Compile Data Set for Download or QSAR
maximum 50k data
Found 91 of ic50 for UniProtKB: P06766
TargetDNA polymerase beta(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50250427((+)-Myristinin D | CHEMBL448072)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of rat recombinant DNA polymerase beta in absence of bovine serum albuminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase beta(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50259787(3-trans-p-coumaroyl maslinic acid | CHEMBL453751)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of rat DNA polymerase beta in absence of BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase beta(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50259782(3beta-hydroxyrus-18,20(30)-dien-28-oic acid | CHEM...)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of rat DNA polymerase beta in absence of BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase beta(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50250426((+)-Myristinin A | CHEMBL465365)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibition of rat recombinant DNA polymerase beta in absence of bovine serum albuminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase beta(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50250305(3alpha-O-trans-p-coumaroyl-7-labden-15-oic acid | ...)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of rat DNA polymerase beta in absence of BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase beta(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50259781(3beta-hydroxyrus-12,19(29)-dien-28-oic acid | CHEM...)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibition of rat DNA polymerase beta in absence of BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase beta(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50079577((4aS,6aS,6bR,10S,12aR,14bS)-10-Hydroxy-2,2,6a,6b,9...)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibition of rat DNA polymerase beta in absence of BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase beta(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50259787(3-trans-p-coumaroyl maslinic acid | CHEMBL453751)
Affinity DataIC50:  4.20E+3nMAssay Description:Inhibition of rat DNA polymerase beta in presence of 0.1 mg/mL BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase beta(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50250427((+)-Myristinin D | CHEMBL448072)
Affinity DataIC50:  4.30E+3nMAssay Description:Inhibition of rat recombinant DNA polymerase beta in presence of bovine serum albuminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase beta(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50250305(3alpha-O-trans-p-coumaroyl-7-labden-15-oic acid | ...)
Affinity DataIC50:  4.70E+3nMAssay Description:Inhibition of rat DNA polymerase beta in presence of BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase beta(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50148911((3beta)-3-hydroxyurs-12-en-28-oic acid | 3beta-hyd...)
Affinity DataIC50:  4.80E+3nMAssay Description:Inhibition of rat DNA polymerase beta in absence of BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase beta(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50259781(3beta-hydroxyrus-12,19(29)-dien-28-oic acid | CHEM...)
Affinity DataIC50:  5.30E+3nMAssay Description:Inhibition of rat DNA polymerase beta in presence of BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase beta(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50259782(3beta-hydroxyrus-18,20(30)-dien-28-oic acid | CHEM...)
Affinity DataIC50:  5.60E+3nMAssay Description:Inhibition of rat DNA polymerase beta in presence of BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase beta(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50203241(1, 3-dihydroxy-5-[14'-(3' ',5' '-dihydroxyphenyl)t...)
Affinity DataIC50:  5.80E+3nMAssay Description:Inhibition of rat DNA polymerase beta assessed as [3H]TTP incorporation after 60 mins by scintillation counting in presence of bovine serum albuminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase beta(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50241611(1, 3-dihydroxy-5-[14'-(3' ',5' '-dihydroxyphenyl)-...)
Affinity DataIC50:  6.50E+3nMAssay Description:Inhibition of rat DNA polymerase beta assessed as [3H]TTP incorporation after 60 mins by scintillation counting in presence of bovine serum albuminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase beta(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM23208((1R,2R,5S,8R,9R,10R,13R,14R,17S,19R)-17-hydroxy-1,...)
Affinity DataIC50:  6.50E+3nMAssay Description:Inhibition of rat DNA polymerase beta in absence of BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase beta(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50079577((4aS,6aS,6bR,10S,12aR,14bS)-10-Hydroxy-2,2,6a,6b,9...)
Affinity DataIC50:  7.50E+3nMAssay Description:Inhibition of rat DNA polymerase beta in presence of BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase beta(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50259786(3-cis-p-coumaroyl maslinic acid | CHEMBL463995)
Affinity DataIC50:  7.50E+3nMAssay Description:Inhibition of rat DNA polymerase beta in absence of BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase beta(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50241610(1,3-dihydroxy-5-[14'-(3' ',5' '-dihydroxyphenyl)-c...)
Affinity DataIC50:  7.50E+3nMAssay Description:Inhibition of rat DNA polymerase beta assessed as [3H]TTP incorporation after 60 mins by scintillation counting in presence of bovine serum albuminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase beta(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50356642(CHEMBL1917196)
Affinity DataIC50:  7.60E+3nMAssay Description:Inhibition of rat pol beta using poly(dA)/oligo(dT)18 (A/T = 2/1) and dTTP as the DNA template-primer and nucleotide substrate after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase beta(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50148911((3beta)-3-hydroxyurs-12-en-28-oic acid | 3beta-hyd...)
Affinity DataIC50:  8.50E+3nMAssay Description:Inhibition of rat DNA polymerase beta in presence of BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase beta(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50020659(CHEMBL3290498)
Affinity DataIC50:  9.50E+3nMAssay Description:Inhibition of rat recombinant DNA polymerase beta expressed in Escherichia coli JMpbeta5 cells assessed as incorporation of [3H]dTTP into poly(dA)/ol...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase beta(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50241570((24E)-3beta-hydroxy-7,24-euphadien-26-oic acid | C...)
Affinity DataIC50:  9.70E+3nMAssay Description:Inhibition of rat recombinant DNA polymerase beta after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase beta(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50153117((S)-4-((5R,10R,13R,17R)-3-Hydroxy-5,10,13-trimethy...)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibitory concentration against rat DNA polymerase beta incubated with 0.05 unitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase beta(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM33388(dehydroaltenusin derivative, 16)
Affinity DataIC50:  1.10E+4nMpH: 7.5 T: 2°CAssay Description:For the DNA polymerase reaction, the dehydroaltenusin derivative was dissolved in dimethyl sulfoxide (DMSO) at various concentrations and sonicated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase beta(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50109030(4-(3-Hydroxy-10,13-dimethyl-hexadecahydro-cyclopen...)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibitory effect of the compound on the activity of rat DNA polymerase beta was determined by inhibitory dose curvesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase beta(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50356643(CHEMBL1917198)
Affinity DataIC50:  1.15E+4nMAssay Description:Inhibition of rat pol beta using poly(dA)/oligo(dT)18 (A/T = 2/1) and dTTP as the DNA template-primer and nucleotide substrate after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase beta(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50375301(CHEMBL260980)
Affinity DataIC50:  1.19E+4nMAssay Description:Inhibition of rat DNA polymerase betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase beta(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50250426((+)-Myristinin A | CHEMBL465365)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of rat recombinant DNA polymerase beta in presence of bovine serum albuminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase beta(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM23208((1R,2R,5S,8R,9R,10R,13R,14R,17S,19R)-17-hydroxy-1,...)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibition of rat DNA polymerase beta in presence of 0.1 mg/mL BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase beta(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50259786(3-cis-p-coumaroyl maslinic acid | CHEMBL463995)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of rat DNA polymerase beta in presence of 0.1 mg/mL BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase beta(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50250362(3-Oximo-olean-12-en-29-oic acid | CHEMBL490347)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of rat DNA polymerase betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase beta(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50375300(TALAROFLAVONE)
Affinity DataIC50:  1.63E+4nMAssay Description:Inhibition of rat DNA polymerase betaMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA polymerase beta(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM23417(α-CA inhibitor, 4 | (-)-Epicatechin | (2R,3R)...)
Affinity DataIC50:  1.85E+4nMAssay Description:Inhibition of lyase activity of rat DNA polymerase beta after 30 mins by deoxyribose phosphate excision assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase beta(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50020663(CHEMBL3290502)
Affinity DataIC50:  1.95E+4nMAssay Description:Inhibition of rat recombinant DNA polymerase beta expressed in Escherichia coli JMpbeta5 cells assessed as incorporation of [3H]dTTP into poly(dA)/ol...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase beta(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50250352(3,4-seco-olean-4(23),12-diene-3,30-dioic acid | CH...)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of rat DNA polymerase betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase beta(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50250348(3-oxo-olean-12-en-29-oic acid | 3-oxoolean-12-en-2...)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of rat DNA polymerase betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase beta(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50237597(7-hydroxy-3,7'-dicoumaryl ether | 7-hydroxy-3-(2-o...)
Affinity DataIC50:  2.25E+4nMAssay Description:Inhibition of lyase activity of rat DNA polymerase beta after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase beta(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50241570((24E)-3beta-hydroxy-7,24-euphadien-26-oic acid | C...)
Affinity DataIC50:  2.30E+4nMAssay Description:Inhibition of rat recombinant DNA polymerase beta after 60 mins in presence of 0.1 mg/mL BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase beta(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM33387(dehydroaltenusin derivative, 15)
Affinity DataIC50:  2.40E+4nMpH: 7.5 T: 2°CAssay Description:For the DNA polymerase reaction, the dehydroaltenusin derivative was dissolved in dimethyl sulfoxide (DMSO) at various concentrations and sonicated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase beta(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50251277(CHEMBL458178 | Kasanosin A)
Affinity DataIC50:  2.73E+4nMAssay Description:Inhibition of rat DNA polymerase betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase beta(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50020676(CHEBI:41846 | CHEMBL566812)
Affinity DataIC50:  3.08E+4nMAssay Description:Inhibition of rat recombinant DNA polymerase beta expressed in Escherichia coli JMpbeta5 cells assessed as incorporation of [3H]dTTP into poly(dA)/ol...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase beta(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50109031(4-(10,13-Dimethyl-3-{3-[5-(2-oxo-hexahydro-thieno[...)
Affinity DataIC50:  3.10E+4nMAssay Description:Inhibitory effect of the compound on the activity of rat DNA polymerase beta was determined by inhibitory dose curvesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase beta(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50109029(4-{10,13-Dimethyl-3-[3-(6-{6-[5-(2-oxo-hexahydro-t...)
Affinity DataIC50:  3.20E+4nMAssay Description:Inhibitory effect of the compound on the activity of mammalian DNA polymerase beta was determined by inhibitory dose curvesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase beta(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM33386(dehydroaltenusin derivative, 14)
Affinity DataIC50:  3.50E+4nMpH: 7.5 T: 2°CAssay Description:For the DNA polymerase reaction, the dehydroaltenusin derivative was dissolved in dimethyl sulfoxide (DMSO) at various concentrations and sonicated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase beta(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50250360(3-benzyloximo-olean-12-en-29-oic acid | CHEMBL4557...)
Affinity DataIC50:  3.50E+4nMAssay Description:Inhibition of rat DNA polymerase betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase beta(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50448689(CHEMBL3127730)
Affinity DataIC50:  3.56E+4nMAssay Description:Inhibition of recombinant rat DNA polymerase beta expressed in Escherichia coli JMpbeta5 assessed as inhibition of incorporation of dTTP into poly(dA...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase beta(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50250361(3-methyloximo-olean-12-en-29-oic acid | CHEMBL5241...)
Affinity DataIC50:  3.60E+4nMAssay Description:Inhibition of rat DNA polymerase betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase beta(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50250349(3alpha-hydroxyolean-12-en-29-oic acid | CHEMBL4905...)
Affinity DataIC50:  3.60E+4nMAssay Description:Inhibition of rat DNA polymerase betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase beta(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50020661(CHEMBL3290500)
Affinity DataIC50:  3.79E+4nMAssay Description:Inhibition of rat recombinant DNA polymerase beta expressed in Escherichia coli JMpbeta5 cells assessed as incorporation of [3H]dTTP into poly(dA)/ol...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 91 total ) | Next | Last >>
Jump to: