Compile Data Set for Download or QSAR
maximum 50k data
Found 801 of ki data for polymerid = 6432
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri

Curated by PDSP Ki Database
LigandPNGBDBM29568(CHEMBL2 | PRAZOSIN | PRAZOSIN HYDROCHLORIDE | [3H]...)
Affinity DataKi:  0.0100nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri

Curated by PDSP Ki Database
LigandPNGBDBM29568(CHEMBL2 | PRAZOSIN | PRAZOSIN HYDROCHLORIDE | [3H]...)
Affinity DataKi:  0.0200nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri

Curated by PDSP Ki Database
LigandPNGBDBM50060964((R)-5-(2-((2-(2-ethoxyphenoxy)ethyl)amino)propyl)-...)
Affinity DataKi:  0.0300nMAssay Description:In vitro binding affinity using [3H]-prazosin as radioligand against adrenoceptor alpha 1AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri

Curated by PDSP Ki Database
LigandPNGBDBM50100221(7,8-Dimethoxy-3-[2-(6-methoxy-1,3,3a,4,5,9b-hexahy...)
Affinity DataKi:  0.0400nMAssay Description:Binding affinity to alpha-1A adrenergic receptor in rat submaxillary glandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri

Curated by PDSP Ki Database
LigandPNGBDBM50100210(6-Methoxy-3-[2-(6-methoxy-1,3,3a,4,5,9b-hexahydro-...)
Affinity DataKi:  0.0400nMAssay Description:Binding affinity to alpha-1A adrenergic receptor in rat submaxillary glandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri

Curated by PDSP Ki Database
LigandPNGBDBM29568(CHEMBL2 | PRAZOSIN | PRAZOSIN HYDROCHLORIDE | [3H]...)
Affinity DataKi:  0.0700nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri

Curated by PDSP Ki Database
LigandPNGBDBM29568(CHEMBL2 | PRAZOSIN | PRAZOSIN HYDROCHLORIDE | [3H]...)
Affinity DataKi:  0.0700nMAssay Description:Inhibition of [3H]- prazosin binding against Alpha-1A adrenergic receptor from rat submaxillary glandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri

Curated by PDSP Ki Database
LigandPNGBDBM69602(2,3-dihydro-1,4-benzodioxin-3-ylmethyl-[2-(2,6-dim...)
Affinity DataKi:  0.0800nMAssay Description:Overall binding displacement in tissues containing only the Alpha-1A adrenergic receptor from rat submaxillary glandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri

Curated by PDSP Ki Database
LigandPNGBDBM50100229(3-[2-(6-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]is...)
Affinity DataKi:  0.0900nMAssay Description:Binding affinity to alpha-1A adrenergic receptor in rat submaxillary glandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri

Curated by PDSP Ki Database
LigandPNGBDBM50100214(3-[2-(6-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]is...)
Affinity DataKi:  0.0900nMAssay Description:Binding affinity to alpha-1A adrenergic receptor in rat submaxillary glandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri

Curated by PDSP Ki Database
LigandPNGBDBM50100238(7-Methoxy-3-[2-(6-methoxy-1,3,3a,4,5,9b-hexahydro-...)
Affinity DataKi:  0.0900nMAssay Description:Binding affinity to alpha-1A adrenergic receptor in rat submaxillary glandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri

Curated by PDSP Ki Database
LigandPNGBDBM29568(CHEMBL2 | PRAZOSIN | PRAZOSIN HYDROCHLORIDE | [3H]...)
Affinity DataKi:  0.120nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri

Curated by PDSP Ki Database
LigandPNGBDBM50060964((R)-5-(2-((2-(2-ethoxyphenoxy)ethyl)amino)propyl)-...)
Affinity DataKi:  0.130nMAssay Description:Displacement of [3H]prazosin from rat salivary gland adrenergic alpha 1A receptor after 45 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri

Curated by PDSP Ki Database
LigandPNGBDBM50393116(CHEMBL2153423)
Affinity DataKi:  0.140nMAssay Description:Displacement of [3H]prazosin from rat salivary gland adrenergic alpha 1A receptor after 45 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri

Curated by PDSP Ki Database
LigandPNGBDBM50133938(Aceperone | CHEMBL136298 | N-{1-[4-(4-Fluoro-pheny...)
Affinity DataKi:  0.170nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri

Curated by PDSP Ki Database
LigandPNGBDBM50029257((3-((4-(2-isopropoxyphenyl)piperazin-1-yl)methyl)p...)
Affinity DataKi:  0.200nMAssay Description:Binding affinity towards alpha-1A adrenergic receptors using alpha1A ligand WB4101More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri

Curated by PDSP Ki Database
LigandPNGBDBM50006952(2-{2-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-ethyl}-...)
Affinity DataKi:  0.210nMAssay Description:Binding affinity for Alpha-1 adrenergic receptor measured by displacing [3H]-prazosin from rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri

Curated by PDSP Ki Database
LigandPNGBDBM50369383(CHEMBL1788222)
Affinity DataKi:  0.230nMAssay Description:Displacement of [3H]prazosin from Alpha-1A adrenergic receptorof rat submaxillary gland membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri

Curated by PDSP Ki Database
LigandPNGBDBM29568(CHEMBL2 | PRAZOSIN | PRAZOSIN HYDROCHLORIDE | [3H]...)
Affinity DataKi:  0.230nMAssay Description:Displacement of [3H]prazosin from adrenergic alpha-1A receptor in rat submaxillary gland membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri

Curated by PDSP Ki Database
LigandPNGBDBM50100233(6,7-Dimethoxy-3-[2-(6-methoxy-1,3,3a,4,5,9b-hexahy...)
Affinity DataKi:  0.240nMAssay Description:Binding affinity to alpha-1A adrenergic receptor in rat submaxillary glandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri

Curated by PDSP Ki Database
LigandPNGBDBM50100206(6,7-Dimethoxy-3-[2-(6-methoxy-1,3,3a,4,5,9b-hexahy...)
Affinity DataKi:  0.25nMAssay Description:Binding affinity to alpha-1A adrenergic receptor in rat submaxillary glandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri

Curated by PDSP Ki Database
LigandPNGBDBM50066109(3-[4-(2-Methoxy-phenyl)-piperazin-1-ylmethyl]-2,6-...)
Affinity DataKi:  0.260nMAssay Description:Displacement of [3H]prazosin from Alpha-1A adrenergic receptorof rat submaxillary gland membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri

Curated by PDSP Ki Database
LigandPNGBDBM50100222(6,7-Dimethoxy-3-[2-(6-methoxy-1,3,3a,4,5,9b-hexahy...)
Affinity DataKi:  0.270nMAssay Description:Binding affinity to alpha-1A adrenergic receptor in rat submaxillary glandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri

Curated by PDSP Ki Database
LigandPNGBDBM50100228(3-[2-(6-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]is...)
Affinity DataKi:  0.270nMAssay Description:Binding affinity to alpha-1A adrenergic receptor in rat submaxillary glandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri

Curated by PDSP Ki Database
LigandPNGBDBM50060965(2-[2-((3aR,9bR)-6-Methoxy-1,3,3a,4,5,9b-hexahydro-...)
Affinity DataKi:  0.270nMAssay Description:In vitro binding affinity using [3H]-prazosin as radioligand against alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri

Curated by PDSP Ki Database
LigandPNGBDBM50087470(3-[2-(6-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]is...)
Affinity DataKi:  0.280nMAssay Description:In vitro binding affinity using [3H]-prazosin as radioligand against alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri

Curated by PDSP Ki Database
LigandPNGBDBM50087488(3-[2-(6-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]is...)
Affinity DataKi:  0.290nMAssay Description:In vitro binding affinity using [3H]-prazosin as radioligand against alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri

Curated by PDSP Ki Database
LigandPNGBDBM81444(CAS_185453 | NSC_185453 | WB 4101 | WB-4101)
Affinity DataKi:  0.300nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri

Curated by PDSP Ki Database
LigandPNGBDBM50231449(CHEMBL398711 | N-(5-(2-(4-(benzo[d]isothiazol-3-yl...)
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H]prazosin from rat adrenergic alpha1A receptor expressed in fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri

Curated by PDSP Ki Database
LigandPNGBDBM29568(CHEMBL2 | PRAZOSIN | PRAZOSIN HYDROCHLORIDE | [3H]...)
Affinity DataKi:  0.300nMAssay Description:Compound was evaluated for its ability to displace [125I]-HEAT binding from rat Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri

Curated by PDSP Ki Database
LigandPNGBDBM29568(CHEMBL2 | PRAZOSIN | PRAZOSIN HYDROCHLORIDE | [3H]...)
Affinity DataKi:  0.310nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri

Curated by PDSP Ki Database
LigandPNGBDBM50006953(2-{2-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-ethyl}-...)
Affinity DataKi:  0.320nMAssay Description:Binding affinity for Alpha-1 adrenergic receptor measured by displacing [3H]-prazosin from rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri

Curated by PDSP Ki Database
LigandPNGBDBM29568(CHEMBL2 | PRAZOSIN | PRAZOSIN HYDROCHLORIDE | [3H]...)
Affinity DataKi:  0.330nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri

Curated by PDSP Ki Database
LigandPNGBDBM50100216(3-[2-(6-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]is...)
Affinity DataKi:  0.330nMAssay Description:Binding affinity to alpha-1A adrenergic receptor in rat submaxillary glandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri

Curated by PDSP Ki Database
LigandPNGBDBM50087485(2-[2-(6-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]is...)
Affinity DataKi:  0.330nMAssay Description:In vitro binding affinity using [3H]-prazosin as radioligand against alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri

Curated by PDSP Ki Database
LigandPNGBDBM50087490(3-Methoxy-7-[2-(6-methoxy-1,3,3a,4,5,9b-hexahydro-...)
Affinity DataKi:  0.350nMAssay Description:In vitro binding affinity using [3H]-prazosin as radioligand against alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri

Curated by PDSP Ki Database
LigandPNGBDBM50090647((4S,5S)-4-(3,4-Difluoro-phenyl)-5-methyl-2-oxo-oxa...)
Affinity DataKi:  0.360nMAssay Description:Binding affinity towards Alpha1A rat adrenergic receptors, using [125I]HEAT as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri

Curated by PDSP Ki Database
LigandPNGBDBM50087484(6-Chloro-2-[2-(6-methoxy-1,3,3a,4,5,9b-hexahydro-b...)
Affinity DataKi:  0.380nMAssay Description:In vitro binding affinity using [3H]-prazosin as radioligand against adrenoceptor alpha 1AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri

Curated by PDSP Ki Database
LigandPNGBDBM50087476(7-[2-(6-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]is...)
Affinity DataKi:  0.390nMAssay Description:In vitro binding affinity using [3H]-prazosin as radioligand against alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri

Curated by PDSP Ki Database
LigandPNGBDBM50087473(3-[2-(6-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]is...)
Affinity DataKi:  0.400nMAssay Description:In vitro binding affinity using [3H]-prazosin as radioligand against alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri

Curated by PDSP Ki Database
LigandPNGBDBM50100217(7-Isopropyl-6-methoxy-3-[2-(6-methoxy-1,3,3a,4,5,9...)
Affinity DataKi:  0.410nMAssay Description:Binding affinity to alpha-1A adrenergic receptor in rat submaxillary glandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri

Curated by PDSP Ki Database
LigandPNGBDBM50100220(CHEMBL61598 | N-{3-[2-(6-Methoxy-1,3,3a,4,5,9b-hex...)
Affinity DataKi:  0.430nMAssay Description:Binding affinity to alpha-1A adrenergic receptor in rat submaxillary glandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri

Curated by PDSP Ki Database
LigandPNGBDBM50087496(8-Chloro-3-[2-(6-methoxy-1,3,3a,4,5,9b-hexahydro-b...)
Affinity DataKi:  0.440nMAssay Description:In vitro binding affinity using [3H]-prazosin as radioligand against alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri

Curated by PDSP Ki Database
LigandPNGBDBM50231441(CHEMBL252031 | N-(5-(2-(4-(benzo[d]isothiazol-3-yl...)
Affinity DataKi:  0.450nMAssay Description:Displacement of [3H]prazosin from rat adrenergic alpha1A receptor expressed in fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri

Curated by PDSP Ki Database
LigandPNGBDBM81980(Butanserin | CAS_87051-46-5 | NSC_65652)
Affinity DataKi:  0.450nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri

Curated by PDSP Ki Database
LigandPNGBDBM50100215(3-[2-(6-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]is...)
Affinity DataKi:  0.480nMAssay Description:Binding affinity to alpha-1A adrenergic receptor in rat submaxillary glandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri

Curated by PDSP Ki Database
LigandPNGBDBM50087493(7-[2-(6-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]is...)
Affinity DataKi:  0.490nMAssay Description:In vitro binding affinity using [3H]-prazosin as radioligand against alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri

Curated by PDSP Ki Database
LigandPNGBDBM50231460(CHEMBL398525 | N-(5-(2-(4-(benzo[d]isothiazol-3-yl...)
Affinity DataKi:  0.490nMAssay Description:Displacement of [3H]prazosin from rat adrenergic alpha1A receptor expressed in fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri

Curated by PDSP Ki Database
LigandPNGBDBM50040253(3-{2-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-ethyl}-...)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]prazosin from Alpha-1A adrenergic receptorof rat submaxillary gland membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri

Curated by PDSP Ki Database
LigandPNGBDBM50048803(5-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)et...)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]prazosin from rat adrenergic alpha1A receptor expressed in fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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