Compile Data Set for Download or QSAR
maximum 50k data
Found 6 of ic50 for UniProtKB: P04786
TargetDNA topoisomerase 1(Saccharomyces cerevisiae S288c)
Virginia Polytechnic Institute And State University

Curated by ChEMBL
LigandPNGBDBM50090044((Z)-2',3'-dihydroxy-3,4,4',5-tetramethoxystilbene ...)
Affinity DataIC50:  4.81E+3nMAssay Description:Inhibition of topoisomerase 1 in Saccharomyces cerevisiae RS321N in galactose medium by microtiter plate assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Saccharomyces cerevisiae S288c)
Virginia Polytechnic Institute And State University

Curated by ChEMBL
LigandPNGBDBM50090044((Z)-2',3'-dihydroxy-3,4,4',5-tetramethoxystilbene ...)
Affinity DataIC50:  5.71E+3nMAssay Description:Inhibition of topoisomerase 1 in Saccharomyces cerevisiae RS321N in glucose medium by microtiter plate assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Saccharomyces cerevisiae S288c)
Virginia Polytechnic Institute And State University

Curated by ChEMBL
LigandPNGBDBM50005480((-)-combretastatin | (Z)-3'-hydroxy-3,4,4',5-tetra...)
Affinity DataIC50:  2.08E+4nMAssay Description:Inhibition of topoisomerase 1 in Saccharomyces cerevisiae RS321N in galactose medium by microtiter plate assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Saccharomyces cerevisiae S288c)
Virginia Polytechnic Institute And State University

Curated by ChEMBL
LigandPNGBDBM50005480((-)-combretastatin | (Z)-3'-hydroxy-3,4,4',5-tetra...)
Affinity DataIC50:  2.33E+4nMAssay Description:Inhibition of topoisomerase 1 in Saccharomyces cerevisiae RS321N in glucose medium by microtiter plate assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Saccharomyces cerevisiae S288c)
Virginia Polytechnic Institute And State University

Curated by ChEMBL
LigandPNGBDBM50478907(CHEMBL497532)
Affinity DataIC50:  1.38E+5nMAssay Description:Inhibition of topoisomerase 1 in Saccharomyces cerevisiae RS321N in galactose medium by microtiter plate assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Saccharomyces cerevisiae S288c)
Virginia Polytechnic Institute And State University

Curated by ChEMBL
LigandPNGBDBM50478907(CHEMBL497532)
Affinity DataIC50: >2.01E+5nMAssay Description:Inhibition of topoisomerase 1 in Saccharomyces cerevisiae RS321N in glucose medium by microtiter plate assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed