Compile Data Set for Download or QSAR
maximum 50k data
Found 147 Enz. Inhib. hit(s) with all data for entry = 50030580
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM15131(5-indazolyl pyridine 3 | 5-{5-[(2S)-2-amino-3-(1H-...)
Affinity DataIC50:  0.160nMAssay Description:Inhibition of AktMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50298443(5-(5-((S)-2-amino-3-(1H-indol-3-yl)propoxy)pyridin...)
Affinity DataIC50:  0.170nMAssay Description:Inhibition of AktMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM16532((2S)-1-(1H-indol-3-yl)-3-{[5-(3-methyl-1H-pyrazolo...)
Affinity DataIC50:  0.340nMAssay Description:Inhibition of AktMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM16534((3Z)-5-(5-{[(2S)-2-amino-3-phenylpropyl]oxy}pyridi...)
Affinity DataIC50:  0.600nMAssay Description:Inhibition of AktMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50298445(5-(5-((S)-2-amino-3-(1H-indol-3-yl)propoxy)pyridin...)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of AktMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50298451((S)-1-(6-ethyl-5-(isoquinolin-6-yl)pyridin-3-yloxy...)
Affinity DataIC50:  0.800nMAssay Description:Inhibition of AktMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50298444(5-(5-((S)-2-amino-3-(1H-indol-3-yl)propoxy)pyridin...)
Affinity DataIC50:  0.900nMAssay Description:Inhibition of AktMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM16784(5-{5-[(2S)-2-amino-3-(1H-indol-3-yl)propoxy]pyridi...)
Affinity DataIC50:  1nMAssay Description:Inhibition of AktMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50298457((S)-1-(5-(3-ethyl-1H-indazol-5-yl)pyridin-3-yloxy)...)
Affinity DataIC50:  1.15nMAssay Description:Inhibition of AktMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50298464((S)-1-(5-(3-(1H-pyrrol-2-yl)-1H-indazol-5-yl)pyrid...)
Affinity DataIC50:  1.20nMAssay Description:Inhibition of AktMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50298461((S)-1-(1H-indol-3-yl)-3-(5-(3-(thiophen-2-yl)-1H-i...)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of AktMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50298433(5-(5-((S)-2-amino-3-phenylpropoxy)pyridin-3-yl)-3-...)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of AktMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50298438(5-(5-((S)-2-amino-3-(1H-indol-3-yl)propoxy)pyridin...)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of AktMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM16783(5-{5-[(2S)-2-amino-3-(1H-indol-3-yl)propoxy]pyridi...)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of AktMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM16938(5-{5-[(2S)-2-amino-3-(1H-indol-3-yl)propoxy]pyridi...)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of AktMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM16957(6-{5-[(2S)-2-amino-3-(1H-indol-3-yl)propoxy]-2-(fu...)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of AktMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM16785(5-{5-[(2S)-2-amino-3-(1H-indol-3-yl)propoxy]pyridi...)
Affinity DataIC50:  1.80nMAssay Description:Inhibition of AktMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM16954(6-{5-[(2S)-2-amino-3-(1H-indol-3-yl)propoxy]-2-chl...)
Affinity DataIC50:  1.80nMAssay Description:Inhibition of AktMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM15067((2S)-1-(1H-indol-3-yl)-3-(5-isoquinolin-6-ylpyridi...)
Affinity DataIC50:  2nMAssay Description:Inhibition of AktMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM16956(6-{5-[(2S)-2-amino-3-(1H-indol-3-yl)propoxy]-2-eth...)
Affinity DataIC50:  2nMAssay Description:Inhibition of AktMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50298479((S)-1-(4-fluoro-3-methylphenyl)-3-(5-(3-methyl-1H-...)
Affinity DataIC50:  2.5nMAssay Description:Inhibition of AktMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50298462((S)-1-(5-(3-cyclopropyl-1H-indazol-5-yl)pyridin-3-...)
Affinity DataIC50:  2.60nMAssay Description:Inhibition of AktMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50298458((S)-5-(5-(2-amino-3-(1H-indol-3-yl)propoxy)pyridin...)
Affinity DataIC50:  2.90nMAssay Description:Inhibition of AktMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM16923(5-{5-[(2S)-2-amino-3-(1H-indol-3-yl)propoxy]pyridi...)
Affinity DataIC50:  3.20nMAssay Description:Inhibition of AktMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50298434(5-(5-((S)-2-amino-3-(1H-indol-3-yl)propoxy)pyridin...)
Affinity DataIC50:  3.30nMAssay Description:Inhibition of AktMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM16978(6-{5-[(2S)-2-amino-3-(1H-indol-3-yl)propoxy]pyridi...)
Affinity DataIC50:  3.40nMAssay Description:Inhibition of AktMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM16968(6-{5-[(2S)-2-amino-3-(1H-indol-3-yl)propoxy]pyridi...)
Affinity DataIC50:  3.5nMAssay Description:Inhibition of AktMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50298460((S)-1-(1H-indol-3-yl)-3-(5-(3-phenyl-1H-indazol-5-...)
Affinity DataIC50:  3.90nMAssay Description:Inhibition of AktMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50298478((S)-1-(5-fluoro-2-methylphenyl)-3-(5-(3-methyl-1H-...)
Affinity DataIC50:  3.90nMAssay Description:Inhibition of AktMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM16934(5-{5-[(2S)-2-amino-3-(1H-indol-3-yl)propoxy]pyridi...)
Affinity DataIC50:  4nMAssay Description:Inhibition of AktMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM16930(6-(5-{[(2S)-2-amino-3-(1H-indol-3-yl)propyl]oxy}py...)
Affinity DataIC50:  4.30nMAssay Description:Inhibition of AktMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM16955(5-[(2S)-2-amino-3-(1H-indol-3-yl)propoxy]-3-(isoqu...)
Affinity DataIC50:  4.60nMAssay Description:Inhibition of AktMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50298477((S)-1-(4-bromophenyl)-3-(5-(3-methyl-1H-pyrazolo[3...)
Affinity DataIC50:  5nMAssay Description:Inhibition of AktMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM16925(5-{5-[(2S)-2-amino-3-(1H-indol-3-yl)propoxy]pyridi...)
Affinity DataIC50:  5.40nMAssay Description:Inhibition of AktMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50298435(5-(5-((S)-2-amino-3-(1H-indol-3-yl)propoxy)pyridin...)
Affinity DataIC50:  5.90nMAssay Description:Inhibition of AktMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50298480((S)-1-(4-fluoro-2-methylphenyl)-3-(5-(3-methyl-1H-...)
Affinity DataIC50:  6nMAssay Description:Inhibition of AktMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM16795(3-[(2S)-2-amino-3-phenylpropoxy]-5-[3-(furan-2-yl)...)
Affinity DataIC50:  6.10nMAssay Description:Inhibition of AktMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50298472((S)-1-(5-(3-methyl-1H-pyrazolo[3,4-c]pyridin-5-yl)...)
Affinity DataIC50:  6.80nMAssay Description:Inhibition of AktMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM16788(5-{5-[(2S)-2-amino-3-(1H-indol-3-yl)propoxy]pyridi...)
Affinity DataIC50:  7.10nMAssay Description:Inhibition of AktMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50298441(5-(5-((S)-2-amino-3-(1H-indol-3-yl)propoxy)pyridin...)
Affinity DataIC50:  7.20nMAssay Description:Inhibition of AktMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM16924(5-{5-[(2S)-2-amino-3-(1H-indol-3-yl)propoxy]pyridi...)
Affinity DataIC50:  7.40nMAssay Description:Inhibition of AktMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50298439(5-(5-((S)-2-amino-3-(1H-indol-3-yl)propoxy)pyridin...)
Affinity DataIC50:  8.20nMAssay Description:Inhibition of AktMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50298467((S)-1-(3-fluorophenyl)-3-(5-(3-methyl-1H-pyrazolo[...)
Affinity DataIC50:  8.40nMAssay Description:Inhibition of AktMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50298463((S)-1-(1H-indol-3-yl)-3-(5-(3-(thiazol-2-yl)-1H-in...)
Affinity DataIC50:  9.80nMAssay Description:Inhibition of AktMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50298446(5-(5-((S)-2-amino-3-(1H-indol-3-yl)propoxy)pyridin...)
Affinity DataIC50:  10nMAssay Description:Inhibition of AktMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50298437(5-(5-((S)-2-amino-3-(1H-indol-3-yl)propoxy)pyridin...)
Affinity DataIC50:  10.3nMAssay Description:Inhibition of AktMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50298436(5-(5-((S)-2-amino-3-(1H-indol-3-yl)propoxy)pyridin...)
Affinity DataIC50:  10.4nMAssay Description:Inhibition of AktMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50298476((S)-1-(5-(3-methyl-1H-pyrazolo[3,4-c]pyridin-5-yl)...)
Affinity DataIC50:  12nMAssay Description:Inhibition of AktMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM16960(6-{5-[(2S)-2-amino-3-(1H-indol-3-yl)propoxy]-6-chl...)
Affinity DataIC50:  12nMAssay Description:Inhibition of AktMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM16794(3-[(2S)-2-amino-3-phenylpropoxy]-5-{3-ethenyl-1H-p...)
Affinity DataIC50:  13nMAssay Description:Inhibition of AktMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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