Compile Data Set for Download or QSAR
maximum 50k data
Found 208 of ec50 data for polymerid = 50000944
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50462106(CHEMBL3736108)
Affinity DataEC50:  7nMAssay Description:Agonist activity at C3aR in human MDM cells assessed as inhibition of C3a-induced Ca2+ response measured for 60 secs by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50462106(CHEMBL3736108)
Affinity DataEC50:  7nMAssay Description:Agonist activity at C3aR in HMDM assessed as induction of Ca2+ release measured for 5 mins by Fluo-3 AM dye-based fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50462106(CHEMBL3736108)
Affinity DataEC50:  7.10nMAssay Description:Agonist activity at C3aR in human MDM cells assessed as inhibition of C3a-induced Ca2+ response measured for 60 secs by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50499185(CHEMBL3736125)
Affinity DataEC50:  7.60nMAssay Description:Agonist activity at C3aR in human MDM cells assessed as inhibition of C3a-induced Ca2+ response measured for 60 secs by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50499185(CHEMBL3736125)
Affinity DataEC50:  8nMAssay Description:Agonist activity at C3aR in human MDM cells assessed as inhibition of C3a-induced Ca2+ response measured for 60 secs by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50587350(CHEMBL5076900)
Affinity DataEC50:  9nMAssay Description:Agonist activity at human C3aR expressed in CHO cells assessed as induction of ERK1/2 phosphorylation at Thr202/Tyr204 residues incubated for 10 mins...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50587347(CHEMBL5081621)
Affinity DataEC50:  11nMAssay Description:Agonist activity at human C3aR expressed in CHO cells assessed as induction of ERK1/2 phosphorylation at Thr202/Tyr204 residues incubated for 10 mins...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50462105(CHEMBL4239035)
Affinity DataEC50:  15nMAssay Description:Agonist activity at C3aR in HMDM assessed as induction of Ca2+ releaseMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50499169(CHEMBL3735507)
Affinity DataEC50:  17nMAssay Description:Agonist activity at C3aR in human MDM cells assessed as inhibition of C3a-induced Ca2+ response measured for 60 secs by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50499169(CHEMBL3735507)
Affinity DataEC50:  17nMAssay Description:Agonist activity at C3aR in human MDM cells assessed as inhibition of C3a-induced Ca2+ response measured for 60 secs by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50499168(CHEMBL3735760)
Affinity DataEC50:  19nMAssay Description:Agonist activity at C3aR in human MDM cells assessed as inhibition of C3a-induced Ca2+ response measured for 60 secs by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50499168(CHEMBL3735760)
Affinity DataEC50:  19nMAssay Description:Agonist activity at C3aR in human MDM cells assessed as inhibition of C3a-induced Ca2+ response measured for 60 secs by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50028696(CHEMBL3342689)
Affinity DataEC50:  25nMAssay Description:Agonist activity against C3AR in HMDMs assessed as increase in intracellular calcium release by Fluo-3 AM dye based FLIPR assay relative to 1 uM C3aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50028696(CHEMBL3342689)
Affinity DataEC50:  25.1nMAssay Description:Agonist activity against C3AR in HMDMs assessed as increase in intracellular calcium release by Fluo-3 AM dye based FLIPR assay relative to 1 uM C3aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50389001(CHEMBL2064016)
Affinity DataEC50:  25.1nMAssay Description:Agonist activity at human C3a receptor expressed in RBL-2H3 cells assessed as beta-hexosaminidase activity in cell supernatant by degranulation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50499172(CHEMBL3736239)
Affinity DataEC50:  27nMAssay Description:Agonist activity at C3aR in human MDM cells assessed as inhibition of C3a-induced Ca2+ response measured for 60 secs by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50499172(CHEMBL3736239)
Affinity DataEC50:  27nMAssay Description:Agonist activity at C3aR in human MDM cells assessed as inhibition of C3a-induced Ca2+ response measured for 60 secs by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50388995(CHEMBL2064019)
Affinity DataEC50:  35.5nMAssay Description:Agonist activity at human C3a receptor expressed in RBL-2H3 cells assessed as beta-hexosaminidase activity in cell supernatant by degranulation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50587351(CHEMBL5080234)
Affinity DataEC50:  37nMAssay Description:Agonist activity at human C3aR expressed in CHO cells assessed as induction of ERK1/2 phosphorylation at Thr202/Tyr204 residues incubated for 10 mins...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50028697(CHEMBL3342690)
Affinity DataEC50:  40nMAssay Description:Agonist activity against C3AR in HMDMs assessed as increase in intracellular calcium release by Fluo-3 AM dye based FLIPR assay relative to 1 uM C3aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50028697(CHEMBL3342690)
Affinity DataEC50:  40nMAssay Description:Agonist activity against C3AR in HMDMs assessed as increase in intracellular calcium release by Fluo-3 AM dye based FLIPR assay relative to 1 uM C3aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50499166(CHEMBL3735048)
Affinity DataEC50:  41nMAssay Description:Agonist activity at C3aR in human MDM cells assessed as inhibition of C3a-induced Ca2+ response measured for 60 secs by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50499166(CHEMBL3735048)
Affinity DataEC50:  41nMAssay Description:Agonist activity at C3aR in human MDM cells assessed as inhibition of C3a-induced Ca2+ response measured for 60 secs by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50499171(CHEMBL3735339)
Affinity DataEC50:  45nMAssay Description:Agonist activity at C3aR in human MDM cells assessed as inhibition of C3a-induced Ca2+ response measured for 60 secs by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50520316(CHEMBL4445758)
Affinity DataEC50:  46nMAssay Description:Agonist activity at C3a receptor in human MDM cells assessed as induction of intracellular calcium release measured at 1 sec interval for => 200 secs...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50520316(CHEMBL4445758)
Affinity DataEC50:  50nMAssay Description:Agonist activity at C3a receptor in human MDM cells assessed as induction of intracellular calcium release measured at 1 sec interval for => 200 secs...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50520303(CHEMBL4459830)
Affinity DataEC50:  50nMAssay Description:Agonist activity at C3a receptor in human MDM cells assessed as induction of intracellular calcium release measured at 1 sec interval for => 200 secs...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50520303(CHEMBL4459830)
Affinity DataEC50:  50nMAssay Description:Agonist activity at C3a receptor in human MDM cells assessed as induction of intracellular calcium release measured at 1 sec interval for => 200 secs...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50499183(CHEMBL3735764)
Affinity DataEC50:  54nMAssay Description:Agonist activity at C3aR in human MDM cells assessed as inhibition of C3a-induced Ca2+ response measured for 60 secs by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50499183(CHEMBL3735764)
Affinity DataEC50:  55nMAssay Description:Agonist activity at C3aR in human MDM cells assessed as inhibition of C3a-induced Ca2+ response measured for 60 secs by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50587346(CHEMBL5085196)
Affinity DataEC50:  62nMAssay Description:Agonist activity at human C3aR expressed in CHO cells assessed as induction of ERK1/2 phosphorylation at Thr202/Tyr204 residues incubated for 10 mins...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50520305(CHEMBL4559976)
Affinity DataEC50:  63nMAssay Description:Agonist activity at C3a receptor in human MDM cells assessed as induction of intracellular calcium release measured at 1 sec interval for => 200 secs...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50520305(CHEMBL4559976)
Affinity DataEC50:  63.1nMAssay Description:Agonist activity at C3a receptor in human MDM cells assessed as induction of intracellular calcium release measured at 1 sec interval for => 200 secs...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50389002(CHEMBL2064017)
Affinity DataEC50:  66.1nMAssay Description:Agonist activity at human C3a receptor expressed in RBL-2H3 cells assessed as beta-hexosaminidase activity in cell supernatant by degranulation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50499184(CHEMBL3735993)
Affinity DataEC50:  72nMAssay Description:Agonist activity at C3aR in human MDM cells assessed as inhibition of C3a-induced Ca2+ response measured for 60 secs by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50499184(CHEMBL3735993)
Affinity DataEC50:  73nMAssay Description:Agonist activity at C3aR in human MDM cells assessed as inhibition of C3a-induced Ca2+ response measured for 60 secs by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50389004(CHEMBL2064021)
Affinity DataEC50:  81.3nMAssay Description:Agonist activity at human C3a receptor expressed in RBL-2H3 cells assessed as beta-hexosaminidase activity in cell supernatant by degranulation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50028695(CHEMBL3342688)
Affinity DataEC50:  126nMAssay Description:Agonist activity against C3AR in HMDMs assessed as increase in intracellular calcium release by Fluo-3 AM dye based FLIPR assay relative to 1 uM C3aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50587343(CHEMBL5080181)
Affinity DataEC50:  129nMAssay Description:Agonist activity at human C3aR expressed in CHO cells assessed as induction of ERK1/2 phosphorylation at Thr202/Tyr204 residues incubated for 10 mins...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50322618((3S,6R,9S)-14-amino-2-((S)-1-((S)-2-((S)-1-((S)-6-...)
Affinity DataEC50:  130nMAssay Description:Agonist activity at human C3a receptor in human U937 cells assessed as induction of intracellular calcium releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50028695(CHEMBL3342688)
Affinity DataEC50:  130nMAssay Description:Agonist activity against C3AR in HMDMs assessed as increase in intracellular calcium release by Fluo-3 AM dye based FLIPR assay relative to 1 uM C3aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50322618((3S,6R,9S)-14-amino-2-((S)-1-((S)-2-((S)-1-((S)-6-...)
Affinity DataEC50:  130nMAssay Description:Antagonist activity at human C3a receptor in human U937 cells assessed as inhibition of intracellular calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50389006(CHEMBL2064020)
Affinity DataEC50:  148nMAssay Description:Agonist activity at human C3a receptor expressed in RBL-2H3 cells assessed as beta-hexosaminidase activity in cell supernatant by degranulation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50388998(CHEMBL2064012)
Affinity DataEC50:  170nMAssay Description:Agonist activity at human C3a receptor expressed in RBL-2H3 cells assessed as beta-hexosaminidase activity in cell supernatant by degranulation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50388996(CHEMBL2063898)
Affinity DataEC50:  195nMAssay Description:Agonist activity at human C3a receptor expressed in RBL-2H3 cells assessed as beta-hexosaminidase activity in cell supernatant by degranulation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50322620((S)-2-((R)-2-((S)-2-((S)-1-((S)-2-((S)-1-((S)-6-am...)
Affinity DataEC50:  220nMAssay Description:Agonist activity at human C3a receptor in human U937 cells assessed as induction of intracellular calcium releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50389003(CHEMBL2064018)
Affinity DataEC50:  224nMAssay Description:Agonist activity at human C3a receptor expressed in RBL-2H3 cells assessed as beta-hexosaminidase activity in cell supernatant by degranulation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50499182(CHEMBL3736020)
Affinity DataEC50:  240nMAssay Description:Agonist activity at C3aR in human MDM cells assessed as inhibition of C3a-induced Ca2+ response measured for 60 secs by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50499182(CHEMBL3736020)
Affinity DataEC50:  240nMAssay Description:Agonist activity at C3aR in human MDM cells assessed as inhibition of C3a-induced Ca2+ response measured for 60 secs by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50587345(CHEMBL5092449)
Affinity DataEC50:  282nMAssay Description:Agonist activity at human C3aR expressed in CHO cells assessed as induction of ERK1/2 phosphorylation at Thr202/Tyr204 residues incubated for 10 mins...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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