Compile Data Set for Download or QSAR
maximum 50k data
Found 174 of kd for UniProtKB: A0A024RAY5
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM289495(1-(4-(6-amino-5-(tri- fluoromethyl)pyridin-3- yl)-...)
Affinity DataKd:  0.110nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM590003((S)-1-(4-(6-amino-5- (trifluoromethyl)pyridin-3-yl...)
Affinity DataKd:  0.120nMAssay Description:A fusion protein of full length of human DLK (amino acids 1-859) and the DNA binding domain of NFkB was expressed in transiently transfected HEK293 c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM589995((R)-1-(4-(6-amino-5-(trifluoromethyl)pyridin-3-yl)...)
Affinity DataKd:  0.210nMAssay Description:A fusion protein of full length of human DLK (amino acids 1-859) and the DNA binding domain of NFkB was expressed in transiently transfected HEK293 c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM589991(US11560366, Example 3b)
Affinity DataKd:  0.240nMAssay Description:A fusion protein of full length of human DLK (amino acids 1-859) and the DNA binding domain of NFkB was expressed in transiently transfected HEK293 c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM289483(1-(4-(6-amino-5- (trifluoromethyl)- pyridin-3-yl)-...)
Affinity DataKd:  0.290nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM590004((S)-1-(4-(6-amino-5- (trifluoromethoxy)pyridin-3-y...)
Affinity DataKd:  0.290nMAssay Description:A fusion protein of full length of human DLK (amino acids 1-859) and the DNA binding domain of NFkB was expressed in transiently transfected HEK293 c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM589992((S)-1-(4-(6-amino-5-(trifluoromethyl)pyridin-3-yl)...)
Affinity DataKd:  0.290nMAssay Description:A fusion protein of full length of human DLK (amino acids 1-859) and the DNA binding domain of NFkB was expressed in transiently transfected HEK293 c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM289483(1-(4-(6-amino-5- (trifluoromethyl)- pyridin-3-yl)-...)
Affinity DataKd:  0.300nMAssay Description:A fusion protein of full length of human DLK (amino acids 1-859) and the DNA binding domain of NFkB was expressed in transiently transfected HEK293 c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM289429((S)-1-(4-(6-amino-5-(trifluoromethoxy)pyridin-3-yl...)
Affinity DataKd:  0.310nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM289505(1-(4-(6-amino-5-(tri- fluoromethyl)pyridin-3- yl)-...)
Affinity DataKd:  0.360nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM289428((S)-1-(4-(6-amino-5-(trifluoromethoxy)pyridin-3-yl...)
Affinity DataKd:  0.360nMAssay Description:A fusion protein of full length of human DLK (amino acids 1-859) and the DNA binding domain of NFkB was expressed in transiently transfected HEK293 c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM289428((S)-1-(4-(6-amino-5-(trifluoromethoxy)pyridin-3-yl...)
Affinity DataKd:  0.360nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM589996((R)-1-(4-(6-amino-5-(trifluoromethoxy)pyridin-3-yl...)
Affinity DataKd:  0.5nMAssay Description:A fusion protein of full length of human DLK (amino acids 1-859) and the DNA binding domain of NFkB was expressed in transiently transfected HEK293 c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM289481(1-(4-(6-amino-5-(tri- fluoromethoxy)pyridin- 3-yl)...)
Affinity DataKd:  0.620nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM589998(US11560366, Example 10a)
Affinity DataKd:  0.620nMAssay Description:A fusion protein of full length of human DLK (amino acids 1-859) and the DNA binding domain of NFkB was expressed in transiently transfected HEK293 c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM289426( (R)-1-(4-(6-amino-5-(trifluoromethyl)pyridin-3-yl...)
Affinity DataKd:  0.740nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM589997(US11560366, Example 9b)
Affinity DataKd:  1nMAssay Description:A fusion protein of full length of human DLK (amino acids 1-859) and the DNA binding domain of NFkB was expressed in transiently transfected HEK293 c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM289481(1-(4-(6-amino-5-(tri- fluoromethoxy)pyridin- 3-yl)...)
Affinity DataKd:  1.10nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM590001((R)-1-(4-(6-amino-5-(trifluoromethoxy)- pyridin-3-...)
Affinity DataKd:  1.60nMAssay Description:A fusion protein of full length of human DLK (amino acids 1-859) and the DNA binding domain of NFkB was expressed in transiently transfected HEK293 c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM289491(1-(4-(6-amino-5- (trifluoromethoxy)- pyridin-3-yl)...)
Affinity DataKd:  1.60nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM289437(4-(3-(2-cyclopropyl-4-(3-(trifluoromethyl)-1H-pyrr...)
Affinity DataKd:  1.90nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM289489(1-(4-(6-amino-5-(tri- fluoromethyl)pyridin-3- yl)-...)
Affinity DataKd:  2.10nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM589988((R)-1-(4-(6-amino-5-(trifluoromethoxy)pyridin-3-yl...)
Affinity DataKd:  2.20nMAssay Description:A fusion protein of full length of human DLK (amino acids 1-859) and the DNA binding domain of NFkB was expressed in transiently transfected HEK293 c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM289425((R)-(4-(6-amino-5-(trifluoromethyl)pyridin-3-yl)-1...)
Affinity DataKd:  2.30nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM289484((4-(6-amino-5-(trifluoro- methyl)pyridin-3- yl)-1-...)
Affinity DataKd:  2.40nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM590000((4-(6-amino-5-(trifluoromethyl)pyridin-3-yl)-1-(3-...)
Affinity DataKd:  2.90nMAssay Description:A fusion protein of full length of human DLK (amino acids 1-859) and the DNA binding domain of NFkB was expressed in transiently transfected HEK293 c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM289447(4-(3-(2-isopropyl-4-(1-(1-(pyridin-2-yl)ethyl)-1H-...)
Affinity DataKd:  2.90nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM589999((4-(6-amino-5-(trifluoromethoxy)pyridin-3-yl)-1-(3...)
Affinity DataKd:  3.10nMAssay Description:A fusion protein of full length of human DLK (amino acids 1-859) and the DNA binding domain of NFkB was expressed in transiently transfected HEK293 c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM289466(5-(2-(cyclopropyl- methyl)-1-(3-(4- methylpiperazi...)
Affinity DataKd:  3.10nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM589990((R)-1-(4-(6-amino-5-(trifluoromethyl)pyridin-3-yl)...)
Affinity DataKd:  4.40nMAssay Description:A fusion protein of full length of human DLK (amino acids 1-859) and the DNA binding domain of NFkB was expressed in transiently transfected HEK293 c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM289509(5-(2-isopropyl-1-(3-(4- methylpiperazin-1-yl)- bic...)
Affinity DataKd:  4.5nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM289480((4-(6-amino-5-(tri- fluoromethoxy)pyridin- 3-yl)-1...)
Affinity DataKd:  5.10nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM50271212(CHEMBL3715238)
Affinity DataKd:  5.10nMAssay Description:Binding affinity to full length wild type human DLK (M1 to P859 residues) expressed in mammalian cells by KINOMEscan assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM589993(US11560366, Example 5)
Affinity DataKd:  5.20nMAssay Description:A fusion protein of full length of human DLK (amino acids 1-859) and the DNA binding domain of NFkB was expressed in transiently transfected HEK293 c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM289471(5-(2-isobutyl-1-(3- morpholinobicyclo- [1.1.1]pent...)
Affinity DataKd:  6nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM289444(5-(1-(3-(bis(2-methoxyethyl)amino)bicyclo[1.1.1]pe...)
Affinity DataKd:  6.40nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM289455(5-(1-(3-morpholino- bicyclo[1.1.1]pentan-1- yl)-2-...)
Affinity DataKd:  6.70nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM289443(5-(2-cyclopropyl-1-(3-((2-methoxyethyl)(methyl)ami...)
Affinity DataKd:  6.80nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM289436(5-(2-cyclopropyl-1-(3-(4-(2-fluoroethyl)piperazin-...)
Affinity DataKd:  6.90nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM289445(1-(3-(4-(6-amino-5-(trifluoromethoxy)pyridin-3-yl)...)
Affinity DataKd:  7nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM289458(5-(2-(cyclopropyl- methyl)-1-(3-morpho- linobicycl...)
Affinity DataKd:  7.20nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM289511(5-(2-cyclopropyl-1-(3- (4-methylpiperazin-1- yl)bi...)
Affinity DataKd:  7.40nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM289510(5-(2-cyclopropyl-1-(3- (4-methylpiperazin-1- yl)bi...)
Affinity DataKd:  7.5nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM589994(US11560366, Example 6)
Affinity DataKd:  7.70nMAssay Description:A fusion protein of full length of human DLK (amino acids 1-859) and the DNA binding domain of NFkB was expressed in transiently transfected HEK293 c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM289424(US10093664, Example 4)
Affinity DataKd:  8.30nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM289473(5-(2-(sec-butyl)-1-(3- morpholinobicyclo- [1.1.1]p...)
Affinity DataKd:  8.60nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM289474(5-(2-(sec-butyl)-1-(3- morpholinobicyclo- [1.1.1]p...)
Affinity DataKd:  9.5nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM289441(4-(3-(4-(6-amino-5-(trifluoromethoxy)pyridin-3-yl)...)
Affinity DataKd:  9.70nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM289456((S)-1-(4-(6-amino-5- (trifluoromethyl)- pyridin-3-...)
Affinity DataKd:  9.70nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM289423(5-(2-isopropyl-1-(3-morpholinobicyclo[1.1.1]pentan...)
Affinity DataKd:  11nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
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