Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Polyamine deacetylase HDAC10 (Danio rerio) | BDBM50438391![]() (CHEMBL2413999) | PDB MMDB KEGG UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid PDB UniChem Similars | PDB PubMed | n/a | n/a | 120 | n/a | n/a | n/a | n/a | n/a | n/a |
University of East Anglia Curated by ChEMBL | Assay Description Inhibition of zebrafish HDAC10 (2 to 675 residues) expressed in Escherichia coli BL21(DE3) cells using N-acetylputrescine as substrate preincubated f... | J Med Chem 63: 12460-12484 (2020) | |||||||||||
More data for this Ligand-Target Pair | ![]() 3D Structure (crystal) |