Affinity DataEC50: 1.60nMAssay Description:Negative logarithm of the molar concentration for agonist activity at mu receptor was determined in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataEC50: 2nMAssay Description:Activity against mu opioid receptor by stimulation of [35S]GTPgammaS binding in CHO-hgamma cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 9nMAssay Description:Activity against mu opioid receptor by stimulation of [35S]GTPgammaS binding in CHO-hgamma cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 21nMAssay Description:Agonist activity at MOR in guinea pig vas deferensMore data for this Ligand-Target Pair
Affinity DataEC50: 27nMAssay Description:Activity against mu opioid receptor by stimulation of [35S]GTPgammaS binding in CHO-hgamma cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 32nMAssay Description:Agonist activity at mu-opioid receptor in guinea pig ileum assessed as inhibition of electrically induced twitchesMore data for this Ligand-Target Pair
Affinity DataEC50: 53nMAssay Description:Agonist activity at mu opioid receptor in guinea pig brain membranes by [35S]-GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 58nMAssay Description:Inhibition of mu opioid receptor mediated GTPgammaS binding to CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataEC50: 100nMAssay Description:Activity against mu opioid receptor by stimulation of [35S]GTPgammaS binding in CHO-hgamma cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 142nMAssay Description:Activity against mu opioid receptor by stimulation of [35S]GTPgammaS binding in CHO-hgamma cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 153nMAssay Description:Inhibition of mu opioid receptor mediated GTPgammaS binding to CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataEC50: 155nMAssay Description:Activity against mu opioid receptor by stimulation of [35S]GTPgammaS binding in CHO-hgamma cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 158nMAssay Description:Agonist activity at MOR in Dunkin-Hartley guinea pig ileum assessed as inhibition of EFS-induced contractions incubated for 60 minsMore data for this Ligand-Target Pair
Affinity DataEC50: 161nMAssay Description:Activity against mu opioid receptor by stimulation of [35S]GTPgammaS binding in CHO-hgamma cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 225nMAssay Description:Agonistic activity towards Opioid receptor mu 1 was determined in [35S]GTP-gamma-S, binding assay in guinea pig caudate; g = not active as an agonistMore data for this Ligand-Target Pair
Affinity DataEC50: 230nMAssay Description:Agonist activity at mu opioid receptor in guinea pig brain membranes by [35S]-GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 290nMAssay Description:In vitro bioassay data to determine the effective concentration required for antagonistic activity against Opioid receptor mu 1 in functional assay,G...More data for this Ligand-Target Pair
Affinity DataEC50: 293nMAssay Description:Effective concentration was measured towards mu opioid receptor using guinea pig ileum (GPI,mu) bioassay in vitroMore data for this Ligand-Target Pair
Affinity DataEC50: 414nMAssay Description:Agonistic activity towards Opioid receptor mu 1 was determined in [35S]GTP-gamma-S, binding assay in guinea pig caudateMore data for this Ligand-Target Pair
Affinity DataEC50: 490nMAssay Description:Negative logarithm of the molar concentration for agonist activity at mu receptor was determined in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataEC50: 525nMAssay Description:Negative logarithm of the molar concentration for agonist activity at mu receptor was determined in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataEC50: 631nMAssay Description:Negative logarithm of the molar concentration for agonist activity at mu receptor was determined in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataEC50: 660nMAssay Description:Agonistic activity towards Opioid receptor mu 1 was determined in [35S]GTP-gamma-S, binding assay in guinea pig caudateMore data for this Ligand-Target Pair
Affinity DataEC50: 794nMAssay Description:Agonist activity at MOR in Dunkin-Hartley guinea pig ileum assessed as inhibition of EFS-induced contractions incubated for 60 minsMore data for this Ligand-Target Pair
Affinity DataEC50: 813nMAssay Description:Negative logarithm of the molar concentration for agonist activity at mu receptor was determined in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataEC50: 900nMAssay Description:Agonistic activity towards Opioid receptor mu 1 was determined in [35S]GTP-gamma-S, binding assay in guinea pig caudate; g = not active as an agonistMore data for this Ligand-Target Pair
Affinity DataEC50: 1.03E+3nMAssay Description:Antagonism of compound towards Opioid receptor mu 1 was determined using PL-017 in guinea pig ileum (GPI) smooth muscle contraction assays; d = agoni...More data for this Ligand-Target Pair
Affinity DataEC50: 1.25E+3nMAssay Description:Tested for electrically induced smooth muscle contractions from guinea pig ileum expressed in mu opioid receptorsMore data for this Ligand-Target Pair
Affinity DataEC50: 1.30E+3nMAssay Description:Inhibition of mu opioid receptor mediated GTPgammaS binding to CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataEC50: 1.31E+3nMAssay Description:Agonistic activity towards Opioid receptor mu 1 was determined in [35S]GTP-gamma-S, binding assay in guinea pig caudate; g = not active as an agonistMore data for this Ligand-Target Pair
Affinity DataEC50: 2.12E+3nMAssay Description:Inhibition of mu opioid receptor mediated GTPgammaS binding to CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataEC50: 2.40E+3nMAssay Description:Inhibition of mu opioid receptor mediated GTPgammaS binding to CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataEC50: 2.45E+3nMAssay Description:Activity against mu opioid receptor by stimulation of [35S]GTPgammaS binding in CHO-hgamma cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 2.90E+3nMAssay Description:Effective concentration was measured towards mu opioid receptor using guinea pig ileum (GPI,mu) bioassay in vitroMore data for this Ligand-Target Pair
Affinity DataEC50: 3.00E+3nMAssay Description:Agonistic activity towards Opioid receptor mu 1 was determined in [35S]GTP-gamma-S, binding assay in guinea pig caudateMore data for this Ligand-Target Pair
Affinity DataEC50: 3.00E+3nMAssay Description:Agonistic activity towards Opioid receptor mu 1 was determined in [35S]GTP-gamma-S, binding assay in guinea pig caudateMore data for this Ligand-Target Pair
Affinity DataEC50: 3.22E+3nMAssay Description:Agonistic activity towards Opioid receptor mu 1 was determined in [35S]GTP-gamma-S, binding assay in guinea pig caudate; g = not active as an agonistMore data for this Ligand-Target Pair
Affinity DataEC50: 3.84E+3nMAssay Description:Effective concentration was measured towards mu opioid receptor using guinea pig ileum (GPI,mu) bioassay in vitroMore data for this Ligand-Target Pair
Affinity DataEC50: 7.30E+3nMAssay Description:In vitro bioassay data to determine the effective concentration required for antagonistic activity against Opioid receptor mu 1 in functional assay,G...More data for this Ligand-Target Pair
Affinity DataEC50: 7.30E+3nMAssay Description:Effective concentration was measured towards mu opioid receptor using guinea pig ileum (GPI,mu) bioassay in vitroMore data for this Ligand-Target Pair
Affinity DataEC50: 7.60E+3nMAssay Description:Tested for electrically induced smooth muscle contractions from guinea pig ileum expressed in mu opioid receptorsMore data for this Ligand-Target Pair
Affinity DataEC50: <1.00E+4nMAssay Description:Negative logarithm of the molar concentration for agonist activity at Opioid receptor mu 1 was determined in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Inhibition of mu opioid receptor mediated GTPgammaS binding to CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Inhibition of mu opioid receptor mediated GTPgammaS binding to CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Inhibition of mu opioid receptor mediated GTPgammaS binding to CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataEC50: <1.00E+4nMAssay Description:Negative logarithm of the molar concentration for agonist activity at Opioid receptor mu 1 was determined in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataEC50: 2.00E+4nMAssay Description:Agonist activity at MOR in Dunkin-Hartley guinea pig ileum assessed as inhibition of EFS-induced contractions incubated for 60 minsMore data for this Ligand-Target Pair
Affinity DataEC50: 3.90E+4nMAssay Description:Tested for electrically induced smooth muscle contractions from guinea pig ileum expressed in mu opioid receptorsMore data for this Ligand-Target Pair
Affinity DataEC50: 5.00E+4nMAssay Description:In vitro bioassay data to determine the effective concentration required for antagonistic activity against Opioid receptor mu 1 in functional assay,G...More data for this Ligand-Target Pair
Affinity DataEC50: 5.01E+7nMAssay Description:Agonist activity at MOR in Dunkin-Hartley guinea pig ileum assessed as inhibition of EFS-induced contractions incubated for 60 minsMore data for this Ligand-Target Pair
