Compile Data Set for Download or QSAR
maximum 50k data
Found 200 of ki for UniProtKB: P30551
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50089269(CHEMBL276192 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2...)
Affinity DataKi:  0.0200nMAssay Description:Inhibition of [125I]BH-CCK-8 binding to Cholecystokinin type A receptor of rat pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50061828(CHEMBL76248 | CID44356929 | N-(1-Carbamoyl-2-pheny...)
Affinity DataKi:  0.0300nMAssay Description:Binding affinity for Cholecystokinin type A receptor using [125I]BH-CCK-8 in rat pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50061829((R)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-({(S)-2-[...)
Affinity DataKi:  0.0300nMAssay Description:Binding affinity for Cholecystokinin type A receptor using [125I]BH-CCK-8 in rat pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50061828(CHEMBL76248 | CID44356929 | N-(1-Carbamoyl-2-pheny...)
Affinity DataKi:  0.0300nMAssay Description:Inhibition of [125I]BH-CCK-8 binding to Cholecystokinin type A receptor of rat pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50089268(CHEMBL267861 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2...)
Affinity DataKi:  0.0500nMAssay Description:Inhibition of [125I]BH-CCK-8 binding to Cholecystokinin type A receptor of rat pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50061832((S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-{(S)-2-[(...)
Affinity DataKi:  0.0700nMAssay Description:Binding affinity for Cholecystokinin type A receptor using [125I]BH-CCK-8 in rat pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataKi:  0.0900nMAssay Description:Binding affinity for Cholecystokinin type A receptor using [125I]BH-CCK-8 in rat pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataKi:  0.0900nMAssay Description:Inhibition of [125I]BH-CCK-8 binding to Cholecystokinin type A receptor of rat pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM81962(S-L-365,260)
Affinity DataKi:  0.148nMAssay Description:Inhibition by displacing [3H]CCK-8S against Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50449787(CHEMBL2062154 | PD-134308)
Affinity DataKi:  0.148nMAssay Description:Inhibition by displacing [3H]CCK-8S against Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50005463((R)-1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-...)
Affinity DataKi:  0.148nMAssay Description:Inhibition by displacing [3H]CCK-8S against Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50061833((R)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-{(S)-2-[(...)
Affinity DataKi:  0.200nMAssay Description:Binding affinity for Cholecystokinin type A receptor using [125I]BH-CCK-8 in rat pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50369326(CHEMBL1791002)
Affinity DataKi:  0.240nMAssay Description:Binding affinity for Cholecystokinin type A receptor using [125I]BH-CCK-8 in rat pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50060321(1H-Indole-2-carboxylic acid ((R)-1-methyl-2-oxo-5-...)
Affinity DataKi:  0.300nMAssay Description:Inhibition of [3H]-pCCK-8 specific binding to Cholecystokinin type A receptor of rat pancreasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataKi:  0.520nMAssay Description:Inhibition of [3H]-pCCK-8 specific binding to Cholecystokinin type A receptor of rat pancreasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50369325(CHEMBL1791005)
Affinity DataKi:  0.530nMAssay Description:Binding affinity for Cholecystokinin type A receptor using [125I]BH-CCK-8 in rat pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50060322(CHEMBL332261 | [(S)-1-((4aS,5S)-2-Benzyl-1,3-dioxo...)
Affinity DataKi:  0.620nMAssay Description:Inhibition of [3H]-pCCK-8 specific binding to Cholecystokinin type A receptor of rat pancreasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50005463((R)-1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-...)
Affinity DataKi:  0.700nMAssay Description:Inhibition of [3H]-L-364,718 binding to cholecystokinin type A receptor in rat pancreas membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50089276(CHEMBL430608 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2...)
Affinity DataKi:  0.980nMAssay Description:Inhibition of [125I]BH-CCK-8 binding to Cholecystokinin type A receptor of rat pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50061834((R)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-{(S)-2-[(...)
Affinity DataKi:  0.980nMAssay Description:Binding affinity for Cholecystokinin type A receptor using [125I]BH-CCK-8 in rat pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50211670(CHEMBL103750)
Affinity DataKi:  1.5nMAssay Description:Binding affinity was measured by its ability to displace [3H]CCK-8S from CCK-A receptor in rat pancreasMore data for this Ligand-Target Pair
In DepthDetails
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50089275(CHEMBL384303 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2...)
Affinity DataKi:  3.40nMAssay Description:Inhibition of [125I]BH-CCK-8 binding to Cholecystokinin type A receptor of rat pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50089277(CHEMBL311187 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-({...)
Affinity DataKi:  4.20nMAssay Description:Inhibition of [125I]BH-CCK-8 binding to Cholecystokinin type A receptor of rat pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50016425((S)-3-{(S)-2-[(S)-2-(2-{(S)-2-[(S)-2-tert-Butoxyca...)
Affinity DataKi:  4.30nMAssay Description:Evaluated for binding affinity measured by inhibiting [3H]Boc[Nle28,31]CCK27-33 specific binding to Cholecystokinin receptor in rat pancreas membrane...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50060156(CHEMBL319795)
Affinity DataKi:  4.60nMAssay Description:Binding affinity was measured by its ability to displace [3H]CCK-8S from CCK-A receptor in rat pancreasMore data for this Ligand-Target Pair
In DepthDetails
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50211668(CHEMBL103968)
Affinity DataKi:  4.90nMAssay Description:Binding affinity was measured by its ability to displace [3H]CCK-8S from CCK-A receptor in rat pancreasMore data for this Ligand-Target Pair
In DepthDetails
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50472887(CHEMBL330773)
Affinity DataKi:  7.40nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataKi:  8.70nMAssay Description:Evaluated for binding affinity measured by inhibiting [3H]Boc[Nle28,31]CCK27-33 specific binding to Cholecystokinin receptor in rat pancreas membrane...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50212321(CHEMBL317081)
Affinity DataKi:  8.90nMAssay Description:Binding affinity was measured by its ability to displace [3H]CCK-8S from CCK-A receptor in rat pancreasMore data for this Ligand-Target Pair
In DepthDetails
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50212326(CHEMBL102867)
Affinity DataKi:  9.80nMAssay Description:Binding affinity was measured by its ability to displace [3H]CCK-8S from CCK-A receptor in rat pancreasMore data for this Ligand-Target Pair
In DepthDetails
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50060323(CHEMBL431858 | [(S)-1-((4aR,5R)-2-Benzyl-1,3-dioxo...)
Affinity DataKi:  10.6nMAssay Description:Inhibition of [3H]-pCCK-8 specific binding to Cholecystokinin type A receptor of rat pancreasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50472882(CHEMBL332403)
Affinity DataKi:  12nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50472876(CHEMBL332568)
Affinity DataKi:  19nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50061830((R)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-{(S)-2-[(...)
Affinity DataKi:  19nMAssay Description:Binding affinity for Cholecystokinin type A receptor using [125I]BH-CCK-8 in rat pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50089272(CHEMBL312359 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2...)
Affinity DataKi:  19nMAssay Description:Inhibition of [125I]BH-CCK-8 binding to Cholecystokinin type A receptor of rat pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50472870(CHEMBL331975)
Affinity DataKi:  22nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50472847(CHEMBL121331)
Affinity DataKi:  22nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50472898(CHEMBL332902)
Affinity DataKi:  23nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50472884(CHEMBL121021)
Affinity DataKi:  36nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50212329(CHEMBL101125)
Affinity DataKi:  42nMAssay Description:Binding affinity was measured by its ability to displace [3H]CCK-8S from CCK-A receptor in rat pancreasMore data for this Ligand-Target Pair
In DepthDetails
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50472892(CHEMBL331262)
Affinity DataKi:  45nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50049805(CHEMBL169703 | Thiophene-3-carboxylic acid [5-(2-f...)
Affinity DataKi:  47nMAssay Description:Binding affinity against Cholecystokinin type A receptor using [125I]-(BH)-CCK-8 as radioligand in rat pancreas.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50472880(CHEMBL338278)
Affinity DataKi:  47nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50472886(CHEMBL421271)
Affinity DataKi:  48nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50472861(CHEMBL121267)
Affinity DataKi:  48nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50005459(4-(3,4-Dichloro-benzoylamino)-4-dipentylcarbamoyl-...)
Affinity DataKi:  49nMAssay Description:Inhibition of [3H]-L-364,718 binding to cholecystokinin type A receptor in rat pancreas membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50472868(CHEMBL120168)
Affinity DataKi:  49nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50089270(CHEMBL308622 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2...)
Affinity DataKi:  51nMAssay Description:Inhibition of [125I]BH-CCK-8 binding to Cholecystokinin type A receptor of rat pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50214389(CHEMBL101063)
Affinity DataKi:  62nMAssay Description:Evaluated in vitro for Cholecystokinin type A receptor affinity by measuring its ability to displace tritiated CCK-8S bound on rat pancreas Cholecyst...More data for this Ligand-Target Pair
In DepthDetails
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50472875(CHEMBL333930)
Affinity DataKi:  63nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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