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Found 54 Enz. Inhib. hit(s) with all data for entry = 50048392
TargetD(4) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213965(CHEMBL21168)
Affinity DataKi:  5nMAssay Description:Binding affinity at cloned human Dopamine receptor D4 expressed in HEK 293 cells, using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetD(4) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50068367(CHEMBL283353 | N-{2-[4-(4-Chloro-phenyl)-piperazin...)
Affinity DataKi:  7.90nMAssay Description:Binding affinity at cloned human Dopamine receptor D4 expressed in HEK 293 cells, using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetD(4) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213866(CHEMBL20655)
Affinity DataKi:  7.90nMAssay Description:Binding affinity at cloned human Dopamine receptor D4 expressed in HEK 293 cells, using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetD(4) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213865(CHEMBL20725)
Affinity DataKi:  7.90nMAssay Description:Binding affinity at cloned human Dopamine receptor D4 expressed in HEK 293 cells, using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetD(4) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213859(CHEMBL20367)
Affinity DataKi:  10nMAssay Description:Binding affinity at cloned human Dopamine receptor D4 expressed in HEK 293 cells, using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetD(4) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213847(CHEMBL20493)
Affinity DataKi:  13nMAssay Description:Binding affinity at cloned human Dopamine receptor D4 expressed in HEK 293 cells, using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetD(4) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213862(CHEMBL20444)
Affinity DataKi:  13nMAssay Description:Binding affinity at cloned human Dopamine receptor D4 expressed in HEK 293 cells, using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetD(4) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50007185(CHEMBL21008 | N-{4-[4-(2-Methoxy-phenyl)-piperazin...)
Affinity DataKi:  13nMAssay Description:Binding affinity at cloned human Dopamine receptor D4 expressed in HEK 293 cells, using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetD(4) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213846(CHEMBL20251)
Affinity DataKi:  16nMAssay Description:Binding affinity at cloned human Dopamine receptor D4 expressed in HEK 293 cells, using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetD(4) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213856(CHEMBL21011)
Affinity DataKi:  16nMAssay Description:Binding affinity at cloned human Dopamine receptor D4 expressed in HEK 293 cells, using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetD(4) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213967(CHEMBL21119)
Affinity DataKi:  20nMAssay Description:Binding affinity at cloned human Dopamine receptor D4 expressed in HEK 293 cells, using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetD(2) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50007185(CHEMBL21008 | N-{4-[4-(2-Methoxy-phenyl)-piperazin...)
Affinity DataKi:  20nMAssay Description:Binding affinity at cloned human Dopamine receptor D2 expressed in CHO cells, using [125I]iodosulpiride as radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetD(4) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213853(CHEMBL282008)
Affinity DataKi:  25nMAssay Description:Binding affinity at cloned human Dopamine receptor D4 expressed in HEK 293 cells, using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetD(4) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213848(CHEMBL20996)
Affinity DataKi:  32nMAssay Description:Binding affinity at cloned human Dopamine receptor D4 expressed in HEK 293 cells, using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetD(4) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213857(CHEMBL277669)
Affinity DataKi:  32nMAssay Description:Binding affinity at cloned human Dopamine receptor D4 expressed in HEK 293 cells, using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetD(4) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213852(CHEMBL21059)
Affinity DataKi:  50nMAssay Description:Binding affinity at cloned human Dopamine receptor D4 expressed in HEK 293 cells, using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetD(4) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213855(CHEMBL20854)
Affinity DataKi:  63nMAssay Description:Binding affinity at cloned human Dopamine receptor D4 expressed in HEK 293 cells, using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetD(4) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213860(CHEMBL20204)
Affinity DataKi:  63nMAssay Description:Binding affinity at cloned human Dopamine receptor D4 expressed in HEK 293 cells, using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetD(2) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213864(CHEMBL283142)
Affinity DataKi:  63nMAssay Description:Binding affinity at cloned human Dopamine receptor D2 expressed in CHO cells, using [125I]iodosulpiride as radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetD(4) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213864(CHEMBL283142)
Affinity DataKi:  79nMAssay Description:Binding affinity at cloned human Dopamine receptor D4 expressed in HEK 293 cells, using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetD(4) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213966(CHEMBL20729)
Affinity DataKi:  100nMAssay Description:Binding affinity at cloned human Dopamine receptor D4 expressed in HEK 293 cells, using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetD(4) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213964(CHEMBL20114)
Affinity DataKi:  126nMAssay Description:Binding affinity at cloned human Dopamine receptor D4 expressed in HEK 293 cells, using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetD(4) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213861(CHEMBL277937)
Affinity DataKi:  126nMAssay Description:Binding affinity at cloned human Dopamine receptor D4 expressed in HEK 293 cells, using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetD(4) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213851(CHEMBL278288)
Affinity DataKi:  126nMAssay Description:Binding affinity at cloned human Dopamine receptor D4 expressed in HEK 293 cells, using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetD(2) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213846(CHEMBL20251)
Affinity DataKi:  158nMAssay Description:Binding affinity at cloned human Dopamine receptor D2 expressed in CHO cells, using [125I]iodosulpiride as radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetD(4) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213858(CHEMBL21205)
Affinity DataKi:  158nMAssay Description:Binding affinity at cloned human Dopamine receptor D4 expressed in HEK 293 cells, using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetD(4) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213850(CHEMBL423287)
Affinity DataKi:  200nMAssay Description:Binding affinity at cloned human Dopamine receptor D4 expressed in HEK 293 cells, using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetD(2) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213966(CHEMBL20729)
Affinity DataKi:  251nMAssay Description:Binding affinity at cloned human Dopamine receptor D2 expressed in CHO cells, using [125I]iodosulpiride as radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetD(4) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213849(CHEMBL21035)
Affinity DataKi:  316nMAssay Description:Binding affinity at cloned human Dopamine receptor D4 expressed in HEK 293 cells, using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetD(4) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213854(CHEMBL20819)
Affinity DataKi:  316nMAssay Description:Binding affinity at cloned human Dopamine receptor D4 expressed in HEK 293 cells, using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetD(2) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213851(CHEMBL278288)
Affinity DataKi:  398nMAssay Description:Binding affinity at cloned human Dopamine receptor D2 expressed in CHO cells, using [125I]iodosulpiride as radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetD(2) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213860(CHEMBL20204)
Affinity DataKi:  398nMAssay Description:Binding affinity at cloned human Dopamine receptor D2 expressed in CHO cells, using [125I]iodosulpiride as radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetD(2) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213965(CHEMBL21168)
Affinity DataKi:  398nMAssay Description:Binding affinity at cloned human Dopamine receptor D2 expressed in CHO cells, using [125I]iodosulpiride as radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetD(2) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213858(CHEMBL21205)
Affinity DataKi:  398nMAssay Description:Binding affinity at cloned human Dopamine receptor D2 expressed in CHO cells, using [125I]iodosulpiride as radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetD(2) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213967(CHEMBL21119)
Affinity DataKi:  631nMAssay Description:Binding affinity at cloned human Dopamine receptor D2 expressed in CHO cells, using [125I]iodosulpiride as radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetD(2) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213849(CHEMBL21035)
Affinity DataKi:  794nMAssay Description:Binding affinity at cloned human Dopamine receptor D2 expressed in CHO cells, using [125I]iodosulpiride as radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetD(2) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213866(CHEMBL20655)
Affinity DataKi:  794nMAssay Description:Binding affinity at cloned human Dopamine receptor D2 expressed in CHO cells, using [125I]iodosulpiride as radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetD(2) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213859(CHEMBL20367)
Affinity DataKi:  1.00E+3nMAssay Description:Binding affinity at cloned human Dopamine receptor D2 expressed in CHO cells, using [125I]iodosulpiride as radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetD(2) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213856(CHEMBL21011)
Affinity DataKi:  1.00E+3nMAssay Description:Binding affinity at cloned human Dopamine receptor D2 expressed in CHO cells, using [125I]iodosulpiride as radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetD(4) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213863(CHEMBL21252)
Affinity DataKi:  1.26E+3nMAssay Description:Binding affinity at cloned human Dopamine receptor D4 expressed in HEK 293 cells, using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetD(2) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213857(CHEMBL277669)
Affinity DataKi:  1.59E+3nMAssay Description:Binding affinity at cloned human Dopamine receptor D2 expressed in CHO cells, using [125I]iodosulpiride as radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetD(2) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213855(CHEMBL20854)
Affinity DataKi:  1.59E+3nMAssay Description:Binding affinity at cloned human Dopamine receptor D2 expressed in CHO cells, using [125I]iodosulpiride as radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetD(2) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213848(CHEMBL20996)
Affinity DataKi:  1.59E+3nMAssay Description:Binding affinity at cloned human Dopamine receptor D2 expressed in CHO cells, using [125I]iodosulpiride as radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetD(2) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213863(CHEMBL21252)
Affinity DataKi:  1.59E+3nMAssay Description:Binding affinity at cloned human Dopamine receptor D2 expressed in CHO cells, using [125I]iodosulpiride as radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetD(2) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213862(CHEMBL20444)
Affinity DataKi:  1.59E+3nMAssay Description:Binding affinity at cloned human Dopamine receptor D2 expressed in CHO cells, using [125I]iodosulpiride as radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetD(2) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213964(CHEMBL20114)
Affinity DataKi:  2.00E+3nMAssay Description:Binding affinity at cloned human Dopamine receptor D2 expressed in CHO cells, using [125I]iodosulpiride as radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetD(2) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213861(CHEMBL277937)
Affinity DataKi:  2.00E+3nMAssay Description:Binding affinity at cloned human Dopamine receptor D2 expressed in CHO cells, using [125I]iodosulpiride as radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetD(2) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213853(CHEMBL282008)
Affinity DataKi:  2.51E+3nMAssay Description:Binding affinity at cloned human Dopamine receptor D2 expressed in CHO cells, using [125I]iodosulpiride as radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetD(2) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213865(CHEMBL20725)
Affinity DataKi:  2.51E+3nMAssay Description:Binding affinity at cloned human Dopamine receptor D2 expressed in CHO cells, using [125I]iodosulpiride as radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetD(2) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213847(CHEMBL20493)
Affinity DataKi:  2.51E+3nMAssay Description:Binding affinity at cloned human Dopamine receptor D2 expressed in CHO cells, using [125I]iodosulpiride as radioligandMore data for this Ligand-Target Pair
In DepthDetails
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