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Found 271 of ic50 for UniProtKB: P06935
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50513893(CHEMBL506092)
Affinity DataIC50:  56nMAssay Description:Inhibition of West Nile virus proteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM35491(Benzoic acid 5-amino-1-(4-methoxy-benzenesulfonyl)...)
Affinity DataIC50:  105nMAssay Description:Inhibition of WNV NS2B-NS3 protease by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM35491(Benzoic acid 5-amino-1-(4-methoxy-benzenesulfonyl)...)
Affinity DataIC50:  105nMAssay Description:The HTS assay to identify Inhibitors of West Nile Virus (WNV) NS2bNS3 Proteinase was proposed by Dr Alex Strongin of the Burnham Institute XO1-MH0776...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM35509(2-thiophenecarboxylic acid [5-amino-1-(4-methoxyph...)
Affinity DataIC50:  110nMAssay Description:Inhibition of WNV NS2B-NS3 protease by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM35509(2-thiophenecarboxylic acid [5-amino-1-(4-methoxyph...)
Affinity DataIC50:  110nMAssay Description:The HTS assay to identify Inhibitors of West Nile Virus (WNV) NS2bNS3 Proteinase was proposed by Dr Alex Strongin of the Burnham Institute XO1-MH0776...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50567466(CHEMBL4862682)
Affinity DataIC50:  120nMAssay Description:Inhibition West Nile virus NS3B/NS3 protease using 7-amino-4-methylcoumarin as substrate by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM39394(2-bromobenzoic acid [5-amino-1-(4-methoxyphenyl)su...)
Affinity DataIC50:  297nMAssay Description:The HTS assay to identify Inhibitors of West Nile Virus (WNV) NS2bNS3 Proteinase was proposed by Dr Alex Strongin of the Burnham Institute XO1-MH0776...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50302021(5-amino-1-(4-methoxyphenylsulfonyl)-1H-pyrazol-3-y...)
Affinity DataIC50:  310nMAssay Description:Inhibition of WNV NS2B-NS3 protease by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50030457(CHEMBL3344314)
Affinity DataIC50:  380nMAssay Description:Inhibition of West Nile virus NS2B-NS3 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50030458(CHEMBL3344313)
Affinity DataIC50:  420nMAssay Description:Inhibition of West Nile virus NS2B-NS3 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50587014(CHEMBL5094815)
Affinity DataIC50:  460nMAssay Description:Inhibition of C-terminal His-tagged WNV NSB2 (52 to 96 amino acids)-NS3 (1 to 184 amino acids) protease expressed in Escherichia coli BL21(DE3) using...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50567470(CHEMBL4862353)
Affinity DataIC50:  510nMAssay Description:Inhibition West Nile virus NS3B/NS3 protease using 7-amino-4-methylcoumarin as substrate by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM32761(2-furancarboxylic acid [5-amino-1-(4-methoxyphenyl...)
Affinity DataIC50:  553nMAssay Description:The HTS assay to identify Inhibitors of West Nile Virus (WNV) NS2bNS3 Proteinase was proposed by Dr Alex Strongin of the Burnham Institute XO1-MH0776...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50109138(CHEMBL3601351)
Affinity DataIC50:  750nMAssay Description:Inhibition of WNV NS2B-NS3 protease expressed in Escherichia coli BL21 lambda (DE3) cells using Abz-Gly-Leu-Lys-Arg-Gly-Gly-3-(NO2)Tyr as substrate p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50567467(CHEMBL4850391)
Affinity DataIC50:  780nMAssay Description:Inhibition West Nile virus NS3B/NS3 protease using 7-amino-4-methylcoumarin as substrate by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50522790(CHEMBL3741422)
Affinity DataIC50:  800nMAssay Description:Inhibition of West Nile virus NS2B-NS3 protease preincubated with protein for 15 mins followed by Abz-Gly-Leu-Lys-Arg-Gly-Gly-3-(NO2)-Tyr substrate a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50567473(CHEMBL4872757)
Affinity DataIC50:  820nMAssay Description:Inhibition West Nile virus NS3B/NS3 protease using 7-amino-4-methylcoumarin as substrate by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50567469(CHEMBL4856850)
Affinity DataIC50:  870nMAssay Description:Inhibition West Nile virus NS3B/NS3 protease using 7-amino-4-methylcoumarin as substrate by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50567468(CHEMBL4853830)
Affinity DataIC50:  930nMAssay Description:Inhibition West Nile virus NS3B/NS3 protease using 7-amino-4-methylcoumarin as substrate by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50302022(5-amino-1-(4-methoxyphenylsulfonyl)-1H-pyrazol-3-y...)
Affinity DataIC50:  970nMAssay Description:Inhibition of WNV NS2B-NS3 protease by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50109050(CHEMBL3601349)
Affinity DataIC50:  1.01E+3nMAssay Description:Inhibition of WNV NS2B-NS3 protease expressed in Escherichia coli BL21 lambda (DE3) cells using Abz-Gly-Leu-Lys-Arg-Gly-Gly-3-(NO2)Tyr as substrate p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50109046(CHEMBL3601345)
Affinity DataIC50:  1.12E+3nMAssay Description:Inhibition of WNV NS2B-NS3 protease expressed in Escherichia coli BL21 lambda (DE3) cells using Abz-Gly-Leu-Lys-Arg-Gly-Gly-3-(NO2)Tyr as substrate p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50109139(CHEMBL3601352)
Affinity DataIC50:  1.13E+3nMAssay Description:Inhibition of WNV NS2B-NS3 protease expressed in Escherichia coli BL21 lambda (DE3) cells using Abz-Gly-Leu-Lys-Arg-Gly-Gly-3-(NO2)Tyr as substrate p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM32783(2-thiophenecarboxylic acid [5-amino-1-(4-fluorophe...)
Affinity DataIC50:  1.16E+3nMAssay Description:The HTS assay to identify Inhibitors of West Nile Virus (WNV) NS2bNS3 Proteinase was proposed by Dr Alex Strongin of the Burnham Institute XO1-MH0776...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50542823(CHEMBL4633312)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of West Nile virus NS2B-NS3 protease expressed in Escherichia coli BL21 lambda (DE3) cells using Abz-Gly-Leu-Lys-Arg-Gly-Gly-3-(NO2)Tyr as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50302023(5-amino-1-(4-methoxyphenylsulfonyl)-1H-pyrazol-3-y...)
Affinity DataIC50:  1.22E+3nMAssay Description:Inhibition of WNV NS2B-NS3 protease by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM39396(2-bromobenzoic acid (5-amino-1-besyl-pyrazol-3-yl)...)
Affinity DataIC50:  1.26E+3nMAssay Description:The HTS assay to identify Inhibitors of West Nile Virus (WNV) NS2bNS3 Proteinase was proposed by Dr Alex Strongin of the Burnham Institute XO1-MH0776...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50109142(CHEMBL3601354)
Affinity DataIC50:  1.27E+3nMAssay Description:Inhibition of WNV NS2B-NS3 protease expressed in Escherichia coli BL21 lambda (DE3) cells using Abz-Gly-Leu-Lys-Arg-Gly-Gly-3-(NO2)Tyr as substrate p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50567471(CHEMBL4876865)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition West Nile virus NS3B/NS3 protease using 7-amino-4-methylcoumarin as substrate by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50567472(CHEMBL4848934)
Affinity DataIC50:  1.34E+3nMAssay Description:Inhibition West Nile virus NS3B/NS3 protease using 7-amino-4-methylcoumarin as substrate by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50109047(CHEMBL3601346)
Affinity DataIC50:  1.35E+3nMAssay Description:Inhibition of WNV NS2B-NS3 protease expressed in Escherichia coli BL21 lambda (DE3) cells using Abz-Gly-Leu-Lys-Arg-Gly-Gly-3-(NO2)Tyr as substrate p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM32778(MLS000081703 | SMR000062919 | [2-(2-cyanoethyl)-5-...)
Affinity DataIC50:  1.35E+3nMAssay Description:Inhibition of WNV NS2B-NS3 protease by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM32778(MLS000081703 | SMR000062919 | [2-(2-cyanoethyl)-5-...)
Affinity DataIC50:  1.35E+3nMAssay Description:The HTS assay to identify Inhibitors of West Nile Virus (WNV) NS2bNS3 Proteinase was proposed by Dr Alex Strongin of the Burnham Institute XO1-MH0776...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PCBioAssay
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50109049(CHEMBL3601348)
Affinity DataIC50:  1.39E+3nMAssay Description:Inhibition of WNV NS2B-NS3 protease expressed in Escherichia coli BL21 lambda (DE3) cells using Abz-Gly-Leu-Lys-Arg-Gly-Gly-3-(NO2)Tyr as substrate p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50127623(CHEMBL3628260)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of West Nile virus NS2B-NS3 protease preincubated with protein for 15 mins followed by Abz-Gly-Leu-Lys-Arg-Gly-Gly-3-(NO2)-Tyr substrate a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM32756(2-furancarboxylic acid [5-amino-1-(4-fluorophenyl)...)
Affinity DataIC50:  1.65E+3nMAssay Description:The HTS assay to identify Inhibitors of West Nile Virus (WNV) NS2bNS3 Proteinase was proposed by Dr Alex Strongin of the Burnham Institute XO1-MH0776...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50109048(CHEMBL3601347)
Affinity DataIC50:  1.69E+3nMAssay Description:Inhibition of WNV NS2B-NS3 protease expressed in Escherichia coli BL21 lambda (DE3) cells using Abz-Gly-Leu-Lys-Arg-Gly-Gly-3-(NO2)Tyr as substrate p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50109112(CHEMBL3601350)
Affinity DataIC50:  1.71E+3nMAssay Description:Inhibition of WNV NS2B-NS3 protease expressed in Escherichia coli BL21 lambda (DE3) cells using Abz-Gly-Leu-Lys-Arg-Gly-Gly-3-(NO2)Tyr as substrate p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50109265(CHEMBL3601102)
Affinity DataIC50:  1.76E+3nMAssay Description:Inhibition of WNV NS2B-NS3 protease expressed in Escherichia coli BL21 lambda (DE3) cells using Abz-Gly-Leu-Lys-Arg-Gly-Gly-3-(NO2)Tyr as substrate p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50567458(CHEMBL4869904)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition West Nile virus NS3B/NS3 protease using 7-amino-4-methylcoumarin as substrate by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50542820(CHEMBL4640021)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of West Nile virus NS2B-NS3 protease expressed in Escherichia coli BL21 lambda (DE3) cells using Abz-Gly-Leu-Lys-Arg-Gly-Gly-3-(NO2)Tyr as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50302024(5-amino-1-(4-methoxyphenylsulfonyl)-1H-pyrazol-3-y...)
Affinity DataIC50:  1.83E+3nMAssay Description:Inhibition of WNV NS2B-NS3 protease by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50542238(CHEMBL4640778)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of West Nile virus NS2B-NS3 proteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50109267(CHEMBL3601104)
Affinity DataIC50:  1.91E+3nMAssay Description:Inhibition of WNV NS2B-NS3 protease expressed in Escherichia coli BL21 lambda (DE3) cells using Abz-Gly-Leu-Lys-Arg-Gly-Gly-3-(NO2)Tyr as substrate p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50302025(5-amino-1-(4-methoxyphenylsulfonyl)-1H-pyrazol-3-y...)
Affinity DataIC50:  1.96E+3nMAssay Description:Inhibition of WNV NS2B-NS3 protease by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50030455(CHEMBL3344316)
Affinity DataIC50:  2.01E+3nMAssay Description:Inhibition of West Nile virus NS2B-NS3 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50109266(CHEMBL3601103)
Affinity DataIC50:  2.03E+3nMAssay Description:Inhibition of WNV NS2B-NS3 protease expressed in Escherichia coli BL21 lambda (DE3) cells using Abz-Gly-Leu-Lys-Arg-Gly-Gly-3-(NO2)Tyr as substrate p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50109141(CHEMBL3601353)
Affinity DataIC50:  2.11E+3nMAssay Description:Inhibition of WNV NS2B-NS3 protease expressed in Escherichia coli BL21 lambda (DE3) cells using Abz-Gly-Leu-Lys-Arg-Gly-Gly-3-(NO2)Tyr as substrate p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50109144(CHEMBL3601356)
Affinity DataIC50:  2.12E+3nMAssay Description:Inhibition of WNV NS2B-NS3 protease expressed in Escherichia coli BL21 lambda (DE3) cells using Abz-Gly-Leu-Lys-Arg-Gly-Gly-3-(NO2)Tyr as substrate p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50030456(CHEMBL3344319)
Affinity DataIC50:  2.20E+3nMAssay Description:Non-competitive inhibition of West Nile virus NS2B-NS3 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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