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Found 37 of ic50 for UniProtKB: P28646
TargetSomatostatin receptor type 1/2/3/4/5(RAT)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50476140(CHEMBL373632)
Affinity DataIC50:  0.100nMAssay Description:Displacement of [125I]SRIF-14 from SSTR of rat AR42J cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1/2/3/4/5(RAT)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM81767(15-28-Somatostatin-28 | CAS_38916-34-6 | CB6417646...)
Affinity DataIC50:  0.200nMAssay Description:Compound was tested for its potency to displace 3-[125I]- - Tyr11-SRIF-14 from somatostatin receptor on membranes of rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails
TargetSomatostatin receptor type 1/2/3/4/5(RAT)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50476137(CHEMBL222751)
Affinity DataIC50:  0.400nMAssay Description:Displacement of [125I]SRIF-14 from SSTR of rat AR42J cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1/2/3/4/5(RAT)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM81767(15-28-Somatostatin-28 | CAS_38916-34-6 | CB6417646...)
Affinity DataIC50:  0.430nMAssay Description:Compound was tested for its inhibitory effect against somatostatin receptor in rat cortex membrane using [125I]Tyr3-octreotide as the radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetSomatostatin receptor type 1/2/3/4/5(RAT)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50214421(SOMATOSTATIN RECEPTOR LIGAND)
Affinity DataIC50:  0.430nMAssay Description:Compound was tested for its inhibitory effect against somatostatin receptor in rat cortex membrane using [125I]Tyr3-octreotide as the radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetSomatostatin receptor type 1/2/3/4/5(RAT)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50476135(CHEMBL374316)
Affinity DataIC50:  0.700nMAssay Description:Displacement of [125I]SRIF-14 from SSTR of rat AR42J cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1/2/3/4/5(RAT)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50476143(CHEMBL376001)
Affinity DataIC50:  1.5nMAssay Description:Displacement of [125I]SRIF-14 from SSTR of rat AR42J cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1/2/3/4/5(RAT)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50476144(CHEMBL434761)
Affinity DataIC50:  24nMAssay Description:Displacement of [125I]SRIF-14 from SSTR of rat AR42J cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1/2/3/4/5(RAT)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50020202(CHEMBL2369466 | D-Tic-c(Cys-Tyr-D-Trp-Lys-Thr-Pen-...)
Affinity DataIC50:  949nMAssay Description:Binding affinity in competition with [125I]- CGP-23996 in somatostatin receptor binding to rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1/2/3/4/5(RAT)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50020209(CHEMBL410090 | CTP)
Affinity DataIC50:  1.46E+3nMAssay Description:Binding affinity in competition with [125I]- CGP-23996 in somatostatin receptor binding to rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1/2/3/4/5(RAT)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50020205(CHEMBL216354 | D-Tic-c(Cys-Tyr-D-Trp-Lys-Thr-Pen-)...)
Affinity DataIC50:  1.50E+3nMAssay Description:Binding affinity in competition with [125I]- CGP-23996 in somatostatin receptor binding to rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1/2/3/4/5(RAT)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50020213(CHEMBL264082 | D-Trpc(-Cys-Tyr-D-Trp-Lys-Thr-Pen-)...)
Affinity DataIC50:  1.60E+3nMAssay Description:Binding affinity in competition with [125I]- CGP-23996 in somatostatin receptor binding to rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1/2/3/4/5(RAT)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50020211(CHEMBL216353 | D-Phec(-Cys-Tyr-D-Trp-Lys-Thr-Pen-)...)
Affinity DataIC50:  1.80E+3nMAssay Description:Binding affinity in competition with [125I]- CGP-23996 in somatostatin receptor binding to rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1/2/3/4/5(RAT)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50020216(CHEMBL413831 | D-Phec(-Cys-Tyr-D-Trp-Lys-Thr-Pen)-...)
Affinity DataIC50:  1.89E+3nMAssay Description:Binding affinity in competition with [125I]- CGP-23996 in somatostatin receptor binding to rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1/2/3/4/5(RAT)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50020198(CHEMBL308471 | D-Phec(-Cys-Tyr-D-Trp-Lys-Thr-Pen-)...)
Affinity DataIC50:  1.94E+3nMAssay Description:Binding affinity in competition with [125I]- CGP-23996 in somatostatin receptor binding to rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1/2/3/4/5(RAT)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50020200(CHEMBL405672 | D-Ticc(-Cys-Tyr-D-Typ-Lys-Thr-Pen-)...)
Affinity DataIC50:  1.99E+3nMAssay Description:Binding affinity in competition with [125I]- CGP-23996 in somatostatin receptor binding to rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1/2/3/4/5(RAT)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50020214(CHEMBL302596 | D-Phec(-Cys-Tyr-D-Trp-Lys-D-Pen-)Th...)
Affinity DataIC50:  6.10E+3nMAssay Description:Binding affinity in competition with [125I]- CGP-23996 in somatostatin receptor binding to rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1/2/3/4/5(RAT)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50214420(CHEMBL330352)
Affinity DataIC50:  6.50E+3nMAssay Description:Compound was tested for its inhibitory effect against somatostatin receptor in rat cortex membrane using [125I]Tyr3-octreotide as the radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetSomatostatin receptor type 1/2/3/4/5(RAT)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50214420(CHEMBL330352)
Affinity DataIC50:  7.00E+3nMAssay Description:Compound was tested for its inhibitory effect against somatostatin receptor in rat cortex membrane using [125I]Tyr3-octreotide as the radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetSomatostatin receptor type 1/2/3/4/5(RAT)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50214420(CHEMBL330352)
Affinity DataIC50:  7.00E+3nMAssay Description:Compound was tested for its inhibitory effect against somatostatin receptor in rat cortex membrane using [125I]Tyr3-octreotide as the radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetSomatostatin receptor type 1/2/3/4/5(RAT)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50020199(CHEMBL441164 | D-N-Me-Phec(-Cys-Tyr-D-Trp-Orn-Thr-...)
Affinity DataIC50:  8.05E+3nMAssay Description:Binding affinity in competition with [125I]- CGP-23996 in somatostatin receptor binding to rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1/2/3/4/5(RAT)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50020212(CHEMBL405244 | D-Phec(-Cys-Tyr-D-Trp-Lys-Thr-Pen-)...)
Affinity DataIC50:  8.30E+3nMAssay Description:Binding affinity in competition with [125I]- CGP-23996 in somatostatin receptor binding to rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1/2/3/4/5(RAT)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50020208(CHEMBL1795717 | TCTAP)
Affinity DataIC50:  8.45E+3nMAssay Description:Binding affinity in competition with [125I]- CGP-23996 in somatostatin receptor binding to rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1/2/3/4/5(RAT)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50213874(CHEMBL432503)
Affinity DataIC50:  1.00E+4nMAssay Description:Compound was tested for its potency to displace 3-[125I]- - Tyr11-SRIF-14 from somatostatin receptor on membranes of rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails
TargetSomatostatin receptor type 1/2/3/4/5(RAT)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50020204(CHEMBL66403 | D-Phec(-Cys-Tyr-Asn-Pen-)Thr-NH2)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity in competition with [125I]- CGP-23996 in somatostatin receptor binding to rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1/2/3/4/5(RAT)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50213872(CHEMBL47019)
Affinity DataIC50:  1.10E+4nMAssay Description:Compound was tested for its potency to displace 3-[125I]- - Tyr11-SRIF-14 from somatostatin receptor on membranes of rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails
TargetSomatostatin receptor type 1/2/3/4/5(RAT)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50213869(CHEMBL3037859)
Affinity DataIC50:  1.20E+4nMAssay Description:Compound was tested for its potency to displace 3-[125I]- - Tyr11-SRIF-14 from somatostatin receptor on membranes of rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails
TargetSomatostatin receptor type 1/2/3/4/5(RAT)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50213871(CHEMBL47648)
Affinity DataIC50:  1.20E+4nMAssay Description:Compound was tested for its potency to displace 3-[125I]- - Tyr11-SRIF-14 from somatostatin receptor on membranes of rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails
TargetSomatostatin receptor type 1/2/3/4/5(RAT)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50452485(CHEMBL2369462)
Affinity DataIC50:  1.36E+4nMAssay Description:Binding affinity in competition with [125I]- CGP-23996 in somatostatin receptor binding to rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1/2/3/4/5(RAT)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50213870(CHEMBL294905)
Affinity DataIC50:  1.40E+4nMAssay Description:Compound was tested for its potency to displace 3-[125I]- - Tyr11-SRIF-14 from somatostatin receptor on membranes of rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails
TargetSomatostatin receptor type 1/2/3/4/5(RAT)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50213873(CHEMBL45323)
Affinity DataIC50:  1.50E+4nMAssay Description:Compound was tested for its potency to displace 3-[125I]- - Tyr11-SRIF-14 from somatostatin receptor on membranes of rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails
TargetSomatostatin receptor type 1/2/3/4/5(RAT)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50020207(CHEMBL2369473 | Gly-D-Ticc(-Cys-Tyr-D-Trp-Orn-Thr-...)
Affinity DataIC50:  1.94E+4nMAssay Description:Binding affinity in competition with [125I]- CGP-23996 in somatostatin receptor binding to rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1/2/3/4/5(RAT)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50020197(CHEMBL2369475 | TCTOP)
Affinity DataIC50:  2.04E+4nMAssay Description:Binding affinity in competition with [125I]- CGP-23996 in somatostatin receptor binding to rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1/2/3/4/5(RAT)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50212468(CHEMBL28415)
Affinity DataIC50:  2.30E+4nMAssay Description:Radioligand binding studies on rat cortex membranes using 125 I-Tyrs-octreotide as ligand was determinedMore data for this Ligand-Target Pair
In DepthDetails
TargetSomatostatin receptor type 1/2/3/4/5(RAT)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50020203(CHEMBL2369474 | D-Ticc(-Cys-Tyr-D-Trp-Lys-Pen-)Thr...)
Affinity DataIC50:  3.43E+4nMAssay Description:Binding affinity in competition with [125I]- CGP-23996 in somatostatin receptor binding to rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1/2/3/4/5(RAT)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50020215(CHEMBL541457 | D-Phec(-Cys-Tyr-D-Trp-Orn-The-Pen-)...)
Affinity DataIC50:  4.73E+4nMAssay Description:Binding affinity in competition with [125I]- CGP-23996 in somatostatin receptor binding to rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1/2/3/4/5(RAT)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50020206(CHEMBL266829 | CTOP)
Affinity DataIC50:  4.77E+4nMAssay Description:Binding affinity in competition with [125I]- CGP-23996 in somatostatin receptor binding to rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed