TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: 2.5nMAssay Description:Inhibition of [3H]-DSLET binding to rat brain membrane Opioid receptor delta 1More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: 9.40nMAssay Description:Binding affinity towards Opioid receptor mu 1 in rat brain membrane using [3H]-DAGO as radioligandMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: 9.60nMAssay Description:Binding affinity towards Opioid receptor mu 1 in rat brain membrane using [3H]-DAGO as radioligandMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Binding affinity towards Opioid receptor mu 1 in rat brain membrane using [3H]-DAGO as radioligandMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Binding affinity towards Opioid receptor mu 1 in rat brain membrane using [3H]-DAGO as radioligandMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Binding affinity towards Opioid receptor mu 1 in rat brain membrane using [3H]-DAGO as radioligandMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: 22nMAssay Description:Binding affinity towards Opioid receptor mu 1 in rat brain membrane using [3H]-DAGO as radioligandMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: 25nMAssay Description:Binding affinity towards Opioid receptor mu 1 in rat brain membrane using [3H]-DAGO as radioligandMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: 273nMAssay Description:Binding affinity towards Opioid receptor mu 1 in rat brain membrane using [3H]-DAGO as radioligandMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: 373nMAssay Description:Inhibition of [3H]-DSLET binding to rat brain membrane Opioid receptor delta 1More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: 422nMAssay Description:Inhibition of [3H]-DSLET binding to rat brain membrane Opioid receptor delta 1More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: 445nMAssay Description:Binding affinity towards mu Opioid receptor in rat brain membrane using [3H]-DAGO as radioligandMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: 849nMAssay Description:Inhibition of [3H]-DSLET binding to rat brain membrane Opioid receptor delta 1More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: 1.32E+3nMAssay Description:Inhibition of [3H]-DSLET binding to rat brain membrane Opioid receptor delta 1More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: 2.22E+3nMAssay Description:Inhibition of [3H]-DSLET binding to rat brain membrane Opioid receptor delta 1More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: 3.04E+3nMAssay Description:Binding affinity towards Opioid receptor mu 1 in rat brain membrane using [3H]-DAGO as radioligandMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: 3.57E+3nMAssay Description:Inhibition of [3H]-DSLET binding to rat brain membrane Opioid receptor delta 1More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: 3.57E+3nMAssay Description:Binding affinity towards Opioid receptor mu 1 in rat brain membrane using [3H]-DAGO as radioligandMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: 4.17E+3nMAssay Description:Inhibition of [3H]-DSLET binding to rat brain membrane Opioid receptor delta 1More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: 4.83E+3nMAssay Description:Binding affinity towards mu Opioid receptor in rat brain membrane using [3H]-DAGO as radioligandMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: 5.06E+3nMAssay Description:Inhibition of [3H]-DSLET binding to rat brain membrane Opioid receptor delta 1More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: 2.81E+4nMAssay Description:Inhibition of [3H]-DSLET binding to rat brain membrane Opioid receptor delta 1More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: >6.00E+4nMAssay Description:Inhibition of [3H]-DSLET binding to rat brain membrane Opioid receptor delta 1More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: >3.80E+5nMAssay Description:Inhibition of [3H]-DSLET binding to rat brain membrane Opioid receptor delta 1More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibitory activity towards delta Opioid receptor using guinea pig ileum (GPI) assay was determined for the compoundMore data for this Ligand-Target Pair
Affinity DataIC50: 36nMAssay Description:Inhibitory activity towards electrically induced contractions in guinea pig ileum expressing mu opioid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 65nMAssay Description:Inhibitory activity towards Opioid receptor mu 1 using guinea pig ileum (GPI) assay was determined for the compoundMore data for this Ligand-Target Pair
Affinity DataIC50: 111nMAssay Description:Inhibitory activity towards electrically induced contractions in guinea pig ileum expressing Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataIC50: 246nMAssay Description:Inhibitory activity towards Opioid receptor mu 1 using guinea pig ileum (GPI) assay was determined for the compoundMore data for this Ligand-Target Pair
Affinity DataIC50: 279nMAssay Description:Inhibitory activity towards electrically induced contractions in guinea pig ileum expressing Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataIC50: 522nMAssay Description:Inhibitory activity towards electrically induced contractions in guinea pig ileum expressing Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataIC50: 632nMAssay Description:Inhibitory activity towards electrically induced contractions in guinea pig ileum expressing Opioid receptor mu 1More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataIC50: 740nMAssay Description:Inhibitory activity towards delta Opioid receptor using guinea pig ileum (GPI) assay was determined for the compoundMore data for this Ligand-Target Pair
Affinity DataIC50: 1.37E+3nMAssay Description:Inhibitory activity towards electrically induced contractions in mouse vas deferens expressing delta opioid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.38E+3nMAssay Description:Inhibitory activity towards electrically induced contractions in mouse vas deferens expressing delta opioid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.66E+3nMAssay Description:Inhibitory activity towards electrically induced contractions in mouse vas deferens expressing delta opioid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 2.03E+3nMAssay Description:Inhibitory activity towards electrically induced contractions in mouse vas deferens expressing delta opioid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 2.34E+3nMAssay Description:Inhibitory activity towards electrically induced contractions in guinea pig ileum expressing Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataIC50: 3.88E+3nMAssay Description:Inhibitory activity towards electrically induced contractions in mouse vas deferens expressing delta opioid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 4.81E+3nMAssay Description:Inhibitory activity towards electrically induced contractions in mouse vas deferens expressing delta opioid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 6.46E+3nMAssay Description:Inhibitory activity towards electrically induced contractions in guinea pig ileum expressing Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataIC50: 8.57E+3nMAssay Description:Inhibitory activity towards electrically induced contractions in mouse vas deferens expressing delta opioid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: >8.64E+3nMAssay Description:Inhibitory activity towards electrically induced contractions in mouse vas deferens expressing delta opioid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.68E+4nMAssay Description:Inhibitory activity towards electrically induced contractions in guinea pig ileum expressing Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataIC50: 1.84E+4nMAssay Description:Inhibitory activity towards electrically induced contractions in guinea pig ileum expressing Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataIC50: >2.10E+4nMAssay Description:Inhibitory activity towards electrically induced contractions in guinea pig ileum expressing Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity towards electrically induced contractions in mouse vas deferens expressing delta opioid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity towards electrically induced contractions in mouse vas deferens expressing delta opioid receptorMore data for this Ligand-Target Pair