Affinity DataIC50: 0.0100nMAssay Description:Compound was tested for its inhibitory activity against Alpha-1 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0200nMAssay Description:Compound was tested for its inhibitory activity against Alpha-1 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0400nMAssay Description:Compound was tested for its inhibitory activity against Alpha-1 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0400nMAssay Description:Compound was tested for its inhibitory activity against Alpha-1 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0700nMAssay Description:Compound was tested for its inhibitory activity against Alpha-1 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.25nMAssay Description:Compound was tested for its inhibitory activity against Alpha-1 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.254nMAssay Description:Displacement of [3H]prazosin from adrenergic alpha1A receptor in Wistar rat submaxillary gland after 60 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.269nMAssay Description:Displacement of [3H]prazosin from rat salivary gland adrenergic alpha 1A receptor after 45 mins by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Antagonist activity at alpha1A adrenoceptor in Sprague-Dawley rat urethra assessed as inhibition of norepinephrine-induced smooth muscle contraction ...More data for this Ligand-Target Pair
Affinity DataIC50: 0.740nMAssay Description:Displacement of [3H]-prazosin from rat alpha1A adrenergic receptor after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 0.800nMAssay Description:Antagonist activity at alpha1A adrenoceptor in Sprague-Dawley rat urethra assessed as inhibition of norepinephrine-induced smooth muscle contraction ...More data for this Ligand-Target Pair
Affinity DataIC50: 0.860nMAssay Description:Inhibitory concentration against human Adenosine A3 receptor expressed in HEK293 cells using 0.1 nM [3H]AB-MECAMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Binding affinity was tested on CEC-pretreated rat hippocampus Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Binding affinity was tested on CEC-pretreated rat hippocampus Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:Binding affinity was tested on CEC-pretreated rat hippocampus Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70nMAssay Description:Inhibition of binding of [3H]imipramine to imipramine receptor in rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Binding affinity was tested on CEC-pretreated rat hippocampus Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 2.5nMAssay Description:Displacement of [3H]-prazosin from rat alpha1A adrenergic receptor after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 3.40nMAssay Description:Displacement of [3H]-prazosin from Alpha-1 adrenergic receptor in whole rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 3.40nMAssay Description:Binding affinity to the alpha-1 adrenergic receptor using a radioligand [3H]-prazosin binding assay in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 4.30nMAssay Description:Displacement of [3H]-prazosin from rat alpha1A adrenergic receptor after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 5.70nMAssay Description:Binding affinity to the alpha-1 adrenergic receptor using a radioligand [3H]-prazosin binding assay in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 6.30nMAssay Description:Displacement of [3H]-prazosin from Alpha-1 adrenergic receptor in whole rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Binding affinity was tested on CEC-pretreated rat hippocampus Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Displacement of [3H]prazosin from rat cerebral cortex alpha1 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Displacement of [3H]-prazosin from Alpha-1 adrenergic receptor in whole rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Binding affinity to the alpha-1 adrenergic receptor using a radioligand [3H]-prazosin binding assay in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Binding affinity to the alpha-1 adrenergic receptor using a radioligand [3H]-prazosin binding assay in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Binding affinity to the alpha-1 adrenergic receptor using a radioligand [3H]-prazosin binding assay in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Binding affinity was tested on CEC-pretreated rat hippocampus Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Binding affinity to the alpha-1 adrenergic receptor using a radioligand [3H]-prazosin binding assay in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Binding affinity to the alpha-1 adrenergic receptor using a radioligand [3H]-prazosin binding assay in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Binding affinity to the alpha-1 adrenergic receptor using a radioligand [3H]-prazosin binding assay in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 19nMAssay Description:Displacement of [3H]-prazosin from Alpha-1 adrenergic receptor in whole rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Displacement of [3H]-prazosin from Alpha-1 adrenergic receptor in whole rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Binding affinity to the alpha-1 adrenergic receptor using a radioligand [3H]-prazosin binding assay in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 24nMAssay Description:Displacement of [3H]-prazosin from Alpha-1 adrenergic receptor in whole rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Displacement of [3H]-prazosin from Alpha-1 adrenergic receptor in whole rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:Binding affinity to the alpha-1 adrenergic receptor using a radioligand [3H]-prazosin binding assay in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 34nMAssay Description:Displacement of [3H]-prazosin from Alpha-1 adrenergic receptor in whole rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 37nMAssay Description:Inhibition of binding of [3H]imipramine to imipramine receptor in rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Binding affinity to the alpha-1 adrenergic receptor using a radioligand [3H]-prazosin binding assay in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 41nMAssay Description:Binding affinity to the alpha-1 adrenergic receptor using a radioligand [3H]-prazosin binding assay in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 43nMAssay Description:Binding affinity to the alpha-1 adrenergic receptor using a radioligand [3H]-prazosin binding assay in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 45nMAssay Description:Antagonist activity at alpha1A adrenoceptor in Sprague-Dawley rat urethra assessed as inhibition of norepinephrine-induced smooth muscle contraction ...More data for this Ligand-Target Pair
Affinity DataIC50: 46nMAssay Description:Antagonist affinity [non competitive (irreversible)] at alpha-1A-adrenoreceptors on isolated prostatic Vas deferens from ratMore data for this Ligand-Target Pair
Affinity DataIC50: 47nMAssay Description:Compound was tested for i the displacement of [3H]-prazosin from alpha-1 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 47nMAssay Description:Compound was tested for the displacement of [3H]-prazosin from alpha-1 adrenergic receptor of rat striatal membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 47nMAssay Description:Binding affinity to the alpha-1 adrenergic receptor using a radioligand [3H]-prazosin binding assay in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 52nMAssay Description:Inhibition of binding of [3H]imipramine to imipramine receptor in rat brainMore data for this Ligand-Target Pair