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Found 21 Enz. Inhib. hit(s) with all data for entry = 50036029
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50001107(2-(3,4-Dichloro-phenyl)-1-(5-hydroxy-1-pyrrolidin-...)
Affinity DataKi:  0.0900nMAssay Description:Receptor binding affinity towards opioid receptor kappaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50001108(2-(3,4-Dichloro-phenyl)-1-(1-pyrrolidin-1-ylmethyl...)
Affinity DataKi:  0.200nMAssay Description:Receptor binding affinity towards opioid receptor kappaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50001104(2-(3,4-Dichloro-phenyl)-1-(3-methyl-1-pyrrolidin-1...)
Affinity DataKi:  0.430nMAssay Description:Receptor binding affinity towards opioid receptor kappaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50001107(2-(3,4-Dichloro-phenyl)-1-(5-hydroxy-1-pyrrolidin-...)
Affinity DataKi:  0.490nMAssay Description:Receptor binding affinity towards opioid receptor muMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50001105(2-(3,4-Dichloro-phenyl)-1-(4-methyl-1-pyrrolidin-1...)
Affinity DataKi:  0.600nMAssay Description:Receptor binding affinity towards opioid receptor kappaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50000296(CHEMBL441765 | CHEMBL482811 | U-50488H | US1149237...)
Affinity DataKi:  2.20nMAssay Description:Receptor binding affinity towards opioid receptor kappaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50001106(2-(3,4-Dichloro-phenyl)-1-(4,4-dimethyl-1-pyrrolid...)
Affinity DataKi:  2.30nMAssay Description:Receptor binding affinity towards opioid receptor kappaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  3.30nMAssay Description:Receptor binding affinity towards opioid receptor muMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50001107(2-(3,4-Dichloro-phenyl)-1-(5-hydroxy-1-pyrrolidin-...)
Affinity DataKi:  7.10nMAssay Description:Receptor binding affinity towards opioid receptor deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50001104(2-(3,4-Dichloro-phenyl)-1-(3-methyl-1-pyrrolidin-1...)
Affinity DataKi:  11nMAssay Description:Receptor binding affinity towards opioid receptor muMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50001108(2-(3,4-Dichloro-phenyl)-1-(1-pyrrolidin-1-ylmethyl...)
Affinity DataKi:  30nMAssay Description:Receptor binding affinity towards opioid receptor muMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50001104(2-(3,4-Dichloro-phenyl)-1-(3-methyl-1-pyrrolidin-1...)
Affinity DataKi:  44nMAssay Description:Receptor binding affinity towards opioid receptor deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50001105(2-(3,4-Dichloro-phenyl)-1-(4-methyl-1-pyrrolidin-1...)
Affinity DataKi:  57nMAssay Description:Receptor binding affinity towards opioid receptor muMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50001108(2-(3,4-Dichloro-phenyl)-1-(1-pyrrolidin-1-ylmethyl...)
Affinity DataKi:  113nMAssay Description:Receptor binding affinity towards opioid receptor deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50001105(2-(3,4-Dichloro-phenyl)-1-(4-methyl-1-pyrrolidin-1...)
Affinity DataKi:  158nMAssay Description:Receptor binding affinity towards opioid receptor deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50001106(2-(3,4-Dichloro-phenyl)-1-(4,4-dimethyl-1-pyrrolid...)
Affinity DataKi:  239nMAssay Description:Receptor binding affinity towards opioid receptor muMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  301nMAssay Description:Receptor binding affinity towards opioid receptor kappaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  456nMAssay Description:Receptor binding affinity towards opioid receptor deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetMu-type opioid receptor(GUINEA PIG)
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50000296(CHEMBL441765 | CHEMBL482811 | U-50488H | US1149237...)
Affinity DataKi:  616nMAssay Description:Receptor binding affinity towards opioid receptor muMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50001106(2-(3,4-Dichloro-phenyl)-1-(4,4-dimethyl-1-pyrrolid...)
Affinity DataKi:  1.01E+3nMAssay Description:Receptor binding affinity towards opioid receptor deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50000296(CHEMBL441765 | CHEMBL482811 | U-50488H | US1149237...)
Affinity DataKi: >1.00E+4nMAssay Description:Receptor binding affinity towards opioid receptor deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed