Compile Data Set for Download or QSAR
maximum 50k data
Found 68 Enz. Inhib. hit(s) with all data for entry = 50000101
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50001456(3-(2-{2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-pro...)
Affinity DataKi:  0.665nMAssay Description:Inhibition of [3H]- ]DSLET binding to delta receptor from rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50001468((S)-3-((S)-2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-phen...)
Affinity DataKi:  1.40nMAssay Description:Inhibition of [3H]- ]DSLET binding to opioid receptor delta from rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50000518(3-(2-{2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-pro...)
Affinity DataKi:  2.13nMAssay Description:Inhibition of [3H]- ]DSLET binding to delta receptor from rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50001465((S)-2-[(S)-2-(2-{2-[(S)-2-Amino-3-(4-hydroxy-pheny...)
Affinity DataKi:  2.5nMAssay Description:Inhibition of [3H]- ]DSLET binding to opioid receptor delta from rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50001463(14-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2...)
Affinity DataKi:  3.70nMAssay Description:Inhibition of [3H]- ]DSLET binding to delta receptor from rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50001462(3-[(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylam...)
Affinity DataKi:  5nMAssay Description:Inhibition of [3H]- ]DSLET binding to Opioid receptor delta 1 from rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50001459(3-[(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylam...)
Affinity DataKi:  6.5nMAssay Description:Inhibition of [3H]- ]DSLET binding to Opioid receptor delta 1 from rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50001458(3-[2-({2-[2-Amino-3-(4-hydroxy-phenyl)-propionyl]-...)
Affinity DataKi:  6.5nMAssay Description:Inhibition of [3H]- ]DSLET binding to Opioid receptor delta 1 from rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50001459(3-[(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylam...)
Affinity DataKi:  6.52nMAssay Description:Inhibition of [3H]- ]DSLET binding to opioid receptor delta from rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50001466(3-[2-(2-{2-[2-({2-[2-Amino-3-(4-hydroxy-phenyl)-pr...)
Affinity DataKi:  8.30nMAssay Description:Inhibition of [3H]- ]DSLET binding to Opioid receptor delta 1 from rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50001465((S)-2-[(S)-2-(2-{2-[(S)-2-Amino-3-(4-hydroxy-pheny...)
Affinity DataKi:  9.40nMAssay Description:Inhibition of [3H]- ]DAMGO binding to opioid receptor mu from rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50001467(12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2...)
Affinity DataKi:  10nMAssay Description:Inhibition of [3H]- ]DAMGO binding to mu receptor from rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50001463(14-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2...)
Affinity DataKi:  18nMAssay Description:Inhibition of [3H]- ]DAMGO binding to mu receptor from rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50001464(3-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylami...)
Affinity DataKi:  67nMAssay Description:Inhibition of [3H]- ]DSLET binding to Opioid receptor delta 1 from rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50001456(3-(2-{2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-pro...)
Affinity DataKi:  117nMAssay Description:Inhibition of [3H]- ]DAMGO binding to mu receptor from rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50000518(3-(2-{2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-pro...)
Affinity DataKi:  143nMAssay Description:Inhibition of [3H]- ]DAMGO binding to mu receptor from rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50001462(3-[(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylam...)
Affinity DataKi:  207nMAssay Description:Inhibition of [3H]- ]DAMGO binding to Opioid receptor mu 1 from rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50001461(CHEMBL338466 | {23-[2-Amino-3-(4-hydroxy-phenyl)-p...)
Affinity DataKi:  248nMAssay Description:Inhibition of [3H]- ]DSLET binding to delta receptor from rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50001468((S)-3-((S)-2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-phen...)
Affinity DataKi:  262nMAssay Description:Inhibition of [3H]- ]DAMGO binding to opioid receptor mu from rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50000518(3-(2-{2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-pro...)
Affinity DataKi:  290nMAssay Description:Inhibition of [3H]- ]DSLET binding to delta receptor from rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50001469(15-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylam...)
Affinity DataKi:  338nMAssay Description:Inhibition of [3H]- ]DAMGO binding to mu receptor from rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50000518(3-(2-{2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-pro...)
Affinity DataKi:  415nMAssay Description:Inhibition of [3H]- ]DAMGO binding to mu receptor from rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50001469(15-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylam...)
Affinity DataKi:  562nMAssay Description:Inhibition of [3H]- ]DSLET binding to delta receptor from rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50001459(3-[(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylam...)
Affinity DataKi:  671nMAssay Description:Inhibition of [3H]- ]DAMGO binding to Opioid receptor mu 1 from rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50001459(3-[(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylam...)
Affinity DataKi:  671nMAssay Description:Inhibition of [3H]- ]DAMGO binding to Opioid receptor mu 1 from rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50001457(17-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylam...)
Affinity DataKi:  724nMAssay Description:Inhibition of [3H]- ]DSLET binding to delta receptor from rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50001461(CHEMBL338466 | {23-[2-Amino-3-(4-hydroxy-phenyl)-p...)
Affinity DataKi:  891nMAssay Description:Inhibition of [3H]- ]DAMGO binding to mu receptor from rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50001457(17-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylam...)
Affinity DataKi:  955nMAssay Description:Inhibition of [3H]- ]DAMGO binding to mu receptor from rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50001467(12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2...)
Affinity DataKi:  2.22E+3nMAssay Description:Inhibition of [3H]- ]DSLET binding to delta receptor from rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50001466(3-[2-(2-{2-[2-({2-[2-Amino-3-(4-hydroxy-phenyl)-pr...)
Affinity DataKi:  4.15E+3nMAssay Description:Inhibition of [3H]- ]DAMGO binding to Opioid receptor mu 1 from rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50001460(3-[(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylam...)
Affinity DataKi:  4.96E+3nMAssay Description:Inhibition of [3H]- ]DSLET binding to delta receptor from rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50001464(3-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylami...)
Affinity DataKi:  8.65E+3nMAssay Description:Inhibition of [3H]- ]DAMGO binding to Opioid receptor mu 1 from rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50001458(3-[2-({2-[2-Amino-3-(4-hydroxy-phenyl)-propionyl]-...)
Affinity DataKi:  9.23E+3nMAssay Description:Inhibition of [3H]- ]DAMGO binding to Opioid receptor mu 1 from rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50001460(3-[(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylam...)
Affinity DataKi:  1.52E+4nMAssay Description:Inhibition of [3H]- ]DAMGO binding to Opioid receptor mu 1 from rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50001462(3-[(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylam...)
Affinity DataIC50:  0.0803nMAssay Description:Inhibition of electrically evoked contractions in mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50001459(3-[(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylam...)
Affinity DataIC50:  0.115nMAssay Description:Inhibition of electrically evoked contractions in mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50001468((S)-3-((S)-2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-phen...)
Affinity DataIC50:  0.147nMAssay Description:Inhibition of electrically evoked contractions in mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50001459(3-[(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylam...)
Affinity DataIC50:  0.163nMAssay Description:Inhibition of [3H]- ]DAMGO binding to Opioid receptor mu 1 from rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50001463(14-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2...)
Affinity DataIC50:  0.467nMAssay Description:Inhibition of electrically evoked contractions in mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50000518(3-(2-{2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-pro...)
Affinity DataIC50:  0.695nMAssay Description:Inhibition of [3H]- ]DSLET binding to opioid receptor delta from rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50001456(3-(2-{2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-pro...)
Affinity DataIC50:  0.712nMAssay Description:Inhibition of electrically evoked contractions in mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50001465((S)-2-[(S)-2-(2-{2-[(S)-2-Amino-3-(4-hydroxy-pheny...)
Affinity DataIC50:  11nMAssay Description:Inhibition of electrically evoked contractions in mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50001461(CHEMBL338466 | {23-[2-Amino-3-(4-hydroxy-phenyl)-p...)
Affinity DataIC50:  17nMAssay Description:Inhibition of electrically evoked contractions in mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50001458(3-[2-({2-[2-Amino-3-(4-hydroxy-phenyl)-propionyl]-...)
Affinity DataIC50:  23nMAssay Description:Inhibition of electrically evoked contractions in mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50001467(12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2...)
Affinity DataIC50:  36nMAssay Description:Inhibition of electrically evoked contractions in Guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50001464(3-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylami...)
Affinity DataIC50:  43nMAssay Description:Inhibition of electrically evoked contractions in mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50001469(15-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylam...)
Affinity DataIC50:  91nMAssay Description:Inhibition of electrically evoked contractions in mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50000518(3-(2-{2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-pro...)
Affinity DataIC50:  98.3nMAssay Description:Inhibition of electrically evoked contractions in mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50001463(14-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2...)
Affinity DataIC50:  102nMAssay Description:Inhibition of electrically evoked contractions in Guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50001456(3-(2-{2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-pro...)
Affinity DataIC50:  241nMAssay Description:Inhibition of electrically evoked contractions in Guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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