Compile Data Set for Download or QSAR
maximum 50k data
Found 54 Enz. Inhib. hit(s) with all data for entry = 50036064
TargetSubstance-P receptor(GUINEA PIG)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001603(2-(1-{2-[2-(5-Amino-pentanoylamino)-3-phenyl-propi...)
Affinity DataEC50:  307nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001607(1-{2-[2-(5-Amino-pentanoylamino)-3-phenyl-propiony...)
Affinity DataEC50:  92nMAssay Description:In vitro agonistic activity against tachykinin receptor 2 of rat colon muscularis mucosae.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001594(CHEMBL335054 | N-(1-{1-[1-({[1-(1-Carbamoyl-3-meth...)
Affinity DataEC50:  61nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001602(2-(1-{2-[2-(5-Amino-pentanoylamino)-3-phenyl-propi...)
Affinity DataEC50:  3.73E+3nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001606(2-(2-{2-[2-(5-Amino-pentanoylamino)-3-phenyl-propi...)
Affinity DataEC50:  86nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001595(1-{2-[2-(5-Amino-pentanoylamino)-3-phenyl-propiony...)
Affinity DataEC50:  13nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001607(1-{2-[2-(5-Amino-pentanoylamino)-3-phenyl-propiony...)
Affinity DataEC50:  830nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001604(2-(2-{2-[2-(5-Amino-pentanoylamino)-3-phenyl-propi...)
Affinity DataEC50:  38nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001600(CHEMBL267712 | N-{1-[1-(1-Benzyl-2-{5-[1-(1-carbam...)
Affinity DataEC50:  1.03E+3nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001447(CHEMBL217406 | His-Lys-Thr-Asp-Ser-Phe-Val-Gly-Leu...)
Affinity DataEC50:  14nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001596(3-(2-Acetylamino-6-amino-hexanoylamino)-N-{1-[1-(1...)
Affinity DataEC50:  44nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001598(2-(1-{2-[2-(5-Amino-pentanoylamino)-3-phenyl-propi...)
Affinity DataEC50:  5.23E+3nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001592(CHEMBL131923 | N-{1-[1-(1-{5-[1-(1-Carbamoyl-3-met...)
Affinity DataEC50:  1.13E+3nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001599(2-(1-{2-[2-(5-Amino-pentanoylamino)-3-phenyl-propi...)
Affinity DataEC50:  545nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50079412((NKB)Asp-Met-His-Asp-Phe-Phe-Val-Gly-Leu-Met-NH2 |...)
Affinity DataEC50:  68nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataEC50:  5.60nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001601(2-(3-{2-[2-(5-Amino-pentanoylamino)-3-phenyl-propi...)
Affinity DataEC50:  86nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001605(2-(1-{2-[2-(5-Amino-pentanoylamino)-3-phenyl-propi...)
Affinity DataEC50:  3.77E+4nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001597(CHEMBL134481 | N-(1-{1-[1-({[1-(1-Carbamoyl-3-meth...)
Affinity DataEC50:  45nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001592(CHEMBL131923 | N-{1-[1-(1-{5-[1-(1-Carbamoyl-3-met...)
Affinity DataEC50:  59nMAssay Description:In vitro agonistic activity against tachykinin receptor 2 of rat colon muscularis mucosae.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001593(CHEMBL131872 | N-{1-[1-(1-{1-[1-(1-Carbamoyl-3-met...)
Affinity DataEC50:  1.18E+3nMAssay Description:In vitro agonistic activity against tachykinin receptor 3 of everted rat protal vein.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001594(CHEMBL335054 | N-(1-{1-[1-({[1-(1-Carbamoyl-3-meth...)
Affinity DataEC50:  870nMAssay Description:In vitro agonistic activity against tachykinin receptor 3 of everted rat protal vein.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001595(1-{2-[2-(5-Amino-pentanoylamino)-3-phenyl-propiony...)
Affinity DataEC50:  1.30E+4nMAssay Description:In vitro agonistic activity against tachykinin receptor 2 of rat colon muscularis mucosae.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001596(3-(2-Acetylamino-6-amino-hexanoylamino)-N-{1-[1-(1...)
Affinity DataEC50:  1.30nMAssay Description:In vitro agonistic activity against tachykinin receptor 2 of rat colon muscularis mucosae.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001597(CHEMBL134481 | N-(1-{1-[1-({[1-(1-Carbamoyl-3-meth...)
Affinity DataEC50:  33nMAssay Description:In vitro agonistic activity against tachykinin receptor 2 of rat colon muscularis mucosae.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001599(2-(1-{2-[2-(5-Amino-pentanoylamino)-3-phenyl-propi...)
Affinity DataEC50: >1.80E+4nMAssay Description:In vitro agonistic activity against tachykinin receptor 3 of everted rat protal vein.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001592(CHEMBL131923 | N-{1-[1-(1-{5-[1-(1-Carbamoyl-3-met...)
Affinity DataEC50:  2.72E+3nMAssay Description:In vitro agonistic activity against tachykinin receptor 3 of everted rat protal vein.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001594(CHEMBL335054 | N-(1-{1-[1-({[1-(1-Carbamoyl-3-meth...)
Affinity DataEC50:  3nMAssay Description:In vitro agonistic activity against tachykinin receptor 2 of rat colon muscularis mucosae.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001600(CHEMBL267712 | N-{1-[1-(1-Benzyl-2-{5-[1-(1-carbam...)
Affinity DataEC50:  45nMAssay Description:In vitro agonistic activity against tachykinin receptor 2 of rat colon muscularis mucosae.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001595(1-{2-[2-(5-Amino-pentanoylamino)-3-phenyl-propiony...)
Affinity DataEC50: >1.00E+4nMAssay Description:In vitro agonistic activity against tachykinin receptor 3 of everted rat protal vein.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001601(2-(3-{2-[2-(5-Amino-pentanoylamino)-3-phenyl-propi...)
Affinity DataEC50:  62nMAssay Description:In vitro agonistic activity against tachykinin receptor 2 of rat colon muscularis mucosae.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001598(2-(1-{2-[2-(5-Amino-pentanoylamino)-3-phenyl-propi...)
Affinity DataEC50:  2.10E+3nMAssay Description:In vitro agonistic activity against tachykinin receptor 2 of rat colon muscularis mucosae.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001598(2-(1-{2-[2-(5-Amino-pentanoylamino)-3-phenyl-propi...)
Affinity DataEC50: >4.70E+4nMAssay Description:In vitro agonistic activity against tachykinin receptor 3 of everted rat protal vein.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001602(2-(1-{2-[2-(5-Amino-pentanoylamino)-3-phenyl-propi...)
Affinity DataEC50:  566nMAssay Description:In vitro agonistic activity against tachykinin receptor 2 of rat colon muscularis mucosae.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataEC50:  167nMAssay Description:In vitro agonistic activity against tachykinin receptor 2 of rat colon muscularis mucosae.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001605(2-(1-{2-[2-(5-Amino-pentanoylamino)-3-phenyl-propi...)
Affinity DataEC50: >8.22E+3nMAssay Description:In vitro agonistic activity against tachykinin receptor 3 of everted rat protal vein.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50079412((NKB)Asp-Met-His-Asp-Phe-Phe-Val-Gly-Leu-Met-NH2 |...)
Affinity DataEC50:  6.30nMAssay Description:In vitro agonistic activity against tachykinin receptor 3 of everted rat protal vein.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001604(2-(2-{2-[2-(5-Amino-pentanoylamino)-3-phenyl-propi...)
Affinity DataEC50:  1.13E+4nMAssay Description:In vitro agonistic activity against tachykinin receptor 3 of everted rat protal vein.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001603(2-(1-{2-[2-(5-Amino-pentanoylamino)-3-phenyl-propi...)
Affinity DataEC50:  1.39E+3nMAssay Description:In vitro agonistic activity against tachykinin receptor 2 of rat colon muscularis mucosae.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001447(CHEMBL217406 | His-Lys-Thr-Asp-Ser-Phe-Val-Gly-Leu...)
Affinity DataEC50:  1.70nMAssay Description:In vitro agonistic activity against tachykinin receptor 2 of rat colon muscularis mucosae.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001597(CHEMBL134481 | N-(1-{1-[1-({[1-(1-Carbamoyl-3-meth...)
Affinity DataEC50:  857nMAssay Description:In vitro agonistic activity against tachykinin receptor 3 of everted rat protal vein.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001593(CHEMBL131872 | N-{1-[1-(1-{1-[1-(1-Carbamoyl-3-met...)
Affinity DataEC50:  3.70nMAssay Description:In vitro agonistic activity against tachykinin receptor 2 of rat colon muscularis mucosae.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001606(2-(2-{2-[2-(5-Amino-pentanoylamino)-3-phenyl-propi...)
Affinity DataEC50:  94nMAssay Description:In vitro agonistic activity against tachykinin receptor 2 of rat colon muscularis mucosae.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001599(2-(1-{2-[2-(5-Amino-pentanoylamino)-3-phenyl-propi...)
Affinity DataEC50:  15nMAssay Description:In vitro agonistic activity against tachykinin receptor 2 of rat colon muscularis mucosae.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001600(CHEMBL267712 | N-{1-[1-(1-Benzyl-2-{5-[1-(1-carbam...)
Affinity DataEC50:  2.63E+3nMAssay Description:In vitro agonistic activity against tachykinin receptor 3 of everted rat protal vein.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001605(2-(1-{2-[2-(5-Amino-pentanoylamino)-3-phenyl-propi...)
Affinity DataEC50:  1.19E+3nMAssay Description:In vitro agonistic activity against tachykinin receptor 2 of rat colon muscularis mucosae.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001447(CHEMBL217406 | His-Lys-Thr-Asp-Ser-Phe-Val-Gly-Leu...)
Affinity DataEC50:  563nMAssay Description:In vitro agonistic activity against tachykinin receptor 3 of everted rat protal vein.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001604(2-(2-{2-[2-(5-Amino-pentanoylamino)-3-phenyl-propi...)
Affinity DataEC50:  1.19E+3nMAssay Description:In vitro agonistic activity against tachykinin receptor 2 of rat colon muscularis mucosae.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001602(2-(1-{2-[2-(5-Amino-pentanoylamino)-3-phenyl-propi...)
Affinity DataEC50: >3.00E+4nMAssay Description:In vitro agonistic activity against tachykinin receptor 3 of everted rat protal vein.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataEC50:  7.50E+3nMAssay Description:In vitro agonistic activity against tachykinin receptor 3 of everted rat protal vein.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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