Compile Data Set for Download or QSAR
maximum 50k data
Found 306 of ki for UniProtKB: P50130
TargetD(1A) dopamine receptor(Sus scrofa)
Purdue University

Curated by ChEMBL
LigandPNGBDBM82247(8-Chloro-3-methyl-5-phenyl-2,3,4,5-tetrahydro-1H-b...)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]SCH-23390 from dopamine D1-like receptor in porcine striata homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50033116((1R,3S)-3-Adamantan-1-yl-1-aminomethyl-isochroman-...)
Affinity DataKi:  3.90nMAssay Description:Displacement of [3H]SCH-23390 from porcine striatum dopamine D1 receptor incubated for 30 mins by radioligand competition binding assay based scintil...More data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(Sus scrofa)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50200353((6aR,12bS)-(+)-2,3-dihydroxy-6a,7,8,12b-tetrahydro...)
Affinity DataKi:  8nMAssay Description:Displacement of [3H]SCH-23390 from dopamine D1-like receptor in porcine striata homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Purdue University

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  9.5nMAssay Description:Displacement of [3H]SCH23390 from porcine striatal membranes D1 receptor by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50328444(4-[4-(2,5-Dimethylphenyl)-4-hydroxypiperidin-1-yl]...)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor in pig striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50010686((6aR,12bS)-10,11-Dihydroxy-5,6,6a,7,8,12b-hexahydr...)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]SCH-23390 from dopamine D1-like receptor in porcine striata homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50200351((+/-)-2,3-dihydroxy-6a,7,8,12b-tetrahydro-6H-chrom...)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]SCH-23390 from dopamine D1-like receptor in porcine striata homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50053414(CHEMBL3318849)
Affinity DataKi:  49nMAssay Description:Displacement of [3H]SCH23390 from porcine striatal membranes D1 receptor by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50053390(CHEMBL3318845)
Affinity DataKi:  59nMAssay Description:Displacement of [3H]SCH23390 from porcine striatal membranes D1 receptor by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50053391(CHEMBL3318824)
Affinity DataKi:  72nMAssay Description:Displacement of [3H]SCH23390 from porcine striatal membranes D1 receptor by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50053415(CHEMBL3318850)
Affinity DataKi:  86nMAssay Description:Displacement of [3H]SCH23390 from porcine striatal membranes D1 receptor by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Purdue University

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  93nMAssay Description:Displacement of [3H]SCH 23390 from pig dopamine D1 receptor in striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Purdue University

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  93nMAssay Description:Displacement of [3H]SCH23390 from D1 receptor from porcine cerebral cortex homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Purdue University

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  98nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor in pig striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50328443(1-(4-Fluorophenyl)-4-[4-([2.2]paracyclophan-4-yl)-...)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor in pig striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50053416(CHEMBL3317465)
Affinity DataKi:  120nMAssay Description:Displacement of [3H]SCH23390 from porcine striatal membranes D1 receptor by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50053376(CHEMBL3318831)
Affinity DataKi:  130nMAssay Description:Displacement of [3H]SCH23390 from porcine striatal membranes D1 receptor by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50298914(CHEMBL572867 | N-(4-(4-(2,3-dichlorophenyl)piperaz...)
Affinity DataKi:  140nMAssay Description:Binding affinity to pig dopamine D1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50053408(Haldol | Haldol Dec | Haloperidol Decanoate | R-13...)
Affinity DataKi:  140nMAssay Description:Displacement of [3H]SCH23390 from porcine striatal membranes D1 receptor by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50053417(CHEMBL3318851)
Affinity DataKi:  150nMAssay Description:Displacement of [3H]SCH23390 from porcine striatal membranes D1 receptor by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50298913(CHEMBL572379 | N-(4-(4-(2,3-dichlorophenyl)piperaz...)
Affinity DataKi:  180nMAssay Description:Binding affinity to pig dopamine D1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50436541(CHEMBL2396663)
Affinity DataKi:  190nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor in porcine striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50053413(CHEMBL3318848)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]SCH23390 from porcine striatal membranes D1 receptor by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50357936(CHEMBL1916720)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]SCH 23390 from pig dopamine D1 receptor in striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50359763(CHEMBL1928122)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]SCH23390 from pig D1 receptor in straital membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50347629(CHEMBL1803023)
Affinity DataKi:  210nMAssay Description:Displacement of [3H]SCH23390 from D1 receptor from porcine cerebral cortex homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50328450(4-[4-(2,5-Dimethylphenyl)piperazin-1-yl]-1-(4-fluo...)
Affinity DataKi:  210nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor in pig striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50347630(CHEMBL1803024)
Affinity DataKi:  220nMAssay Description:Displacement of [3H]SCH 23390 from pig dopamine D1 receptor in striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50342714(3,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-y...)
Affinity DataKi:  220nMAssay Description:Displacement of [3H]SCH-23390 from dopamine D1 receptor in pig striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50053378(CHEMBL3318833)
Affinity DataKi:  220nMAssay Description:Displacement of [3H]SCH23390 from porcine striatal membranes D1 receptor by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50053377(CHEMBL3318832)
Affinity DataKi:  220nMAssay Description:Displacement of [3H]SCH23390 from porcine striatal membranes D1 receptor by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50347630(CHEMBL1803024)
Affinity DataKi:  220nMAssay Description:Displacement of [3H]SCH23390 from D1 receptor from porcine cerebral cortex homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50347634(CHEMBL1803028)
Affinity DataKi:  220nMAssay Description:Displacement of [3H]SCH23390 from D1 receptor from porcine cerebral cortex homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50347631(CHEMBL1803025)
Affinity DataKi:  250nMAssay Description:Displacement of [3H]SCH23390 from D1 receptor from porcine cerebral cortex homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50359762(CHEMBL1928121)
Affinity DataKi:  250nMAssay Description:Displacement of [3H]SCH23390 from pig D1 receptor in straital membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50053411(CHEMBL3318847)
Affinity DataKi:  260nMAssay Description:Displacement of [3H]SCH23390 from porcine striatal membranes D1 receptor by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50331549(CHEMBL567286 | [11C]-3-(2-oxo-3-(2-(4-(trifluorome...)
Affinity DataKi:  270nMAssay Description:Displacement of [3H]SCH 23990 from dopamine D1 receptor in porcine cerebral cortex membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50200352((6aS,12bR)-(-)-2,3-dihydroxy-6a,7,8,12b-tetrahydro...)
Affinity DataKi:  270nMAssay Description:Displacement of [3H]SCH-23390 from dopamine D1-like receptor in porcine striata homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50347635(CHEMBL1803029)
Affinity DataKi:  270nMAssay Description:Displacement of [3H]SCH23390 from D1 receptor from porcine cerebral cortex homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50053379(CHEMBL3318834)
Affinity DataKi:  280nMAssay Description:Displacement of [3H]SCH23390 from porcine striatal membranes D1 receptor by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50436542(CHEMBL2397389)
Affinity DataKi:  300nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor in porcine striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50347632(CHEMBL1803026)
Affinity DataKi:  300nMAssay Description:Displacement of [3H]SCH23390 from D1 receptor from porcine cerebral cortex homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50357935(CHEMBL1916548)
Affinity DataKi:  330nMAssay Description:Displacement of [3H]SCH 23390 from pig dopamine D1 receptor in striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50167933(CHEMBL370297 | N-{4-[4-(2,3-dichlorophenyl)piperaz...)
Affinity DataKi:  330nMAssay Description:Inhibition of [3H]-SCH- 23390 binding to dopamine receptor D1 of porcine striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50370760(CHEMBL1203924)
Affinity DataKi:  330nMAssay Description:Displacement of [3H]SCH-23390 from dopamine D1-like receptor in porcine striata homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50155520(4-[4-(4-Chloro-phenyl)-piperazin-1-yl]-1-(4-fluoro...)
Affinity DataKi:  340nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor in pig striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50053409(CHEMBL3318846)
Affinity DataKi:  360nMAssay Description:Displacement of [3H]SCH23390 from porcine striatal membranes D1 receptor by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50342706(3,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-y...)
Affinity DataKi:  380nMAssay Description:Displacement of [3H]SCH-23390 from dopamine D1 receptor in pig striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50347633(CHEMBL1803027)
Affinity DataKi:  390nMAssay Description:Displacement of [3H]SCH23390 from D1 receptor from porcine cerebral cortex homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50347626(CHEMBL1803053)
Affinity DataKi:  400nMAssay Description:Displacement of [3H]SCH23390 from D1 receptor from porcine cerebral cortex homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 306 total ) | Next | Last >>
Jump to: