Compile Data Set for Download or QSAR
maximum 50k data
Found 38 Enz. Inhib. hit(s) with all data for entry = 1122
TargetAcetylcholinesterase(Rattus norvegicus (rat))
National Defense Medical Center

LigandPNGBDBM9054(6-chloro-N-{7-[(6-chloro-1,2,3,4-tetrahydroacridin...)
Affinity DataIC50:  0.0700nMpH: 7.4 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
National Defense Medical Center

LigandPNGBDBM8963(CHEMBL32823 | Homodimeric Tacrine Analog 3b | N-[7...)
Affinity DataIC50:  0.200nMpH: 7.4 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
National Defense Medical Center

LigandPNGBDBM9055(6-chloro-N-{8-[(6-chloro-1,2,3,4-tetrahydroacridin...)
Affinity DataIC50:  0.300nMpH: 7.4 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
National Defense Medical Center

LigandPNGBDBM9053(6-chloro-N-{6-[(6-chloro-1,2,3,4-tetrahydroacridin...)
Affinity DataIC50:  0.600nMpH: 7.4 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
National Defense Medical Center

LigandPNGBDBM9051(6-fluoro-N-{7-[(6-fluoro-1,2,3,4-tetrahydroacridin...)
Affinity DataIC50:  0.600nMpH: 7.4 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
National Defense Medical Center

LigandPNGBDBM9052(6-fluoro-N-{8-[(6-fluoro-1,2,3,4-tetrahydroacridin...)
Affinity DataIC50:  0.700nMpH: 7.4 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
National Defense Medical Center

LigandPNGBDBM9050(6-fluoro-N-{6-[(6-fluoro-1,2,3,4-tetrahydroacridin...)
Affinity DataIC50:  0.900nMpH: 7.4 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
National Defense Medical Center

LigandPNGBDBM9057(Homodimeric Tacrine Analog 3k | N,N-Bis-(1,2,3,4-t...)
Affinity DataIC50:  1.30nMpH: 7.4 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
National Defense Medical Center

LigandPNGBDBM9047(Bis-THA inhibitor 5 | CHEMBL73800 | Hexylene-Linke...)
Affinity DataIC50:  1.40nMpH: 7.4 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
National Defense Medical Center

LigandPNGBDBM9061(Homodimeric Tacrine Analog 4c | N,N-Bis-(2,3,4,5-t...)
Affinity DataIC50:  1.60nMpH: 7.4 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
National Defense Medical Center

LigandPNGBDBM8964(CHEMBL75274 | Homodimeric Tacrine Analog 3c | N-[8...)
Affinity DataIC50:  1.60nMpH: 7.4 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
National Defense Medical Center

LigandPNGBDBM9058(Homodimeric Tacrine Analog 3m | N,N-Bis-(1,2,3,4-t...)
Affinity DataIC50:  1.90nMpH: 7.4 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
National Defense Medical Center

LigandPNGBDBM9059(Homodimeric Tacrine Analog 4a | N,N-Bis-(2,3,4,5-t...)
Affinity DataIC50:  2.5nMpH: 7.4 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
National Defense Medical Center

LigandPNGBDBM9060(Homodimeric Tacrine Analog 4b | N,N-Bis-(2,3,4,5-t...)
Affinity DataIC50:  2.60nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
National Defense Medical Center

LigandPNGBDBM9060(Homodimeric Tacrine Analog 4b | N,N-Bis-(2,3,4,5-t...)
Affinity DataIC50:  2.70nMpH: 7.4 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
National Defense Medical Center

LigandPNGBDBM9059(Homodimeric Tacrine Analog 4a | N,N-Bis-(2,3,4,5-t...)
Affinity DataIC50:  3.30nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
National Defense Medical Center

LigandPNGBDBM9061(Homodimeric Tacrine Analog 4c | N,N-Bis-(2,3,4,5-t...)
Affinity DataIC50:  3.80nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
National Defense Medical Center

LigandPNGBDBM9056(Homodimeric Tacrine Analog 3j | N,N-Bis-(1,2,3,4-t...)
Affinity DataIC50:  4.80nMpH: 7.4 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
National Defense Medical Center

LigandPNGBDBM9046(Homodimeric Tacrine Analog 2c | N,N-Bis-(2,3-dihyd...)
Affinity DataIC50:  22nMpH: 7.4 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
National Defense Medical Center

LigandPNGBDBM9058(Homodimeric Tacrine Analog 3m | N,N-Bis-(1,2,3,4-t...)
Affinity DataIC50:  23nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
National Defense Medical Center

LigandPNGBDBM9054(6-chloro-N-{7-[(6-chloro-1,2,3,4-tetrahydroacridin...)
Affinity DataIC50:  26nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
National Defense Medical Center

LigandPNGBDBM9050(6-fluoro-N-{6-[(6-fluoro-1,2,3,4-tetrahydroacridin...)
Affinity DataIC50:  45nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
National Defense Medical Center

LigandPNGBDBM8964(CHEMBL75274 | Homodimeric Tacrine Analog 3c | N-[8...)
Affinity DataIC50:  53nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
National Defense Medical Center

LigandPNGBDBM8963(CHEMBL32823 | Homodimeric Tacrine Analog 3b | N-[7...)
Affinity DataIC50:  54nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
National Defense Medical Center

LigandPNGBDBM9057(Homodimeric Tacrine Analog 3k | N,N-Bis-(1,2,3,4-t...)
Affinity DataIC50:  59nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
National Defense Medical Center

LigandPNGBDBM9045(Homodimeric Tacrine Analog 2b | N,N-Bis-(2,3-dihyd...)
Affinity DataIC50:  75nMpH: 7.4 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
National Defense Medical Center

LigandPNGBDBM9047(Bis-THA inhibitor 5 | CHEMBL73800 | Hexylene-Linke...)
Affinity DataIC50:  83nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
National Defense Medical Center

LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataIC50:  89nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
TargetCholinesterase(Homo sapiens (Human))
National Defense Medical Center

LigandPNGBDBM9056(Homodimeric Tacrine Analog 3j | N,N-Bis-(1,2,3,4-t...)
Affinity DataIC50:  93nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
National Defense Medical Center

LigandPNGBDBM9044(Homodimeric Tacrine Analog 2a | N,N-Bis-(2,3-dihyd...)
Affinity DataIC50:  115nMpH: 7.4 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
National Defense Medical Center

LigandPNGBDBM9052(6-fluoro-N-{8-[(6-fluoro-1,2,3,4-tetrahydroacridin...)
Affinity DataIC50:  164nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
National Defense Medical Center

LigandPNGBDBM9046(Homodimeric Tacrine Analog 2c | N,N-Bis-(2,3-dihyd...)
Affinity DataIC50:  165nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
National Defense Medical Center

LigandPNGBDBM9055(6-chloro-N-{8-[(6-chloro-1,2,3,4-tetrahydroacridin...)
Affinity DataIC50:  194nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
National Defense Medical Center

LigandPNGBDBM9051(6-fluoro-N-{7-[(6-fluoro-1,2,3,4-tetrahydroacridin...)
Affinity DataIC50:  257nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
National Defense Medical Center

LigandPNGBDBM9044(Homodimeric Tacrine Analog 2a | N,N-Bis-(2,3-dihyd...)
Affinity DataIC50:  273nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
National Defense Medical Center

LigandPNGBDBM9053(6-chloro-N-{6-[(6-chloro-1,2,3,4-tetrahydroacridin...)
Affinity DataIC50:  312nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
National Defense Medical Center

LigandPNGBDBM9045(Homodimeric Tacrine Analog 2b | N,N-Bis-(2,3-dihyd...)
Affinity DataIC50:  328nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
National Defense Medical Center

LigandPNGBDBM9061(Homodimeric Tacrine Analog 4c | N,N-Bis-(2,3,4,5-t...)
Affinity DataIC50:  333nMpH: 7.4 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed