Compile Data Set for Download or QSAR
maximum 50k data
Found 353 of ic50 for UniProtKB: P48974
TargetVasopressin V1b receptor(RAT)
Msd

Curated by ChEMBL
LigandPNGBDBM50338810(CHEMBL1684573 | N-isopropyl-2-(2-(3-methoxyphenyl)...)
Affinity DataIC50:  2nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in CHO cells by whole cell binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50137948(Biphenyl-2-carboxylic acid [2-[3-(4-methyl-[1,4]di...)
Affinity DataIC50:  2nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50137945(Biphenyl-2-carboxylic acid [2-[4-(4-methyl-piperaz...)
Affinity DataIC50:  3nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(RAT)
Msd

Curated by ChEMBL
LigandPNGBDBM50338811(2-(2-(3-chlorophenyl)-4-oxo-6-(3-(piperidin-1-yl)p...)
Affinity DataIC50:  4nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in CHO cells by whole cell binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50137953(Biphenyl-2-carboxylic acid [2-[4-(4-diethylamino-p...)
Affinity DataIC50:  4nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50137940(Biphenyl-2-carboxylic acid [2-[4-(4-dimethylamino-...)
Affinity DataIC50:  6nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50291329(8-arginine vasopressin trisulphide | CHEMBL267405)
Affinity DataIC50:  9.5nMAssay Description:Tested for the TYR(Me)2 arginine-vasopressin as radioligand at 0.3 nM in A7r5 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetVasopressin V1a/V1b receptor(RAT)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM35667(AVP | CHEMBL373742 | US10131692, 44 (AVP) | [3H]Ar...)
Affinity DataIC50:  10nMAssay Description:Tested for the TYR(Me)2 arginine-vasopressin as radioligand at 0.3 nM in A7r5 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetVasopressin V1a/V1b receptor(RAT)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50137946(Biphenyl-2-carboxylic acid [2-[2-(4-dimethylamino-...)
Affinity DataIC50:  20nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50137951(Biphenyl-2-carboxylic acid [2-{4-[(2-dimethylamino...)
Affinity DataIC50:  20nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50137949(Biphenyl-2-carboxylic acid [2-[4-(4-methyl-[1,4]di...)
Affinity DataIC50:  20nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50137942(Biphenyl-2-carboxylic acid [2-(4-[1,4']bipiperidin...)
Affinity DataIC50:  20nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50137956(Biphenyl-2-carboxylic acid [2-[4-(4-methyl-piperaz...)
Affinity DataIC50:  20nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50043204(1N-[2-hydroxy-7,7-dimethyl-1-spiro[1H-indene-1,4'-...)
Affinity DataIC50:  67nMAssay Description:Inhibition of radioligand [3H]AVP binding to the vasopressin V1 receptor in rat liver tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50043080(3-[7,7-dimethyl-1-spiro[2,3-dihydro-1H-indene-1,4'...)
Affinity DataIC50:  110nMAssay Description:Inhibition of radioligand [3H]AVP binding to the vasopressin V1 receptor in rat liver tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50043141(5-(3-amino-1H-1,2,4-triazol-5-ylaminomethyl)-3-[7,...)
Affinity DataIC50:  120nMAssay Description:Inhibition of radioligand [3H]AVP binding to the vasopressin V1 receptor in rat liver tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50043114(3-{1-[7,7-dimethyl-1-spiro[2,3-dihydro-1H-indene-1...)
Affinity DataIC50:  160nMAssay Description:Inhibition of radioligand [3H]AVP binding to the vasopressin V1 receptor in rat liver tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50137941(Biphenyl-2-carboxylic acid {4-[8-(2-pyrrolidin-1-y...)
Affinity DataIC50:  200nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50204026(CHEMBL369150)
Affinity DataIC50:  200nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50137943(Biphenyl-2-carboxylic acid (4-{8-[2-(4-methyl-pipe...)
Affinity DataIC50:  200nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(RAT)
Msd

Curated by ChEMBL
LigandPNGBDBM50325847(CHEMBL1223814 | N-(cyclopropylmethyl)-2-(6-(3-morp...)
Affinity DataIC50:  210nMAssay Description:Displacement of [3H]AVP from rat vasopressin V3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50043180(1N-[2-hydroxy-7,7-dimethyl-1-spiro[1H-indene-1,4'-...)
Affinity DataIC50:  290nMAssay Description:Inhibition of radioligand [3H]AVP binding to the vasopressin V1 receptor in rat liver tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50043075(1N-[7,7-dimethyl-1-spiro[2,3-dihydro-1H-indene-1,4...)
Affinity DataIC50: >300nMAssay Description:Inhibition of radioligand [3H]AVP binding to the vasopressin V1 receptor in rat liver tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50043106(CHEMBL335886 | methyl 3-[2-hydroxy-7,7-dimethyl-1-...)
Affinity DataIC50: >300nMAssay Description:Inhibition of radioligand [3H]AVP binding to the vasopressin V1 receptor in rat liver tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50043155(1N-[7,7-dimethyl-1-spiro[2,3-dihydro-1H-indene-1,4...)
Affinity DataIC50: >300nMAssay Description:Inhibition of radioligand [3H]AVP binding to the vasopressin V1 receptor in rat liver tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50043090(1N-[2-hydroxy-7,7-dimethyl-1-spiro[1H-indene-1,4'-...)
Affinity DataIC50: >300nMAssay Description:Inhibition of radioligand [3H]AVP binding to the vasopressin V1 receptor in rat liver tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50043145(3N-[2-hydroxy-7,7-dimethyl-1-spiro[1H-indene-1,4'-...)
Affinity DataIC50: >300nMAssay Description:Inhibition of radioligand [3H]AVP binding to the vasopressin V1 receptor in rat liver tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50043117(1-[7,7-dimethyl-1-spiro[2,3-dihydro-1H-indene-1,4'...)
Affinity DataIC50: >300nMAssay Description:Inhibition of radioligand [3H]AVP binding to the vasopressin V1 receptor in rat liver tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50043189(1N-[7,7-dimethyl-1-spiro[2,3-dihydro-1H-indene-1,4...)
Affinity DataIC50: >300nMAssay Description:Inhibition of radioligand [3H]AVP binding to the vasopressin V1 receptor in rat liver tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50043055(2-{3-[7,7-dimethyl-1-spiro[2,3-dihydro-1H-indene-1...)
Affinity DataIC50: >300nMAssay Description:Inhibition of radioligand [3H]AVP binding to the vasopressin V1 receptor in rat liver tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50043116(1N-{2-[2-hydroxy-7,7-dimethyl-1-spiro[1H-indene-1,...)
Affinity DataIC50: >300nMAssay Description:Inhibition of radioligand [3H]AVP binding to the vasopressin V1 receptor in rat liver tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50043059(1N-[2-hydroxy-7,7-dimethyl-1-spiro[1H-indene-1,4'-...)
Affinity DataIC50: >300nMAssay Description:Inhibition of radioligand [3H]AVP binding to the vasopressin V1 receptor in rat liver tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50137954(Biphenyl-2-carboxylic acid {4-[8-(2-dimethylamino-...)
Affinity DataIC50:  300nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50043088(3-[7,7-dimethyl-1-spiro[2,3-dihydro-1H-indene-1,4'...)
Affinity DataIC50: >300nMAssay Description:Inhibition of radioligand [3H]-AVP binding to the vasopressin V2 receptor in rat kidney tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50043143(1N-[2-hydroxy-7,7-dimethyl-1-spiro[1H-indene-1,4'-...)
Affinity DataIC50:  310nMAssay Description:Inhibition of radioligand [3H]-AVP binding to the vasopressin V2 receptor in rat kidney tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50043120(1N-[7,7-dimethyl-1-spiro[2,3-dihydro-1H-indene-1,4...)
Affinity DataIC50:  320nMAssay Description:Inhibition of radioligand [3H]AVP binding to the vasopressin V1 receptor in rat liver tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50043093(3-[7,7-dimethyl-1-spiro[2,3-dihydro-1H-indene-1,4'...)
Affinity DataIC50:  370nMAssay Description:Inhibition of radioligand [3H]AVP binding to the vasopressin V1 receptor in rat liver tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50043077(2-{1-[7,7-dimethyl-1-spiro[2,3-dihydro-1H-indene-1...)
Affinity DataIC50:  410nMAssay Description:Inhibition of radioligand [3H]AVP binding to the vasopressin V1 receptor in rat liver tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50043118(3-[7,7-dimethyl-1-spiro[2,3-dihydro-1H-indene-1,4'...)
Affinity DataIC50:  420nMAssay Description:Inhibition of radioligand [3H]AVP binding to the vasopressin V1 receptor in rat liver tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50043118(3-[7,7-dimethyl-1-spiro[2,3-dihydro-1H-indene-1,4'...)
Affinity DataIC50:  420nMAssay Description:Inhibition of radioligand [3H]AVP binding to the vasopressin V1 receptor in rat liver tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50043118(3-[7,7-dimethyl-1-spiro[2,3-dihydro-1H-indene-1,4'...)
Affinity DataIC50:  420nMAssay Description:Inhibition of radioligand [3H]AVP binding to the vasopressin V1 receptor in rat liver tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50043092(1N-[2-hydroxy-7,7-dimethyl-1-spiro[1H-indene-1,4'-...)
Affinity DataIC50:  430nMAssay Description:Inhibition of radioligand [3H]AVP binding to the vasopressin V1 receptor in rat liver tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50043102(1N-[7,7-dimethyl-1-spiro[2,3-dihydro-1H-indene-1,4...)
Affinity DataIC50:  440nMAssay Description:Inhibition of radioligand [3H]AVP binding to the vasopressin V1 receptor in rat liver tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50043186(1N-[7,7-dimethyl-1-spiro[2,3-dihydro-1H-indene-1,4...)
Affinity DataIC50:  440nMAssay Description:Inhibition of radioligand [3H]AVP binding to the vasopressin V1 receptor in rat liver tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50043136(2N-[2-hydroxy-7,7-dimethyl-1-spiro[1H-indene-1,4'-...)
Affinity DataIC50:  470nMAssay Description:Inhibition of radioligand [3H]AVP binding to the vasopressin V1 receptor in rat liver tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50043165(1N-[2-hydroxy-7,7-dimethyl-1-spiro[1H-indene-1,4'-...)
Affinity DataIC50:  480nMAssay Description:Inhibition of radioligand [3H]AVP binding to the vasopressin V1 receptor in rat liver tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50043060(1N-[7,7-dimethyl-1-spiro[2,3-dihydro-1H-indene-1,4...)
Affinity DataIC50:  490nMAssay Description:Inhibition of radioligand [3H]AVP binding to the vasopressin V1 receptor in rat liver tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50043197(5-aminomethyl-3-[7,7-dimethyl-1-spiro[2,3-dihydro-...)
Affinity DataIC50:  490nMAssay Description:Inhibition of radioligand [3H]AVP binding to the vasopressin V1 receptor in rat liver tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50137950(Biphenyl-2-carboxylic acid [4-(8-pyridin-3-ylmethy...)
Affinity DataIC50:  500nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50043148(3-[7,7-dimethyl-1-spiro[2,3-dihydro-1H-indene-1,4'...)
Affinity DataIC50:  500nMAssay Description:Inhibition of radioligand [3H]AVP binding to the vasopressin V1 receptor in rat liver tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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