Compile Data Set for Download or QSAR
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Found 6 of ec50 for UniProtKB: A0A024R7T2
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Homo sapiens (Human))
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM60665(BDBM50249542 | US9145414, R406 | US9212178, R406)
Affinity DataEC50:  36nMAssay Description:Inhibition of Ret in human SK-M-MC cells assessed as assessed as phosphorylation after 1 hr incubationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Homo sapiens (Human))
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50242740(CHEMBL459850 | N-(3-(7-Amino-1-methyl-2-oxo-1,2-di...)
Affinity DataEC50:  77nMAssay Description:Inhibition of Ret by cellular assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Homo sapiens (Human))
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM60665(BDBM50249542 | US9145414, R406 | US9212178, R406)
Affinity DataEC50:  80nMAssay Description:Inhibition of Ret in human SK-N-SH cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Homo sapiens (Human))
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50015448(CHEMBL3265032)
Affinity DataEC50: >1.00E+3nMAssay Description:Inhibition of Ret in human SK-M-MC cells assessed as assessed as phosphorylation after 1 hr incubationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Homo sapiens (Human))
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM482158(BDBM50242742 | TAE684)
Affinity DataEC50: >1.00E+3nMAssay Description:Inhibition of Ret by cellular assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Homo sapiens (Human))
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50551644(CHEMBL4745937)
Affinity DataEC50:  2.49E+3nMAssay Description:Inhibition of human RET incubated for 30 mins by Kinobead based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed