Compile Data Set for Download or QSAR
maximum 50k data
Found 48 Enz. Inhib. hit(s) with all data for entry = 50001899
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50007329((R)-2-[(R)-2-(2-{2-[(R)-2-Amino-3-(4-hydroxy-pheny...)
Affinity DataKi:  2.5nMAssay Description:Inhibition of [3H]-DSLET binding to rat brain membrane Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50007329((R)-2-[(R)-2-(2-{2-[(R)-2-Amino-3-(4-hydroxy-pheny...)
Affinity DataKi:  9.40nMAssay Description:Binding affinity towards Opioid receptor mu 1 in rat brain membrane using [3H]-DAGO as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50018637(12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2...)
Affinity DataKi:  9.60nMAssay Description:Binding affinity towards Opioid receptor mu 1 in rat brain membrane using [3H]-DAGO as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50001467(12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2...)
Affinity DataKi:  10nMAssay Description:Binding affinity towards Opioid receptor mu 1 in rat brain membrane using [3H]-DAGO as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50018640(10-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7...)
Affinity DataKi:  11nMAssay Description:Binding affinity towards Opioid receptor mu 1 in rat brain membrane using [3H]-DAGO as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50018631(12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-3...)
Affinity DataKi:  12nMAssay Description:Binding affinity towards Opioid receptor mu 1 in rat brain membrane using [3H]-DAGO as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50018635(12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2...)
Affinity DataKi:  22nMAssay Description:Binding affinity towards Opioid receptor mu 1 in rat brain membrane using [3H]-DAGO as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50018639(11-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2...)
Affinity DataKi:  25nMAssay Description:Binding affinity towards Opioid receptor mu 1 in rat brain membrane using [3H]-DAGO as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50018638(12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2...)
Affinity DataKi:  273nMAssay Description:Binding affinity towards Opioid receptor mu 1 in rat brain membrane using [3H]-DAGO as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50018640(10-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7...)
Affinity DataKi:  373nMAssay Description:Inhibition of [3H]-DSLET binding to rat brain membrane Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50018635(12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2...)
Affinity DataKi:  422nMAssay Description:Inhibition of [3H]-DSLET binding to rat brain membrane Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50018633(12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2...)
Affinity DataKi:  445nMAssay Description:Binding affinity towards mu Opioid receptor in rat brain membrane using [3H]-DAGO as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50018631(12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-3...)
Affinity DataKi:  849nMAssay Description:Inhibition of [3H]-DSLET binding to rat brain membrane Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50018637(12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2...)
Affinity DataKi:  1.32E+3nMAssay Description:Inhibition of [3H]-DSLET binding to rat brain membrane Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50001467(12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2...)
Affinity DataKi:  2.22E+3nMAssay Description:Inhibition of [3H]-DSLET binding to rat brain membrane Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50018632(12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2...)
Affinity DataKi:  3.04E+3nMAssay Description:Binding affinity towards Opioid receptor mu 1 in rat brain membrane using [3H]-DAGO as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50018633(12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2...)
Affinity DataKi:  3.57E+3nMAssay Description:Inhibition of [3H]-DSLET binding to rat brain membrane Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50018636(12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2...)
Affinity DataKi:  3.57E+3nMAssay Description:Binding affinity towards Opioid receptor mu 1 in rat brain membrane using [3H]-DAGO as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50018639(11-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2...)
Affinity DataKi:  4.17E+3nMAssay Description:Inhibition of [3H]-DSLET binding to rat brain membrane Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50018634(12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2...)
Affinity DataKi:  4.83E+3nMAssay Description:Binding affinity towards mu Opioid receptor in rat brain membrane using [3H]-DAGO as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50018638(12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2...)
Affinity DataKi:  5.06E+3nMAssay Description:Inhibition of [3H]-DSLET binding to rat brain membrane Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50018636(12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2...)
Affinity DataKi:  2.81E+4nMAssay Description:Inhibition of [3H]-DSLET binding to rat brain membrane Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50018634(12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2...)
Affinity DataKi: >6.00E+4nMAssay Description:Inhibition of [3H]-DSLET binding to rat brain membrane Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50018632(12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2...)
Affinity DataKi: >3.80E+5nMAssay Description:Inhibition of [3H]-DSLET binding to rat brain membrane Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50007329((R)-2-[(R)-2-(2-{2-[(R)-2-Amino-3-(4-hydroxy-pheny...)
Affinity DataIC50:  11nMAssay Description:Inhibitory activity towards delta Opioid receptor using guinea pig ileum (GPI) assay was determined for the compoundMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50001467(12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2...)
Affinity DataIC50:  36nMAssay Description:Inhibitory activity towards electrically induced contractions in guinea pig ileum expressing mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50018640(10-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7...)
Affinity DataIC50:  65nMAssay Description:Inhibitory activity towards Opioid receptor mu 1 using guinea pig ileum (GPI) assay was determined for the compoundMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50018631(12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-3...)
Affinity DataIC50:  111nMAssay Description:Inhibitory activity towards electrically induced contractions in guinea pig ileum expressing Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50007329((R)-2-[(R)-2-(2-{2-[(R)-2-Amino-3-(4-hydroxy-pheny...)
Affinity DataIC50:  246nMAssay Description:Inhibitory activity towards Opioid receptor mu 1 using guinea pig ileum (GPI) assay was determined for the compoundMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50018639(11-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2...)
Affinity DataIC50:  279nMAssay Description:Inhibitory activity towards electrically induced contractions in guinea pig ileum expressing Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50018637(12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2...)
Affinity DataIC50:  522nMAssay Description:Inhibitory activity towards electrically induced contractions in guinea pig ileum expressing Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50018635(12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2...)
Affinity DataIC50:  632nMAssay Description:Inhibitory activity towards electrically induced contractions in guinea pig ileum expressing Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50018640(10-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7...)
Affinity DataIC50:  740nMAssay Description:Inhibitory activity towards delta Opioid receptor using guinea pig ileum (GPI) assay was determined for the compoundMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50018631(12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-3...)
Affinity DataIC50:  1.37E+3nMAssay Description:Inhibitory activity towards electrically induced contractions in mouse vas deferens expressing delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50018636(12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2...)
Affinity DataIC50:  1.38E+3nMAssay Description:Inhibitory activity towards electrically induced contractions in mouse vas deferens expressing delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50018633(12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2...)
Affinity DataIC50:  1.66E+3nMAssay Description:Inhibitory activity towards electrically induced contractions in mouse vas deferens expressing delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50018639(11-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2...)
Affinity DataIC50:  2.03E+3nMAssay Description:Inhibitory activity towards electrically induced contractions in mouse vas deferens expressing delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50018638(12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2...)
Affinity DataIC50:  2.34E+3nMAssay Description:Inhibitory activity towards electrically induced contractions in guinea pig ileum expressing Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50001467(12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2...)
Affinity DataIC50:  3.88E+3nMAssay Description:Inhibitory activity towards electrically induced contractions in mouse vas deferens expressing delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50018635(12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2...)
Affinity DataIC50:  4.81E+3nMAssay Description:Inhibitory activity towards electrically induced contractions in mouse vas deferens expressing delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50018636(12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2...)
Affinity DataIC50:  6.46E+3nMAssay Description:Inhibitory activity towards electrically induced contractions in guinea pig ileum expressing Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50018637(12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2...)
Affinity DataIC50:  8.57E+3nMAssay Description:Inhibitory activity towards electrically induced contractions in mouse vas deferens expressing delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50018632(12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2...)
Affinity DataIC50: >8.64E+3nMAssay Description:Inhibitory activity towards electrically induced contractions in mouse vas deferens expressing delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50018634(12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2...)
Affinity DataIC50:  1.68E+4nMAssay Description:Inhibitory activity towards electrically induced contractions in guinea pig ileum expressing Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50018633(12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2...)
Affinity DataIC50:  1.84E+4nMAssay Description:Inhibitory activity towards electrically induced contractions in guinea pig ileum expressing Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50018632(12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2...)
Affinity DataIC50: >2.10E+4nMAssay Description:Inhibitory activity towards electrically induced contractions in guinea pig ileum expressing Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50018638(12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity towards electrically induced contractions in mouse vas deferens expressing delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50018634(12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity towards electrically induced contractions in mouse vas deferens expressing delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed