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Compile Data Set for Download or QSAR

Found 3 hits of affinity data for UniProtKB/TrEMBL: Q9H3H5   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
UDP-N-acetylglucosamine--dolichyl-phosphate N-acetylglucosaminephosphotransferase


(Homo sapiens)
BDBM50553598
PNG
(CHEMBL4776441)
Show SMILES NC[C@H]1O[C@@H](O[C@@H]([C@H](NCCCC(=O)NCc2ccc(cc2)N2CCC(CC2)Oc2ccc(OC(F)(F)F)cc2)C(N)=O)[C@H]2O[C@H]([C@H](O)[C@@H]2O)n2ccc(=O)[nH]c2=O)[C@H](O)[C@@H]1O
PDB
MMDB

Reactome pathway
KEGG

UniProtKB/SwissProt

DrugBank
GoogleScholar
PC cid
PC sid
UniChem
PubMed
n/an/a 10n/an/an/an/an/an/a



University of Tennessee Health Science Center

Curated by ChEMBL


Assay Description
Inhibition of human DPAGT1 expressed in HEK293 (Expi293) cells incubated for 2 hrs using UDP-GlcN-Cg-FITC and alpha-dihydroundecap-renyl phosphate by...


J Med Chem 63: 10855-10878 (2020)

More data for this
Ligand-Target Pair
UDP-N-acetylglucosamine--dolichyl-phosphate N-acetylglucosaminephosphotransferase


(Homo sapiens)
BDBM50553592
PNG
(CHEMBL4753142)
Show SMILES CO[C@H]1[C@@H](O)[C@@H](O[C@@H]1[C@@H](O[C@H]1OC(=C[C@H](O)[C@@H]1O)C(=O)NCc1ccc(cc1)N1CCC(CC1)Oc1ccc(OC(F)(F)F)cc1)C(N)=O)n1ccc(=O)[nH]c1=O
PDB
MMDB

Reactome pathway
KEGG

UniProtKB/SwissProt

DrugBank
GoogleScholar
PC cid
PC sid
UniChem
PubMed
n/an/a 200n/an/an/an/an/an/a



University of Tennessee Health Science Center

Curated by ChEMBL


Assay Description
Inhibition of human DPAGT1 expressed in HEK293 (Expi293) cells incubated for 2 hrs using UDP-GlcN-Cg-FITC and alpha-dihydroundecap-renyl phosphate by...


J Med Chem 63: 10855-10878 (2020)

More data for this
Ligand-Target Pair
UDP-N-acetylglucosamine--dolichyl-phosphate N-acetylglucosaminephosphotransferase


(Homo sapiens)
BDBM50553593
PNG
(CHEMBL4752744)
Show SMILES CO[C@@H]1[C@H](O)[C@H](O[C@H]1n1ccc(=O)[nH]c1=O)[C@@H](O[C@H]1OC(=C[C@H](O)[C@@H]1O)C(=O)NCc1ccc(cc1)N1CCC(CC1)Oc1ccc(OC(F)(F)F)cc1)C(N)=O
PDB
MMDB

Reactome pathway
KEGG

UniProtKB/SwissProt

DrugBank
GoogleScholar
PC cid
PC sid
UniChem
PubMed
n/an/a 600n/an/an/an/an/an/a



University of Tennessee Health Science Center

Curated by ChEMBL


Assay Description
Inhibition of human DPAGT1 expressed in HEK293 (Expi293) cells incubated for 2 hrs using UDP-GlcN-Cg-FITC and alpha-dihydroundecap-renyl phosphate by...


J Med Chem 63: 10855-10878 (2020)

More data for this
Ligand-Target Pair