKi:  457nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM25392(4-[1-hydroxy-2-(isopropylamino)ethyl]pyrocatechol;...)
Affinity DataKi:  468nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM50002154(5-Bromo-8-(4-methyl-piperazin-1-yl)-imidazo[1,2-a]...)
Affinity DataKi:  500nMAssay Description:Binding affinity at Beta-1 adrenergic receptor in guinea pigs by [125I]CYP displacementMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM50002157(3,5-Dibromo-8-piperazin-1-yl-imidazo[1,2-a]pyrazin...)
Affinity DataKi:  630nMAssay Description:Binding affinity at Beta-1 adrenergic receptor in guinea pigs by [125I]CYP displacementMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM82502(TMQ, 8-Iodo)
Affinity DataKi:  631nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM82504(TMQ, 5-TrifluoroMe)
Affinity DataKi:  1.10E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM82485(TMQ, N-benzyl)
Affinity DataKi:  1.10E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM82497(TMQ, R-(-)-8-Fluoro)
Affinity DataKi:  1.15E+3nMAssay Description:Binding affinity against Beta-1 adrenergic receptor in guinea pig left ventricleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM82497(TMQ, R-(-)-8-Fluoro)
Affinity DataKi:  1.15E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM50019059((+/-)3-Fluoro-4-(1-hydroxy-2-methylamino-ethyl)-be...)
Affinity DataKi:  1.80E+3nMAssay Description:Binding affinity against beta-1 adrenergic receptor in guinea pig cerebral cortical membranes by displacement of Dihydro-[3H]-alprenololMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM50002139(3-Methyl-8-piperazin-1-yl-imidazo[1,2-a]pyrazine; ...)
Affinity DataKi:  2.40E+3nMAssay Description:Binding affinity at Beta-1 adrenergic receptor in guinea pigs by [125I]CYP displacementMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM50002145(5-Methyl-8-(4-methyl-piperazin-1-yl)-imidazo[1,2-a...)
Affinity DataKi:  2.80E+3nMAssay Description:Binding affinity at Beta-1 adrenergic receptor in guinea pigs by [125I]CYP displacementMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM50002149(3-Isopropyl-8-piperazin-1-yl-imidazo[1,2-a]pyrazin...)
Affinity DataKi:  2.99E+3nMAssay Description:Binding affinity at Beta-1 adrenergic receptor in guinea pigs by [125I]CYP displacementMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM50019061((+/-)4-(2-Amino-1-hydroxy-ethyl)-5-fluoro-benzene-...)
Affinity DataKi: >3.00E+3nMAssay Description:Binding affinity against beta-1 adrenergic receptor in guinea pig cerebral cortical membranes by displacement of Dihydro-[3H]-alprenololMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM50029050((-)-(R)-epinephrine | (-)-3,4-dihydroxy-alpha-((me...)
Affinity DataKi:  3.00E+3nMAssay Description:Binding affinity against beta-1 adrenergic receptor in guinea pig cerebral cortical membranes by displacement of Dihydro-[3H]-alprenololMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM82495(TMQ, N-dichlorobenzyl)
Affinity DataKi:  3.55E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM50131281(5-(1-hydroxy-2-(1-(4-hydroxyphenyl)propan-2-ylamin...)
Affinity DataKi:  4.17E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM50002143(3-Ethyl-8-piperazin-1-yl-imidazo[1,2-a]pyrazine; 2...)
Affinity DataKi:  5.00E+3nMAssay Description:Binding affinity at Beta-1 adrenergic receptor in guinea pigs by [125I]CYP displacementMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM82490(TMQ, N-hydroxyethyl)
Affinity DataKi:  5.37E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM82492(TMQ, N-chloro-benzyl)
Affinity DataKi:  6.17E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM50002140(3-Bromo-8-(4-methyl-piperazin-1-yl)-imidazo[1,2-a]...)
Affinity DataKi:  6.30E+3nMAssay Description:Binding affinity at Beta-1 adrenergic receptor in guinea pigs by [125I]CYP displacementMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM50002147(8-Piperazin-1-yl-3-propyl-imidazo[1,2-a]pyrazine; ...)
Affinity DataKi:  7.79E+3nMAssay Description:Binding affinity at Beta-1 adrenergic receptor in guinea pigs by [125I]CYP displacementMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM82483(TMQ, R-(+) | US11001595, Compound TMQ)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM82472(BW-723C86 | CAS_5311036 | NSC_5311036)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(RABBIT)
Roche Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM85098(N-[5-[5-(2,4-Dioxo-1,3,8-triazaspiro[4.5]decan-8-y...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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