Compile Data Set for Download or QSAR
maximum 50k data
Found 66 of ki data for polymerid = 50002434
TargetAdenosine receptor A2b(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50455533(CHEMBL4205635)
Affinity DataKi:  0.180nMAssay Description:Displacement of [3H]PSB-603 from recombinant rat adenosine A2B receptor expressed in CHO cell membranes after 75 mins by liquid scintillation countin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50086170((4-Cyano-phenyl)-carbamic acid 4-(2,6-dioxo-1,3-di...)
Affinity DataKi:  12.8nMAssay Description:Inhibition of [125I]-APOBX binding to rat Adenosine A2B receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50086170((4-Cyano-phenyl)-carbamic acid 4-(2,6-dioxo-1,3-di...)
Affinity DataKi:  12.8nMAssay Description:Binding affinity to rat adenosine A2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50086170((4-Cyano-phenyl)-carbamic acid 4-(2,6-dioxo-1,3-di...)
Affinity DataKi:  13nMAssay Description:Binding affinity to rat A2B adenosine receptor by radio-ligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM60917(9-chloranyl-5-(4-hydroxyphenyl)-2,3,4,5-tetrahydro...)
Affinity DataKi:  35nMAssay Description:Compound was tested for its binding affinity against Alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails
TargetAdenosine receptor A2b(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50213356(CHEMBL310997)
Affinity DataKi:  58nMAssay Description:Compound was tested for its binding affinity against Alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails
TargetAdenosine receptor A2b(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50550821(CHEMBL4763881)
Affinity DataKi: >100nMAssay Description:Displacement of [3H]PSB-603 from rat adenosine receptor A2B expressed in CHO cell membranes incubated for 75 mins by radioligand competition assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50550834(CHEMBL4784975)
Affinity DataKi: >100nMAssay Description:Displacement of [3H]PSB-603 from rat adenosine receptor A2B expressed in CHO cell membranes incubated for 75 mins by radioligand competition assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50550814(CHEMBL4747947)
Affinity DataKi: >100nMAssay Description:Displacement of [3H]PSB-603 from rat adenosine receptor A2B expressed in CHO cell membranes incubated for 75 mins by radioligand competition assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50550815(CHEMBL4752438)
Affinity DataKi: >100nMAssay Description:Displacement of [3H]PSB-603 from rat adenosine receptor A2B expressed in CHO cell membranes incubated for 75 mins by radioligand competition assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50550816(CHEMBL4758461)
Affinity DataKi: >100nMAssay Description:Displacement of [3H]PSB-603 from rat adenosine receptor A2B expressed in CHO cell membranes incubated for 75 mins by radioligand competition assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50550817(CHEMBL4745527)
Affinity DataKi: >100nMAssay Description:Displacement of [3H]PSB-603 from rat adenosine receptor A2B expressed in CHO cell membranes incubated for 75 mins by radioligand competition assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50550818(CHEMBL4797325)
Affinity DataKi: >100nMAssay Description:Displacement of [3H]PSB-603 from rat adenosine receptor A2B expressed in CHO cell membranes incubated for 75 mins by radioligand competition assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50550819(CHEMBL4796077)
Affinity DataKi: >100nMAssay Description:Displacement of [3H]PSB-603 from rat adenosine receptor A2B expressed in CHO cell membranes incubated for 75 mins by radioligand competition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50550820(CHEMBL4746936)
Affinity DataKi: >100nMAssay Description:Displacement of [3H]PSB-603 from rat adenosine receptor A2B expressed in CHO cell membranes incubated for 75 mins by radioligand competition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50550822(CHEMBL4757397)
Affinity DataKi: >100nMAssay Description:Displacement of [3H]PSB-603 from rat adenosine receptor A2B expressed in CHO cell membranes incubated for 75 mins by radioligand competition assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50550823(CHEMBL4780555)
Affinity DataKi: >100nMAssay Description:Displacement of [3H]PSB-603 from rat adenosine receptor A2B expressed in CHO cell membranes incubated for 75 mins by radioligand competition assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50550824(CHEMBL4797181)
Affinity DataKi: >100nMAssay Description:Displacement of [3H]PSB-603 from rat adenosine receptor A2B expressed in CHO cell membranes incubated for 75 mins by radioligand competition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50550825(CHEMBL4790122)
Affinity DataKi: >100nMAssay Description:Displacement of [3H]PSB-603 from rat adenosine receptor A2B expressed in CHO cell membranes incubated for 75 mins by radioligand competition assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50550826(CHEMBL4795542)
Affinity DataKi: >100nMAssay Description:Displacement of [3H]PSB-603 from rat adenosine receptor A2B expressed in CHO cell membranes incubated for 75 mins by radioligand competition assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50550827(CHEMBL4755914)
Affinity DataKi: >100nMAssay Description:Displacement of [3H]PSB-603 from rat adenosine receptor A2B expressed in CHO cell membranes incubated for 75 mins by radioligand competition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50550828(CHEMBL1242892)
Affinity DataKi: >100nMAssay Description:Displacement of [3H]PSB-603 from rat adenosine receptor A2B expressed in CHO cell membranes incubated for 75 mins by radioligand competition assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50550829(CHEMBL1242426)
Affinity DataKi: >100nMAssay Description:Displacement of [3H]PSB-603 from rat adenosine receptor A2B expressed in CHO cell membranes incubated for 75 mins by radioligand competition assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50550830(CHEMBL4787673)
Affinity DataKi: >100nMAssay Description:Displacement of [3H]PSB-603 from rat adenosine receptor A2B expressed in CHO cell membranes incubated for 75 mins by radioligand competition assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50550831(CHEMBL1242247)
Affinity DataKi: >100nMAssay Description:Displacement of [3H]PSB-603 from rat adenosine receptor A2B expressed in CHO cell membranes incubated for 75 mins by radioligand competition assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50550832(CHEMBL4764086)
Affinity DataKi: >100nMAssay Description:Displacement of [3H]PSB-603 from rat adenosine receptor A2B expressed in CHO cell membranes incubated for 75 mins by radioligand competition assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50550833(CHEMBL4779033)
Affinity DataKi: >100nMAssay Description:Displacement of [3H]PSB-603 from rat adenosine receptor A2B expressed in CHO cell membranes incubated for 75 mins by radioligand competition assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50397728(CHEMBL2181976)
Affinity DataKi:  163nMAssay Description:Displacement of [3H] DPCPX from rat adenosine A2B receptor expressed in HEK293 cells incubated for 60 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50020960(1-Allyl-3-methyl-8-phenyl-3,7-dihydro-purine-2,6-d...)
Affinity DataKi:  174nMAssay Description:Inhibition of [125I]-APOBX binding to rat Adenosine A2B receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50058225(CHEMBL45244 | N-((4-(2-cyanophenyl)piperazin-1-yl)...)
Affinity DataKi:  177nMAssay Description:Binding affinity of the compound at Alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM21173(1,3-dipropyl-8-cyclopentylxanthine | 8-cyclopentyl...)
Affinity DataKi:  186nMAssay Description:Inhibition of [125I]-APOBX binding to rat Adenosine A2B receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50213353(CHEMBL308295)
Affinity DataKi:  302nMAssay Description:Compound was tested for its binding affinity against Alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails
TargetAdenosine receptor A2b(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50213354(CHEMBL80974)
Affinity DataKi:  933nMAssay Description:Compound was tested for its binding affinity against Alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails
TargetAdenosine receptor A2b(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM55121(3-HYDROXYTYRAMINE HYDROCHLORIDE | 4-(2-aminoethyl)...)
Affinity DataKi:  977nMAssay Description:Compound was tested for its binding affinity against Alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails
TargetAdenosine receptor A2b(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50187588(CHEMBL3827201)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]PSB-603 from recombinant rat adenosine receptor A2b expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50187585(CHEMBL3827074)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]PSB-603 from recombinant rat adenosine receptor A2b expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50187584(CHEMBL3827187)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]PSB-603 from recombinant rat adenosine receptor A2b expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50187587(CHEMBL3827598)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]PSB-603 from recombinant rat adenosine receptor A2b expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50187589(CHEMBL3827859)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]PSB-603 from recombinant rat adenosine receptor A2b expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50187586(CHEMBL3827623)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]PSB-603 from recombinant rat adenosine receptor A2b expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50014154(2-(5-Methyl-1H-imidazol-4-ylmethyl)-4-phenyl-thiaz...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity for Alpha-2 adrenergic receptor was determined by using [3H]p-aminoclonidine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50048466(2-(furan-2-yl)-7-phenethyl-7H-pyrazolo[4,3-e][1,2,...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-CGS- 21680 from rat striatal membrane adenosine A2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50187590(CHEMBL3827583)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]PSB-603 from recombinant rat adenosine receptor A2b expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50070518((R)-3-{2-[4-(3,4-Dimethyl-phenyl)-piperazin-1-yl]-...)
Affinity DataKi:  1.02E+3nMAssay Description:In vivo binding affinity was evaluated against Alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50187591(CHEMBL3827331)
Affinity DataKi:  1.10E+3nMAssay Description:Displacement of [3H]PSB-603 from recombinant rat adenosine receptor A2b expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50213355(CHEMBL80686)
Affinity DataKi:  1.45E+3nMAssay Description:Compound was tested for its binding affinity against Alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails
TargetAdenosine receptor A2b(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50113237(1-Allyl-7-(2-chloro-ethyl)-3-methyl-8-phenyl-3,7-d...)
Affinity DataKi:  1.70E+3nMAssay Description:Inhibition of [125I]-APOBX binding to rat Adenosine A2B receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50070514((S)-3-{2-[4-(3,4-Dimethyl-phenyl)-piperazin-1-yl]-...)
Affinity DataKi:  1.71E+3nMAssay Description:In vivo binding affinity was evaluated against Alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50001490(1-Propyl-3,7-dihydro-purine-2,6-dione | CHEMBL3998...)
Affinity DataKi:  1.88E+3nMAssay Description:Inhibition of [125I]-APOBX binding to rat Adenosine A2B receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50042208(3-Methyl-1-prop-2-ynyl-3,7-dihydro-purine-2,6-dion...)
Affinity DataKi:  2.15E+3nMAssay Description:Inhibition of [125I]-APOBX binding to rat Adenosine A2B receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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