Compile Data Set for Download or QSAR
maximum 50k data
Found 12 Enz. Inhib. hit(s) with all data for entry = 50000547
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Washington

Curated by ChEMBL
LigandPNGBDBM50007095(6,11-Diethyl-3-furan-3-ylmethyl-1,2,3,4,5,6-hexahy...)
Affinity DataIC50:  1.60nMAssay Description:Displacement of [3H]-bremazocine from opioid receptor kappa of guinea pig membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Washington

Curated by ChEMBL
LigandPNGBDBM50007102(6,11-Dimethyl-3-(tetrahydro-furan-2-ylmethyl)-1,2,...)
Affinity DataIC50:  1.70nMAssay Description:Displacement of [3H]-bremazocine from opioid receptor kappa of guinea pig membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Washington

Curated by ChEMBL
LigandPNGBDBM50453067(CHEMBL2367762)
Affinity DataIC50:  5.40nMAssay Description:Displacement of [3H]-bremazocine from opioid receptor kappa of guinea pig membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Washington

Curated by ChEMBL
LigandPNGBDBM50007096(3-Furan-2-ylmethyl-6,11-dimethyl-1,2,3,4,5,6-hexah...)
Affinity DataIC50:  5.70nMAssay Description:Displacement of [3H]-bremazocine from opioid receptor kappa of guinea pig membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Washington

Curated by ChEMBL
LigandPNGBDBM50453069(CHEMBL2367764)
Affinity DataIC50:  7.30nMAssay Description:Displacement of [3H]-bremazocine from opioid receptor kappa of guinea pig membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Washington

Curated by ChEMBL
LigandPNGBDBM60212((4R,4aS,7aR,12bS)-3-(cyclopropylmethyl)-4a,9-bis(o...)
Affinity DataIC50:  9.5nMAssay Description:Displacement of [3H]-bremazocine from opioid receptor kappa of guinea pig membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Washington

Curated by ChEMBL
LigandPNGBDBM50453075(CHEMBL2367603)
Affinity DataIC50:  70nMAssay Description:Displacement of [3H]-bremazocine from opioid receptor kappa of guinea pig membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Washington

Curated by ChEMBL
LigandPNGBDBM50453071(CHEMBL2367758)
Affinity DataIC50:  74nMAssay Description:Displacement of [3H]-bremazocine from opioid receptor kappa of guinea pig membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Washington

Curated by ChEMBL
LigandPNGBDBM50007098(6,11-Dimethyl-3-(tetrahydro-furan-2-ylmethyl)-1,2,...)
Affinity DataIC50:  400nMAssay Description:Displacement of [3H]-bremazocine from opioid receptor kappa of guinea pig membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Washington

Curated by ChEMBL
LigandPNGBDBM50453066(CHEMBL2367761)
Affinity DataIC50:  400nMAssay Description:Displacement of [3H]-bremazocine from opioid receptor kappa of guinea pig membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type/Kappa-type/Mu-type opioid receptor(Homo sapiens (Human))
University Of Washington

Curated by ChEMBL
LigandPNGBDBM50229519(CHEMBL81021 | MR-2035)
Affinity DataIC50:  1.00E+3nMAssay Description:Displacement of 0.5 nM [3H]bremazocine from opioid receptor sites in guinea pig membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type/Kappa-type/Mu-type opioid receptor(Homo sapiens (Human))
University Of Washington

Curated by ChEMBL
LigandPNGBDBM50229516(CHEMBL2367763)
Affinity DataIC50:  1.30E+3nMAssay Description:Displacement of 0.5 nM [3H]bremazocine from opioid receptor sites in guinea pig membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed