Compile Data Set for Download or QSAR
maximum 50k data
Found 710 of ic50 data for polymerid = 49000277
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50236697(5-L-isoleucineangiotensin II | 5-isoleucine-angiot...)
Affinity DataIC50:  0.0800nMAssay Description:Displacement of [125I]CGP 42112A from human recombinant AT2 receptor expressed in HEK293 cells measured after 4 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50155247(CHEMBL385433)
Affinity DataIC50:  0.0800nMAssay Description:Displacement of [125I]CGP42112A from human recombinant AT2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50030711(CHEMBL338027 | L-163958 | Pentanoic acid {4-bromo-...)
Affinity DataIC50:  0.120nMAssay Description:Inhibition of Angiotensin II receptor, type 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50009718(2-Ethyl-5,7-dimethyl-3-[2'-(1H-tetrazol-5-yl)-biph...)
Affinity DataIC50:  0.200nMAssay Description:Binding affinity to angiotensin AT2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50043280(4'-((1,4'-dimethyl-2'-propyl(2,6'-bi-1H-benzimidaz...)
Affinity DataIC50:  0.330nMAssay Description:Displacement of [125I]Sar1 Ile8-Ang 2 from angiotensin 2 AT2 receptor after 180 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50048114(CHEMBL384352 | c[Sar1-Arg2-Mpt3-Tyr4-Hcy5-His6-Pro...)
Affinity DataIC50:  0.470nMAssay Description:In vitro binding affinity at angiotensin II (type 2) receptor in rabbit uterus.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50283763(CHEMBL321531 | N-(3-{3-Butyl-4-[2'-(2-chloro-benzo...)
Affinity DataIC50:  0.480nMAssay Description:Inhibitory concentration of the compound against cloned human AT1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50009338((S)-2-((S)-1-((S)-2-((S)-2-((S)-2-((S)-2-((S)-5-(d...)
Affinity DataIC50:  0.530nMAssay Description:Inhibition of human angiotensin II AT2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50282401(CHEMBL157510 | PD-126055 | Potassium; (S)-5-benzyl...)
Affinity DataIC50:  0.580nMAssay Description:Inhibitory activity against angiotensin II type 2 (AT2) receptor in rabbit uterine membranes.More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50049182((S)-5-Benzyloxy-2-diphenylacetyl-6-methoxy-1,2,3,4...)
Affinity DataIC50:  0.580nMAssay Description:In vitro binding affinity of compound was measured against angiotensin II (AT2) receptorMore data for this Ligand-Target Pair
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50049182((S)-5-Benzyloxy-2-diphenylacetyl-6-methoxy-1,2,3,4...)
Affinity DataIC50:  0.600nMAssay Description:Inhibitory activity was evaluated against Angiotensin II receptor, type 2More data for this Ligand-Target Pair
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50228195(Angiotensin Ii | CHEBI:2719)
Affinity DataIC50:  0.617nMAssay Description:Displacement of [125-I]-[Sar1, Ile8] from recombinant human AT2R transfected in human HEK293 cells incubated for 2 hrs by liquid scintillation counte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50030707(CHEMBL122273 | Pentanoic acid (4-bromo-3-{3-ethyl-...)
Affinity DataIC50:  0.640nMAssay Description:In vitro inhibitory activity against Angiotensin II receptor type 2 in human adrenal membrane preparations.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50048119(CHEMBL385283 | c[Sar1-Arg2-Hcy3-Tyr4-MPt5-His6-Pro...)
Affinity DataIC50:  0.650nMAssay Description:In vitro binding affinity at angiotensin II (type 2) receptor in rabbit uterus.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50283244(Biphenylsulfonylcarbamate compound | CHEMBL71125)
Affinity DataIC50:  0.690nMAssay Description:Binding affinity for angiotensin II AT-2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50049206(5-Ethyl-3-(3-fluoro-2'-isopentyloxycarbaronylsulfa...)
Affinity DataIC50:  0.690nMAssay Description:Inhibition of Angiotensin II receptor, type 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50049206(5-Ethyl-3-(3-fluoro-2'-isopentyloxycarbaronylsulfa...)
Affinity DataIC50:  0.700nMAssay Description:Binding affinity for angiotensin II AT-2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50141059(CHEMBL289614 | L-162782 | N-Butyloxycarbonyl-4'-(2...)
Affinity DataIC50:  0.700nMAssay Description:Binding affinity to type-2 angiotensin-2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50141059(CHEMBL289614 | L-162782 | N-Butyloxycarbonyl-4'-(2...)
Affinity DataIC50:  0.700nMAssay Description:Binding affinity to AT2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50141059(CHEMBL289614 | L-162782 | N-Butyloxycarbonyl-4'-(2...)
Affinity DataIC50:  0.700nMAssay Description:Binding affinity of the compound towards Angiotensin II receptor, type 2 was measured through displacement of [125I]-Ang II in pig uterus myometrial ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM82433(CHEMBL302102 | L-159,689 | L-159689 | N-Pentyl-N-[...)
Affinity DataIC50:  0.700nMAssay Description:Inhibitory concentration against angiotensin II receptor, type 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50048113(CHEMBL414533 | c[Sar1-Arg2-Cys3-Tyr4-MPt5-His6-Pro...)
Affinity DataIC50:  0.820nMAssay Description:In vitro binding affinity at angiotensin II (type 2) receptor in rabbit uterus.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50030732(CHEMBL323506 | N-{3-[3-Butyl-4-(3-fluoro-2'(tert-b...)
Affinity DataIC50:  0.820nMAssay Description:Inhibitory concentration of the compound against cloned human AT1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50049182((S)-5-Benzyloxy-2-diphenylacetyl-6-methoxy-1,2,3,4...)
Affinity DataIC50:  0.840nMAssay Description:Inhibitory activity against angiotensin II type 2 (AT2) receptor in rabbit uterine membranes.More data for this Ligand-Target Pair
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50049182((S)-5-Benzyloxy-2-diphenylacetyl-6-methoxy-1,2,3,4...)
Affinity DataIC50:  0.840nMAssay Description:Inhibitory activity against angiotensin II type 2 (AT2) receptor in rabbit uterine membranes.More data for this Ligand-Target Pair
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50030709(CHEMBL338434 | Pentanoic acid {3-[3-butyl-4-(3-flu...)
Affinity DataIC50:  0.880nMAssay Description:In vitro inhibitory activity against Angiotensin II receptor, type 2 in human adrenal membrane preparations. For this assay, only 0.02%BSA was presen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50280907((S)-1,4-Bis-diphenylcarbamoyl-piperazine-2-carboxy...)
Affinity DataIC50:  0.890nMAssay Description:Inhibitory activity against angiotensin II type 2 (AT2) receptor in rabbit uterine membranes.More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50283200(Biphenylsulfonylcarbamate compound | CHEMBL71172)
Affinity DataIC50:  0.900nMAssay Description:Binding affinity for angiotensin II AT-2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50283199(Biphenylsulfonylcarbamate compound | CHEMBL71220)
Affinity DataIC50:  0.900nMAssay Description:Binding affinity for angiotensin II AT-2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50285762(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  0.900nMAssay Description:In vitro binding affinity at Angiotensin II Type 2 receptor in rabbit uterus membrane by [125I]-AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50032362(3-(2'-Isopentyloxycarbonylsulfamoyl-3-fluoro-biphe...)
Affinity DataIC50:  1nMAssay Description:Inhibition of Angiotensin II receptor, type 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50283213(Biphenylsulfonylcarbamate compound | CHEMBL307318)
Affinity DataIC50:  1nMAssay Description:Binding affinity for angiotensin II AT-2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50283245(Biphenylsulfonylcarbamate compound | CHEMBL70789)
Affinity DataIC50:  1nMAssay Description:Binding affinity for angiotensin II AT-2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50283238(Biphenylsulfonylcarbamate compound | CHEMBL70867)
Affinity DataIC50:  1nMAssay Description:Binding affinity for angiotensin II AT-2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50283204(Biphenylsulfonylcarbamate compound | CHEMBL311625)
Affinity DataIC50:  1nMAssay Description:Binding affinity for angiotensin II AT-2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50283234(Biphenylsulfonylcarbamate compound | CHEMBL72595)
Affinity DataIC50:  1nMAssay Description:Binding affinity for angiotensin II AT-2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50283220(Biphenylsulfonylcarbamate compound | CHEMBL302579)
Affinity DataIC50:  1nMAssay Description:Binding affinity for angiotensin II AT-2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50285763(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  1.10nMAssay Description:In vitro binding affinity at Angiotensin II Type 2 receptor in rabbit uterus membrane by [125I]-AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50285752(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  1.10nMAssay Description:In vitro binding affinity at Angiotensin II Type 2 receptor in rabbit uterus membrane by [125I]-AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50285757(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  1.10nMAssay Description:In vitro binding affinity at Angiotensin II Type 2 receptor in rabbit uterus membrane by [125I]-AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50030693(CHEMBL338687 | Pentanoic acid {4-bromo-3-[3-ethyl-...)
Affinity DataIC50:  1.10nMAssay Description:In vitro inhibitory activity against Angiotensin II receptor type 2 in human adrenal membrane preparations.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50282404(5-Benzyloxy-2-(2-cyclopentyl-2-phenyl-acetyl)-6-me...)
Affinity DataIC50:  1.10nMAssay Description:Inhibitory activity against angiotensin II type 2 (AT2) receptor in rabbit uterine membranes.More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50030684(CHEMBL339722 | N-{3-[3-Butyl-4-(3-fluoro-2-(N-t-bu...)
Affinity DataIC50:  1.20nMAssay Description:In vitro inhibitory activity against Angiotensin II receptor, type 2 in human adrenal membrane preparations. For this assay, only 0.02%BSA was presen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50030687(CHEMBL339256 | N-(3-{3-Butyl-4-[2'-(2-chloro-benzo...)
Affinity DataIC50:  1.30nMAssay Description:In vitro inhibitory activity against Angiotensin II receptor, type 2 in human adrenal membrane preparations. For this assay, only 0.02%BSA was presen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50009338((S)-2-((S)-1-((S)-2-((S)-2-((S)-2-((S)-2-((S)-5-(d...)
Affinity DataIC50:  1.30nMAssay Description:In vitro binding affinity at angiotensin II (type 2) receptor in rabbit uterus.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50030700(CHEMBL436396 | N-{4-Bromo-3-[4-(3-fluoro-2'-(N-t-b...)
Affinity DataIC50:  1.40nMAssay Description:In vitro inhibitory activity against Angiotensin II receptor type 2 in human adrenal membrane preparations.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50030691(CHEMBL122380 | Pentanoic acid (4-bromo-3-{4-[2'-(2...)
Affinity DataIC50:  1.5nMAssay Description:In vitro inhibitory activity against Angiotensin II receptor type 2 in human adrenal membrane preparations.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50030708(CHEMBL125760 | N-{4-Chloro-3-[3-ethyl-4-(3-fluoro-...)
Affinity DataIC50:  1.5nMAssay Description:In vitro inhibitory activity against Angiotensin II receptor type 2 in human adrenal membrane preparations.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50280907((S)-1,4-Bis-diphenylcarbamoyl-piperazine-2-carboxy...)
Affinity DataIC50:  1.5nMAssay Description:In vitro binding affinity of compound was measured against Angiotensin II receptor, type 2More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50283248(Biphenylsulfonylcarbamate compound | CHEMBL70726)
Affinity DataIC50:  1.60nMAssay Description:Binding affinity for angiotensin II AT-2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
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