Compile Data Set for Download or QSAR
maximum 50k data
Found 137 of kd data for polymerid = 49000249
TargetBeta-2 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50292219((-)-3-morpholino-4-(3-tert-butylamino-2-hydroxypro...)
Affinity DataKd:  0.240nMAssay Description:In vitro beta-2 adrenergic receptor activity was determined by measuring inhibition of the isoproterenol induced relaxation in isolated guinea pig tr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50365058(CHEMBL1951067)
Affinity DataKd:  0.708nMAssay Description:Competitive antagonist activity at beta2-adrenoreceptor in guinea pig tracheal ring in the presence of N-(5-((1R)-2-(4-(4-(3,4-dimethoxyphenol)-1-oxo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50404804(CHEMBL13365)
Affinity DataKd:  1.26nMAssay Description:Ability to block Beta-2 adrenergic receptor in guinea pig trachea preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM81886(CAS_3506-09-0 | CHEMBL287651 | PROPRANOLOL, dl)
Affinity DataKd:  1.26nMAssay Description:In vitro ability to block beta-2 adrenergic receptor in guinea pig trachea.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50404808(CHEMBL281967)
Affinity DataKd:  1.26nMAssay Description:Ability to block Beta-2 adrenergic receptor in guinea pig trachea preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM25761(Anapriline | Avlocardyl | CHEMBL27 | PROPANOLOL(-)...)
Affinity DataKd:  1.26nMAssay Description:Ability to block Beta-2 adrenergic receptor in guinea pig trachea preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50404805(CHEMBL281294)
Affinity DataKd:  1.60nMAssay Description:Ability to block Beta-2 adrenergic receptor in guinea pig trachea preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50405013(CHEMBL285972)
Affinity DataKd:  2.14nMAssay Description:Beta-2 adrenergic receptor blocking activity in trachea of guinea pig.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM25761(Anapriline | Avlocardyl | CHEMBL27 | PROPANOLOL(-)...)
Affinity DataKd:  3.02nMAssay Description:In vitro beta-2 adrenergic receptor activity was determined by measuring inhibition of the isoproterenol induced relaxation in isolated guinea pig tr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM25761(Anapriline | Avlocardyl | CHEMBL27 | PROPANOLOL(-)...)
Affinity DataKd:  3.39nMAssay Description:Beta-2 adrenergic receptor blocking activity in trachea of guinea pig.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM25761(Anapriline | Avlocardyl | CHEMBL27 | PROPANOLOL(-)...)
Affinity DataKd:  3.39nMAssay Description:The apparent pA2 value was measured for beta-2 adrenergic blocking activity on the trachea of guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50060974(CHEMBL3393402)
Affinity DataKd:  5.10nMAssay Description:Agonist activity at adrenergic beta2 receptor in Hartley guinea pig tracheal ring at basal tone assessed as bronchorelaxation activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50404770(CHEMBL31021)
Affinity DataKd:  6.31nMAssay Description:In vitro ability to block beta-2 adrenergic receptor in guinea pig trachea.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50404785(CHEMBL31529)
Affinity DataKd:  7.94nMAssay Description:In vitro ability to block beta-2 adrenergic receptor in guinea pig trachea.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50405012(CHEMBL24644)
Affinity DataKd:  8.91nMAssay Description:Beta-2 adrenergic receptor blocking activity in trachea of guinea pig.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50404987(CHEMBL3085291)
Affinity DataKd:  8.91nMAssay Description:In vitro beta-2 adrenergic receptor activity was determined by measuring inhibition of the isoproterenol induced relaxation in isolated guinea pig tr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50404488(CHEMBL1161386)
Affinity DataKd:  9.55nMAssay Description:The apparent pA2 value was measured for beta-2 adrenergic blocking activity on the trachea of guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50405017(CHEMBL24045)
Affinity DataKd:  12.6nMAssay Description:Beta-2 adrenergic receptor blocking activity in trachea of guinea pig.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50404790(CHEMBL13284)
Affinity DataKd:  12.6nMAssay Description:Ability to block Beta-2 adrenergic receptor in guinea pig trachea preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50404787(CHEMBL284909)
Affinity DataKd:  12.6nMAssay Description:Ability to block Beta-2 adrenergic receptor in guinea pig trachea preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50404807(CHEMBL31335)
Affinity DataKd:  15.8nMAssay Description:Ability to block Beta-2 adrenergic receptor in guinea pig trachea preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50405018(CHEMBL24500)
Affinity DataKd:  16.6nMAssay Description:Beta-2 adrenergic receptor blocking activity in trachea of guinea pig.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM25392(4-[1-hydroxy-2-(isopropylamino)ethyl]pyrocatechol;...)
Affinity DataKd:  18nMAssay Description:Agonist activity at adrenergic beta2 receptor in Hartley guinea pig tracheal ring assessed as bronchorelaxation activity against histamine-induced co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50404492(CHEMBL155714)
Affinity DataKd:  20.9nMAssay Description:The apparent pA2 value was measured for beta-2 adrenergic blocking activity on the trachea of guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50405014(CHEMBL24480)
Affinity DataKd:  22.4nMAssay Description:Beta-2 adrenergic receptor blocking activity in trachea of guinea pig.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50404502(CHEMBL555848)
Affinity DataKd:  22.4nMAssay Description:The apparent pA2 value was measured for beta-2 adrenergic blocking activity on the trachea of guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50405011(CHEMBL26059)
Affinity DataKd:  22.9nMAssay Description:Beta-2 adrenergic receptor blocking activity in trachea of guinea pig.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM25392(4-[1-hydroxy-2-(isopropylamino)ethyl]pyrocatechol;...)
Affinity DataKd:  25nMAssay Description:Agonist activity at adrenergic beta2 receptor in Hartley guinea pig tracheal ring at basal tone assessed as bronchorelaxation activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50060974(CHEMBL3393402)
Affinity DataKd:  28nMAssay Description:Agonist activity at adrenergic beta2 receptor in Hartley guinea pig tracheal ring assessed as bronchorelaxation activity against histamine-induced co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50404487(CHEMBL156871)
Affinity DataKd:  30.2nMAssay Description:The apparent pA2 value was measured for beta-2 adrenergic blocking activity on the trachea of guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50404484(CHEMBL1161388 | CHEMBL26003)
Affinity DataKd:  32.4nMAssay Description:Beta-2 adrenergic receptor blocking activity in trachea of guinea pig.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50404484(CHEMBL1161388 | CHEMBL26003)
Affinity DataKd:  32.4nMAssay Description:The apparent pA2 value was measured for beta-2 adrenergic blocking activity on the trachea of guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50404982(CHEMBL366769)
Affinity DataKd:  33.1nMAssay Description:In vitro beta-2 adrenergic receptor activity was determined by measuring inhibition of the isoproterenol induced relaxation in isolated guinea pig tr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50404784(CHEMBL31811)
Affinity DataKd:  39.8nMAssay Description:In vitro ability to block beta-2 adrenergic receptor in guinea pig trachea.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50404783(CHEMBL32902)
Affinity DataKd:  39.8nMAssay Description:In vitro ability to block beta-2 adrenergic receptor in guinea pig trachea.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50404810(CHEMBL281298)
Affinity DataKd:  39.8nMAssay Description:Ability to block Beta-2 adrenergic receptor in guinea pig trachea preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50404763(CHEMBL283289)
Affinity DataKd:  39.8nMAssay Description:In vitro ability to block beta-2 adrenergic receptor in guinea pig trachea.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM25761(Anapriline | Avlocardyl | CHEMBL27 | PROPANOLOL(-)...)
Affinity DataKd:  43.6nMAssay Description:Antagonist activity of compound against Beta-2 adrenergic receptor in isolated guinea pig tracheaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50405015(CHEMBL26049)
Affinity DataKd:  47.9nMAssay Description:Beta-2 adrenergic receptor blocking activity in trachea of guinea pig.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50404776(CHEMBL287242)
Affinity DataKd:  50.1nMAssay Description:In vitro ability to block beta-2 adrenergic receptor in guinea pig trachea.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50404994(CHEMBL2096752)
Affinity DataKd:  57.5nMAssay Description:In vitro beta-2 adrenergic receptor activity was determined by measuring inhibition of the isoproterenol induced relaxation in isolated guinea pig tr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50404809(CHEMBL31450)
Affinity DataKd:  63.1nMAssay Description:Ability to block Beta-2 adrenergic receptor in guinea pig trachea preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50404813(CHEMBL13358)
Affinity DataKd:  79.4nMAssay Description:Ability to block Beta-2 adrenergic receptor in guinea pig trachea preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50405024(CHEMBL286783)
Affinity DataKd:  81.3nMAssay Description:Beta-2 adrenergic receptor blocking activity in trachea of guinea pig.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50404498(CHEMBL1161383)
Affinity DataKd:  81.3nMAssay Description:The apparent pA2 value was measured for beta-2 adrenergic blocking activity on the trachea of guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50404696(CHEMBL427310)
Affinity DataKd:  81.3nMAssay Description:Antagonist activity of compound against Beta-2 adrenergic receptor in isolated guinea pig tracheaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50405027(CHEMBL25929)
Affinity DataKd:  97.7nMAssay Description:Beta-2 adrenergic receptor blocking activity in trachea of guinea pig.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50404767(CHEMBL448775)
Affinity DataKd:  100nMAssay Description:In vitro ability to block beta-2 adrenergic receptor in guinea pig trachea.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50404771(CHEMBL31938)
Affinity DataKd:  100nMAssay Description:In vitro ability to block beta-2 adrenergic receptor in guinea pig trachea.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50405521(ALO 1401-02 | ALO-1401-02 | BETAXOLOL HYDROCHLORID...)
Affinity DataKd:  105nMAssay Description:In vitro beta-2 adrenergic receptor activity was determined by measuring inhibition of the isoproterenol induced relaxation in isolated guinea pig tr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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