Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Transient receptor potential cation channel subfamily V member 5 (Homo sapiens) | BDBM50550078![]() (CHEMBL4777551) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar | PC cid PC sid PDB UniChem | PubMed | n/a | n/a | 560 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bern Curated by ChEMBL | Assay Description Inhibition of human TRPV5 expressed in HEK293 cells assessed as reduction in Cd2+ influx by calcium-5 fluorescence dye-based FLIPR assay | RSC Med Chem 11: 1032-1040 (2020) | |||||||||||
More data for this Ligand-Target Pair |