Compile Data Set for Download or QSAR
maximum 50k data
Found 70 of ic50 for UniProtKB: O08786
TargetCholecystokinin receptor type A(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284146(CHEMBL355608 | [(S)-1-[(S)-1-((R)-3-Benzyl-5-oxo-p...)
Affinity DataIC50:  14nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [125I]- CCK-8 to CCK receptors on mouse pancreatic membranes (CCK-A)More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284148(CHEMBL171310 | [(S)-1-[(S)-1-((R)-3-Benzyl-5-oxo-p...)
Affinity DataIC50:  46nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [125I]- CCK-8 to CCK receptors on mouse pancreatic membranes (CCK-A)More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284156(CHEMBL169174 | [(S)-1-[(S)-1-((S)-3-Benzyl-5-oxo-p...)
Affinity DataIC50:  64nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [125I]- CCK-8 to CCK receptors on mouse pancreatic membranes (CCK-A)More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287255(CHEMBL30821 | N-[2-(2-Guanidino-thiazol-4-ylmethyl...)
Affinity DataIC50:  120nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287253(6-(2-{3-[3-((R)-1-Methyl-2-oxo-5-phenyl-2,3-dihydr...)
Affinity DataIC50:  190nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287234(3-(2-{3-[3-((R)-1-Methyl-2-oxo-5-phenyl-2,3-dihydr...)
Affinity DataIC50:  190nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284147(CHEMBL354363 | [(S)-1-[(S)-1-((S)-3-Benzyl-5-oxo-p...)
Affinity DataIC50:  270nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [125I]- CCK-8 to CCK receptors on mouse pancreatic membranes (CCK-A)More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287265(CHEMBL406844 | {2-[3-(3-Piperidin-1-ylmethyl-pheno...)
Affinity DataIC50:  310nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287250(4-(2-{3-[3-((R)-1-Methyl-2-oxo-5-phenyl-2,3-dihydr...)
Affinity DataIC50:  330nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287251(CHEMBL262125 | N-[2-(2-Guanidino-thiazol-4-ylmethy...)
Affinity DataIC50:  330nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287256(6-(2-{3-[3-((R)-1-Methyl-2-oxo-5-phenyl-2,3-dihydr...)
Affinity DataIC50:  340nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287233(CHEMBL280980 | N-[2-(2-Guanidino-thiazol-4-ylmethy...)
Affinity DataIC50:  380nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287259(CHEMBL286908 | N-[2-(2-Guanidino-thiazol-4-ylmethy...)
Affinity DataIC50:  390nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287244(2-[2-Oxo-5-phenyl-3-(3-m-tolyl-ureido)-2,3-dihydro...)
Affinity DataIC50:  430nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284160(CHEMBL169178 | [(S)-1-[(S)-1-((S)-3-Benzyl-5-oxo-p...)
Affinity DataIC50:  430nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [125I]- CCK-8 to CCK receptors on mouse pancreatic membranes (CCK-A)More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284161((E)-N-[(S)-1-[(S)-1-((S)-3-Benzyl-5-oxo-piperazine...)
Affinity DataIC50:  520nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [125I]- CCK-8 to CCK receptors on mouse pancreatic membranes (CCK-A)More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287248(CHEMBL30430 | N-[2-(2-Guanidino-thiazol-4-ylmethyl...)
Affinity DataIC50:  560nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284151(((2S,5S)-1-{(S)-2-[(S)-2-tert-Butoxycarbonylamino-...)
Affinity DataIC50:  630nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [125I]- CCK-8 to CCK receptors on mouse pancreatic membranes (CCK-A)More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287238(6-{2-[2-Oxo-5-phenyl-3-(3-m-tolyl-ureido)-2,3-dihy...)
Affinity DataIC50:  650nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287236(CHEMBL286907 | N-[2-(2-Guanidino-thiazol-4-ylmethy...)
Affinity DataIC50:  720nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287272(CHEMBL33412 | [2-(4-{2-[3-(3-Piperidin-1-ylmethyl-...)
Affinity DataIC50:  740nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287254(CHEMBL281082 | N-{[2-(2-Guanidino-thiazol-4-ylmeth...)
Affinity DataIC50:  760nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284158(((2S,5S)-5-Benzyl-1-{(S)-2-[(S)-2-tert-butoxycarbo...)
Affinity DataIC50:  840nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [125I]- CCK-8 to CCK receptors on mouse pancreatic membranes (CCK-A)More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287246(4-{2-[2-Oxo-5-phenyl-3-(3-m-tolyl-ureido)-2,3-dihy...)
Affinity DataIC50:  900nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287271((3-{2-[2-(2,2-Diamino-vinyl)-thiazol-4-ylmethylsul...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287239(CHEMBL30656 | N-{[2-(2-Guanidino-thiazol-4-ylmethy...)
Affinity DataIC50:  1.09E+3nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287252(3-{2-[2-Oxo-5-phenyl-3-(3-m-tolyl-ureido)-2,3-dihy...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287261((3-{2-[2-(2,2-Diamino-vinyl)-thiazol-4-ylmethylsul...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284159(((2S,5S)-5-Benzyl-1-{(S)-2-[(1H-indole-3-carbonyl)...)
Affinity DataIC50:  1.40E+3nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [125I]- CCK-8 to CCK receptors on mouse pancreatic membranes (CCK-A)More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287273(CHEMBL285719 | [3-(4-{2-[3-(3-Piperidin-1-ylmethyl...)
Affinity DataIC50:  1.65E+3nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287245(CHEMBL285586 | N-[2-(2-Guanidino-thiazol-4-ylmethy...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287232(CHEMBL31726 | N-[2-(2-Guanidino-thiazol-4-ylmethyl...)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287258(3-[3-((R)-1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1H-b...)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284150(((2R,5S)-5-Benzyl-1-{(S)-2-[(S)-2-tert-butoxycarbo...)
Affinity DataIC50:  2.80E+3nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [125I]- CCK-8 to CCK receptors on mouse pancreatic membranes (CCK-A)More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287270(CHEMBL432671 | [(2-{2-[2-(2,2-Diamino-vinyl)-thiaz...)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50019202(7-Chloro-3-(1H-indol-3-ylmethyl)-5-phenyl-1,3-dihy...)
Affinity DataIC50:  3.40E+3nMAssay Description:Half-maximal inhibition of [125I]CCK-33 binding to cholecystokinin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50280054((S)-3-((S)-2-((S)-2-(tert-butoxycarbonyl)-3-(1H-in...)
Affinity DataIC50:  3.50E+3nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [125I]- CCK-8 to CCK receptors on mouse pancreatic membranes (CCK-A)More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50280054((S)-3-((S)-2-((S)-2-(tert-butoxycarbonyl)-3-(1H-in...)
Affinity DataIC50:  3.50E+3nMAssay Description:Concentration of compound required to inhibit binding of [125I]J-BH-CCK-8 radioligand to CCKA in mouse pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284155(((2S,5R)-5-Benzyl-1-{(S)-2-[(S)-2-tert-butoxycarbo...)
Affinity DataIC50:  3.60E+3nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [125I]- CCK-8 to CCK receptors on mouse pancreatic membranes (CCK-A)More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287269(CHEMBL33698 | {3-[3-(3-Piperidin-1-ylmethyl-phenox...)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287240(6-(2-{3-[1-Methyl-2-oxo-3-(3-m-tolyl-ureido)-2,3-d...)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287264(CHEMBL287295 | {3-[3-(3-Piperidin-1-ylmethyl-pheno...)
Affinity DataIC50:  3.80E+3nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287257(2-{3-[3-((R)-1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1...)
Affinity DataIC50:  4.10E+3nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287267(CHEMBL284975 | {2-[3-(3-Piperidin-1-ylmethyl-pheno...)
Affinity DataIC50:  4.20E+3nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287260((3-{2-[2-(2,2-Diamino-vinyl)-thiazol-4-ylmethylsul...)
Affinity DataIC50:  4.40E+3nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287262(CHEMBL33743 | {3-[3-(3-Piperidin-1-ylmethyl-phenox...)
Affinity DataIC50:  4.60E+3nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287241(CHEMBL285746 | N-[2-(2-Guanidino-thiazol-4-ylmethy...)
Affinity DataIC50:  4.80E+3nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287266(CHEMBL290122 | {3-[3-(3-Piperidin-1-ylmethyl-pheno...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287243(2-{3-[1-Methyl-2-oxo-3-(3-m-tolyl-ureido)-2,3-dihy...)
Affinity DataIC50:  5.20E+3nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287237(CHEMBL29888 | N-[2-(2-Guanidino-thiazol-4-ylmethyl...)
Affinity DataIC50:  5.40E+3nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
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